Assignee
ARENA PHARM INC
US·153 granted patents·127 pending applications·1,831 citations·filing 1998–2025
Top patents by PatentIndex Score
280 records- 0197US11091435B2Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3, 4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(compound1) for use in S1P1 receptor-associated disordersARENA PHARM INC·Filed 2020·Granted Aug 17, 2021·11 cites·15 claims
- 0297US10676435B2Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(Compound 1) for use in SIPI receptor-associated disordersARENA PHARM INC·Filed 2019·Granted Jun 9, 2020·12 cites·25 claims
- 0397US9556149B2Processes for the preparation of pyrazole derivatives useful as modulators of the 5-HT2A serotonin receptorARENA PHARM INC·Filed 2014·Granted Jan 31, 2017·16 cites·21 claims
- 0497US6953787B25HT2C receptor modulatorsARENA PHARM INC·Filed 2003·Granted Oct 11, 2005·79 cites·77 claims
- 0597US6140509ANon-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereofARENA PHARM INC·Filed 1999·Granted Oct 31, 2000·180 cites·1 claims
- 0696US11884626B2Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(Compound1) for use in S1P1 receptor-associated disordersARENA PHARM INC·Filed 2021·Granted Jan 30, 2024·3 cites·16 claims
- 0796US11771695B2Cannabinoid receptor modulatorsARENA PHARM INC·Filed 2021·Granted Oct 3, 2023·4 cites·11 claims
- 0896US7977329B25HT2C receptor modulatorsARENA PHARM INC·Filed 2006·Granted Jul 12, 2011·33 cites·18 claims
- 0996US7884101B23-phenyl-pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related theretoARENA PHARM INC·Filed 2006·Granted Feb 8, 2011·42 cites·2 claims
- 1096US6555339B1Non-endogenous, constitutively activated human protein-coupled receptorsARENA PHARM INC·Filed 1998·Granted Apr 29, 2003·161 cites·2 claims
- 1196US6150393ASmall molecule modulators of non-endogenous, constitutively activated human serotonin receptorsARENA PHARM INC·Filed 1999·Granted Nov 21, 2000·136 cites·12 claims
- 1295US11426377B2Method of treating conditions related to the PGI2 receptorARENA PHARM INC·Filed 2021·Granted Aug 30, 2022·5 cites·22 claims
- 1395US11149292B2Processes for the preparation of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[B]indol-3-yl)acetic acid and salts thereofARENA PHARM INC·Filed 2016·Granted Oct 19, 2021·8 cites·21 claims
- 1495US11000500B2Method of treating conditions related to the PGI2 receptorARENA PHARM INC·Filed 2020·Granted May 11, 2021·7 cites·23 claims
- 1595US10479797B2Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of disorders related theretoARENA PHARM INC·Filed 2019·Granted Nov 19, 2019·9 cites·30 claims
- 1695US9732039B2Pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related theretoARENA PHARM INC·Filed 2015·Granted Aug 15, 2017·17 cites·13 claims
- 1795US7108991B2Human orphan G protein-coupled receptorsARENA PHARM INC·Filed 2003·Granted Sep 19, 2006·38 cites·11 claims
- 1894US11560369B2Crystalline forms and processes for the preparation of cannabinoid receptor modulatorsARENA PHARM INC·Filed 2021·Granted Jan 24, 2023·2 cites·20 claims
- 1994US7838525B2Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related theretoARENA PHARM INC·Filed 2006·Granted Nov 23, 2010·39 cites·69 claims
- 2094US7368539B2Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereofARENA PHARM INC·Filed 2004·Granted May 6, 2008·29 cites·1 claims
- 2194US6846919B2Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereofARENA PHARM INC·Filed 2002·Granted Jan 25, 2005·29 cites·1 claims
- 2294US6107324A5-HT2A receptor inverse agonistsARENA PHARM INC·Filed 1999·Granted Aug 22, 2000·179 cites·7 claims
- 2393US10981895B2Crystalline forms and processes for the preparation of cannabinoid receptor modulatorsARENA PHARM INC·Filed 2018·Granted Apr 20, 2021·4 cites·16 claims
- 2493US10301262B2Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(Compund1) for use in SIPI receptor-associated disordersARENA PHARM INC·Filed 2016·Granted May 28, 2019·11 cites·50 claims
- 2593US10183930B2Crystalline forms and processes for the preparation of cannabinoid receptor modulatorsARENA PHARM INC·Filed 2016·Granted Jan 22, 2019·10 cites·11 claims
