Assignee
ARQULE INC
US·71 granted patents·13 pending applications·833 citations·filing 1993–2025
Top patents by PatentIndex Score
84 records- 0196USD369415SSample holderARQULE INC·Filed 1994·Granted Apr 30, 1996·62 cites·1 claims
- 0295US9630968B1Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereofARQULE INC·Filed 2015·Granted Apr 25, 2017·17 cites·6 claims
- 0393US10093632B2Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amineARQULE INC·Filed 2017·Granted Oct 9, 2018·5 cites·20 claims
- 0493US5712171AMethod of generating a plurality of chemical compounds in a spatially arranged arrayARQULE INC·Filed 1995·Granted Jan 27, 1998·149 cites·29 claims
- 0591US8357694B2Substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compoundsARQULE INC·Filed 2009·Granted Jan 22, 2013·12 cites·39 claims
- 0690US10245263B2Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereofARQULE INC·Filed 2017·Granted Apr 2, 2019·4 cites·4 claims
- 0790US7713969B2Compositions and methods for treatment of cancerARQULE INC·Filed 2006·Granted May 11, 2010·15 cites·13 claims
- 0890US7501430B2RAF inhibitors and their usesARQULE INC·Filed 2007·Granted Mar 10, 2009·18 cites·10 claims
- 0989US9981921B2Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compoundsARQULE INC·Filed 2016·Granted May 29, 2018·3 cites·39 claims
- 1089US7812051B2Pharmaceutical compositions of β-lapachone and β-lapachone analogs with improved tumor targeting potentialARQULE INC·Filed 2005·Granted Oct 12, 2010·6 cites·2 claims
- 1188US7960134B1Kinase inhibition models and their usesARQULE INC·Filed 2008·Granted Jun 14, 2011·11 cites·2 claims
- 1288US7960158B1Kinase inhibition models and their usesARQULE INC·Filed 2010·Granted Jun 14, 2011·11 cites·4 claims
- 1388US7166622B2Substituted phenylsulfonamide inhibitors of beta amyloid productionARQULE INC·Filed 2003·Granted Jan 23, 2007·26 cites·17 claims
- 1487US9834519B2Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amineARQULE INC·Filed 2016·Granted Dec 5, 2017·3 cites·15 claims
- 1587US5736412AMethod of generating a plurality of chemical compounds in a spatially arranged arrayARQULE INC·Filed 1996·Granted Apr 7, 1998·79 cites·40 claims
- 1686US2025339437A1Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereofARQULE INC·Filed 2025·Application pending·0 cites
- 1785US5807754ACombinatorial synthesis and high-throughput screening of a Rev-inhibiting arylidenediamide arrayARQULE INC·Filed 1995·Granted Sep 15, 1998·74 cites·9 claims
- 1885US5766481AMethod for rapid purification, analysis and characterizations of collections of chemical compoundsARQULE INC·Filed 1997·Granted Jun 16, 1998·86 cites·19 claims
- 1983US11020400B2Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereofARQULE INC·Filed 2019·Granted Jun 1, 2021·1 cites·15 claims
- 2082US10933065B2Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereofARQULE INC·Filed 2019·Granted Mar 2, 2021·1 cites·12 claims
- 2180US10717710B2Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compoundsARQULE INC·Filed 2019·Granted Jul 21, 2020·1 cites·37 claims
- 2280US10227311B2Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compoundsARQULE INC·Filed 2018·Granted Mar 12, 2019·1 cites·22 claims
- 2380US8377927B2Compositions and methods for treatment of cancerARQULE INC·Filed 2010·Granted Feb 19, 2013·4 cites·18 claims
- 2480US7074824B2Pharmaceutical compositions containing beta-lapachone, or derivatives or analogs thereof, and methods of using sameARQULE INC·Filed 2002·Granted Jul 11, 2006·9 cites·34 claims
- 2579US8962619B2Substituted imidazopyridinyl-aminopyridine compoundsARQULE INC·Filed 2013·Granted Feb 24, 2015·4 cites·6 claims
