Assignee
PHARMACOPEIA DRUG DISCOVERY
US·31 granted patents·8 pending applications·325 citations·filing 1997–2014
Top patents by PatentIndex Score
39 records- 0194US7132445B23,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligandsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Nov 7, 2006·58 cites·82 claims
- 0291US7119200B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2004·Granted Oct 10, 2006·45 cites·13 claims
- 0388US7161003B1Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jan 9, 2007·32 cites·31 claims
- 0486US7202050B2Methods for measuring phosphatase activityPHARMACOPEIA DRUG DISCOVERY·Filed 2005·Granted Apr 10, 2007·5 cites·8 claims
- 0585US6942987B2Methods for measuring kinase activityPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted Sep 13, 2005·16 cites·8 claims
- 0685US6903131B23,4-di-substituted maleimide compounds as CXC chemokine receptor antagonistsPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted Jun 7, 2005·28 cites·21 claims
- 0785US6694197B1Single channel reformatterPHARMACOPEIA DRUG DISCOVERY·Filed 2000·Granted Feb 17, 2004·34 cites·8 claims
- 0882US7078525B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jul 18, 2006·15 cites·27 claims
- 0978US7179819B2VLA-4 inhibitor compoundsPHARMACOPEIA DRUG DISCOVERY·Filed 2004·Granted Feb 20, 2007·7 cites·24 claims
- 1077US7084271B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Aug 1, 2006·9 cites·28 claims
- 1177US6887889B2Aryl and biaryl piperdines with MCH modulatory activityPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted May 3, 2005·11 cites·27 claims
- 1276US6943161B2Pyrimidine and triazine kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted Sep 13, 2005·7 cites·30 claims
- 1376US6756378B2VLA-4 inhibitor compoundsPHARMACOPEIA DRUG DISCOVERY·Filed 2001·Granted Jun 29, 2004·6 cites·28 claims
- 1472US9062007B2Cyclic amide BACE-1 inhibitors having a benzamide substituentPHARMACOPEIA DRUG DISCOVERY·Filed 2014·Granted Jun 23, 2015·1 cites·6 claims
- 1572US7985748B2ALPHA2C adrenoreceptor agonistsPHARMACOPEIA DRUG DISCOVERY·Filed 2010·Granted Jul 26, 2011·2 cites·15 claims
- 1672US7067661B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jun 27, 2006·5 cites·21 claims
- 1770US6900213B2Bisaryl derivatives having FSH modulatory activityPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted May 31, 2005·5 cites·13 claims
- 1867US7074924B2Pyrazolopyrimidines as cyclin dependent kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted Jul 11, 2006·2 cites·28 claims
- 1966US7037916B2Pyrimidine derivatives as IL-8 receptor antagonistsPHARMACOPEIA DRUG DISCOVERY·Filed 2003·Granted May 2, 2006·3 cites·33 claims
- 2066US6887865B2N-heterocyclic derivatives as NOS inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted May 3, 2005·1 cites·8 claims
- 2163US6919347B2Bradykinin B1 receptor antagonistsPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted Jul 19, 2005·2 cites·64 claims
- 2262US7034056B2Aryl and biaryl compounds having MCH modulatory activityPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted Apr 25, 2006·1 cites·26 claims
- 2362US6806056B2Fluorescent capture assay for kinase activity employing an anti-phosphotyrosine antibody as both the capture agent and detecting agentPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted Oct 19, 2004·5 cites·9 claims
- 2461US2007054909A1VLA-4 inhibitor compoundsPHARMACOPEIA DRUG DISCOVERY·Filed 2006·Application pending·0 cites
- 2559US6627447B2Methods and apparatus for high throughput plate to plate or plate to membrane transferPHARMACOPEIA DRUG DISCOVERY·Filed 2001·Granted Sep 30, 2003·3 cites·13 claims
- 2657US6890491B1Method and apparatus for universal fluid exchangePHARMACOPEIA DRUG DISCOVERY·Filed 1997·Granted May 10, 2005·20 cites·42 claims
- 2756US7309470B2Methods and apparatus for improved fluid control utilizing a U-valve employing a bidirectional check valvePHARMACOPEIA DRUG DISCOVERY·Filed 2004·Granted Dec 18, 2007·0 cites·5 claims
- 2855US6846461B2Methods and apparatus for improved fluid control utilizing a U-valve employing a flow-interruption devicePHARMACOPEIA DRUG DISCOVERY·Filed 2001·Granted Jan 25, 2005·1 cites·18 claims
- 2954US2005277642A1Pyrimidine kinase inhibitorsPHARMACOPEIA DRUG DISCOVERY·Filed 2005·Application pending·0 cites
- 3051US7041463B2Orthologues of human receptors and methods of usePHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted May 9, 2006·0 cites·5 claims
- 3144US6642417B2Photocleavable and acid cleavable linkers for combinatorial chemistryPHARMACOPEIA DRUG DISCOVERY·Filed 2001·Granted Nov 4, 2003·0 cites·19 claims
- 3244US2009005568A1Substituted 2-aminothiazoles for treating neurodegenerative diseasesPHARMACOPEIA DRUG DISCOVERY·Filed 2006·Application pending·0 cites
- 3343US7038054B1Diazabicyclononane scaffold for combinatorial synthesisPHARMACOPEIA DRUG DISCOVERY·Filed 2002·Granted May 2, 2006·0 cites·8 claims
- 3443US2008119496A17-Substituted Purine Derivatives for ImmunosuppressionPHARMACOPEIA DRUG DISCOVERY·Filed 2006·Application pending·0 cites
- 3543US2009023723A1Purinone derivatives for treating neurodegenerative diseasesPHARMACOPEIA DRUG DISCOVERY·Filed 2006·Application pending·0 cites
- 3642US2007225304A1Aminopurine derivatives for treating neurodegenerative diseasesPHARMACOPEIA DRUG DISCOVERY·Filed 2006·Application pending·0 cites
- 3741US2008312215A1Substituted [1,4]-diazepanes as CXCR3 antagonists and their use in the treatment of inflammatory disordersPHARMACOPEIA DRUG DISCOVERY·Filed 2006·Application pending·0 cites
- 3839US2006206269A1One-dimensional QSAR modelsPHARMACOPEIA DRUG DISCOVERY·Filed 2005·Application pending·0 cites
- 3933US6790965B1Combinatorial dihydrobenzopyran libraryPHARMACOPEIA DRUG DISCOVERY·Filed 1999·Granted Sep 14, 2004·1 cites·5 claims
Counts cover granted patents and pending applications in the PatentIndex corpus. How scoring works →