- 2693US9447041B2Processes for the preparation of (R)-2-(7-4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[B]indol-3-yl)acetic acid and salts thereofARENA PHARM INC·Filed 2015·Granted Sep 20, 2016·12 cites·22 claims
- 2793US9273035B2Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related theretoARENA PHARM INC·Filed 2014·Granted Mar 1, 2016·15 cites·26 claims
- 2893US9126932B2Substituted 1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid derivatives useful in the treatment of autoimmune and inflammatory disordersARENA PHARM INC·Filed 2013·Granted Sep 8, 2015·17 cites·61 claims
- 2993US7514422B25HT2c receptor modulatorsARENA PHARM INC·Filed 2004·Granted Apr 7, 2009·36 cites·54 claims
- 3093US7132426B2Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related theretoARENA PHARM INC·Filed 2004·Granted Nov 7, 2006·56 cites·57 claims
- 3192US11826337B2Method of treating conditions related to the PGI2 receptorARENA PHARM INC·Filed 2022·Granted Nov 28, 2023·1 cites·22 claims
- 3292US11214548B2Cannabinoid receptor modulatorsARENA PHARM INC·Filed 2019·Granted Jan 4, 2022·3 cites·8 claims
- 3392US10668033B2Modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related theretoARENA PHARM INC·Filed 2017·Granted Jun 2, 2020·4 cites·32 claims
- 3492US10632134B2Cannabinoid receptor modulatorsARENA PHARM INC·Filed 2017·Granted Apr 28, 2020·5 cites·16 claims
- 3592US9522133B2Substituted 1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid derivatives useful in the treatment of autoimmune and inflammatory disordersARENA PHARM INC·Filed 2015·Granted Dec 20, 2016·9 cites·42 claims
- 3692US9353064B2Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related theretoARENA PHARM INC·Filed 2015·Granted May 31, 2016·9 cites·51 claims
- 3792US9175320B2Processes for the preparation of (R)-2-(7-4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[B]indol-3-yl)acetic acid and salts thereofARENA PHARM INC·Filed 2014·Granted Nov 3, 2015·15 cites·42 claims
- 3892US6420541B1Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereofARENA PHARM INC·Filed 2000·Granted Jul 16, 2002·40 cites·1 claims
- 3991US10927123B2Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of disorders related theretoARENA PHARM INC·Filed 2020·Granted Feb 23, 2021·2 cites·6 claims
- 4091US10688076B2Method of treating conditions related to the PGI2 receptorARENA PHARM INC·Filed 2019·Granted Jun 23, 2020·7 cites·17 claims
- 4191US10662200B2Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of disorders related theretoARENA PHARM INC·Filed 2019·Granted May 26, 2020·3 cites·24 claims
- 4291US10537546B2Method of treating conditions related to the PGI2 receptorARENA PHARM INC·Filed 2015·Granted Jan 21, 2020·9 cites·17 claims
- 4391US10059691B2Processes for the preparation of pyrazole derivatives useful as modulators of the 5-HT2A serotonin receptorARENA PHARM INC·Filed 2017·Granted Aug 28, 2018·4 cites·3 claims
- 4491US9867822B2Cannabinoid receptor modulatorsARENA PHARM INC·Filed 2016·Granted Jan 16, 2018·7 cites·18 claims
- 4591US9492447B2Cannabinoid receptor modulatorsARENA PHARM INC·Filed 2015·Granted Nov 15, 2016·9 cites·20 claims
- 4691US9328107B2Primary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related theretoARENA PHARM INC·Filed 2014·Granted May 3, 2016·12 cites·34 claims
- 4791USRE45336EPrimary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related theretoARENA PHARM INC·Filed 2007·Granted Jan 13, 2015·12 cites·22 claims
- 4891US7470699B2Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related theretoARENA PHARM INC·Filed 2004·Granted Dec 30, 2008·41 cites·57 claims
- 4990US12378198B2Crystalline l-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(compound1) for use in SIPI receptor-associated disordersARENA PHARM INC·Filed 2023·Granted Aug 5, 2025·0 cites·40 claims
- 5090US9221755B2Ethers, secondary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related theretoARENA PHARM INC·Filed 2014·Granted Dec 29, 2015·11 cites·30 claims
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