- 2678US7790765B2Hydroxy sulfonate of quinone compounds and their usesARQULE INC·Filed 2008·Granted Sep 7, 2010·7 cites·18 claims
- 2777US11020398B2Amino-pyrrolopyrimidinone compounds and methods of use thereofARQULE INC·Filed 2017·Granted Jun 1, 2021·2 cites·38 claims
- 2876US8754078B2Compositions and methods for treatment of cancerARQULE INC·Filed 2013·Granted Jun 17, 2014·2 cites·29 claims
- 2976US6962944B2Pharmaceutical compositions containing beta-lapachone, or derivatives or analogs thereof, and methods of using sameARQULE INC·Filed 2001·Granted Nov 8, 2005·10 cites·34 claims
- 3075US6452050B1Synthesis and use of α-ketoamide derivatives and arraysARQULE INC·Filed 2000·Granted Sep 17, 2002·7 cites·11 claims
- 3173US2021145837A1Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereofARQULE INC·Filed 2021·Application pending·0 cites
- 3272US5705585AAminimide-containing molecules and materials as molecular recognition agentsARQULE INC·Filed 1993·Granted Jan 6, 1998·25 cites·8 claims
- 3371US11279679B2Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[f]isoquinolin-2-amineARQULE INC·Filed 2019·Granted Mar 22, 2022·0 cites·44 claims
- 3471US9447088B2Compositions and methods for treatment of cancerARQULE INC·Filed 2014·Granted Sep 20, 2016·1 cites·17 claims
- 3571US7649013B2Methods of protecting against radiation injuryARQULE INC·Filed 2004·Granted Jan 19, 2010·5 cites·20 claims
- 3671US5962736ALogically ordered arrays of compounds and methods of making and using the sameARQULE INC·Filed 1998·Granted Oct 5, 1999·30 cites·2 claims
- 3770US8349827B2Substituted dipyrido-pyrimido-diazepine and benzo-pyrido-pyrimido compoundsARQULE INC·Filed 2010·Granted Jan 8, 2013·1 cites·19 claims
- 3870US6143931ASynthesis and use of α-ketoamide derivatives and arraysARQULE INC·Filed 1998·Granted Nov 7, 2000·12 cites·24 claims
- 3969US10766868B2Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[f]isoquinolin-2-amineARQULE INC·Filed 2019·Granted Sep 8, 2020·0 cites·17 claims
- 4069US6358750B1Spiro[pyrrolidine-2,3′-oxindole] compounds and method of useARQULE INC·Filed 2000·Granted Mar 19, 2002·4 cites·13 claims
- 4165US9499540B2Purified pyrroloquinolinyl-pyrrolidine-2,5-dione compositions and methods for preparing and using sameARQULE INC·Filed 2014·Granted Nov 22, 2016·0 cites·5 claims
- 4265US7902192B2Inhibitors of P38 and methods of using the sameARQULE INC·Filed 2004·Granted Mar 8, 2011·2 cites·11 claims
- 4365US6114540ASpiro[pyrrolidine-2,3'-oxindole] compounds and methods of useARQULE INC·Filed 1998·Granted Sep 5, 2000·10 cites·24 claims
- 4463US7361691B2Method of treating cancers using β-lapachone or analogs or derivatives thereofARQULE INC·Filed 2003·Granted Apr 22, 2008·0 cites·19 claims
- 4562US2003212497A1Relative rates of cytochrome p450 metabolismARQULE INC·Filed 2003·Application pending·0 cites
- 4661US8871933B2Purified pyrroloquinolinyl-pyrrolidine-2,5-dione compositions and methods for preparing and using sameARQULE INC·Filed 2013·Granted Oct 28, 2014·0 cites·14 claims
- 4761US7902354B2Lapachone compounds and methods of use thereofARQULE INC·Filed 2007·Granted Mar 8, 2011·0 cites·50 claims
- 4860US6753449B2Cleavable linker for solid phase synthesisARQULE INC·Filed 2001·Granted Jun 22, 2004·3 cites·15 claims
- 4957US10975087B2Solid forms of tetrahydropyranyl amino-pyrrolopyrimidinone compoundsARQULE INC·Filed 2019·Granted Apr 13, 2021·0 cites·9 claims
- 5057US9834556B2Process of preparing 3-(3-(4-aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-B]pyridin-2-YL)pyridin-2-amineARQULE INC·Filed 2016·Granted Dec 5, 2017·0 cites·8 claims
Showing the top 50 of 84 patent records by PatentIndex Score.
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