Assignee
SYNTEX LLC
US97 patents
Top patents by PatentIndex Score
US6784166B2Aug 31, 2004
4′-substituted nucleoside derivatives as inhibitors of HCV RNA replication.
SYNTEX LLC251 citations98
US6844466B2Jan 18, 2005
Alkyl urea retinoid agonists
SYNTEX LLC23 citations92
US6696566B2Feb 24, 2004
6-substituted pyrido-pyrimidines
SYNTEX LLC27 citations92
US6506749B2Jan 14, 2003
7-oxo-pyridopyrimidines (I)
SYNTEX LLC17 citations92
US6479507B2Nov 12, 2002
p38 MAP kinase inhibitors
SYNTEX LLC37 citations92
US6417186B1Jul 9, 2002
Substituted-phenyl ketone derivatives as IP antagonists
SYNTEX LLC22 citations92
US6376506B1Apr 23, 2002
Sulfamide-metalloprotease inhibitors
SYNTEX LLC47 citations92
US6323223B1Nov 27, 2001
Cyclic amine derivatives- CCR-3 receptor antagonists
SYNTEX LLC18 citations92
US6316464B1Nov 13, 2001
P38 MAP kinase inhibitors
SYNTEX LLC26 citations92
US6300350B1Oct 9, 2001
Treatment of emphysema using RARy selective retinoid agonists
SYNTEX LLC25 citations92
US6197976B1Mar 6, 2001
Preparation of ketorolac
SYNTEX LLC24 citations92
US6967093B2Nov 22, 2005
Glycosyl sulfotransferase-3
SYNTEX LLC20 citations91
US6518276B2Feb 11, 2003
7-oxo-pyridopyrimidines (II)
SYNTEX LLC27 citations91
US6479490B2Nov 12, 2002
3-indolyl-4-phenyl-1H-pyrrole-2,5-dione derivatives as inhibitors of glycogen synthase kinase-3β
SYNTEX LLC27 citations91
US6849657B2Feb 1, 2005
2-pyrrolidone derivatives as prostanoid agonists
SYNTEX LLC21 citations90
US6693098B2Feb 17, 2004
Carboxylic acid derivatives as IP antagonists
SYNTEX LLC27 citations90
US6451804B1Sep 17, 2002
Heteroalkylamino-substituted bicyclic nitrogen heterocycles
SYNTEX LLC35 citations90
US6319920B1Nov 20, 2001
2-arylethyl-(piperidin-4-ylmethyl)amine derivatives
SYNTEX LLC29 citations90
US6787535B2Sep 7, 2004
Indole derivatives with 5HT6 receptor affinity
SYNTEX LLC29 citations89
US6479259B1Nov 12, 2002
Human peripheral nerve, tetrodotoxin-resistant sodium channel α-subunit polypeptide
SYNTEX LLC15 citations89
US6790848B2Sep 14, 2004
4-piperazinylindole derivatives with 5-HT6 receptor affinity
SYNTEX LLC25 citations87
US6339107B1Jan 15, 2002
Methods for treatment of Emphysema using 13-cis retinoic acid
SYNTEX LLC17 citations87
US6224911B1May 1, 2001
Process for the preparation of enteric coated pharmaceutical dosage forms
SYNTEX LLC24 citations85
US6838472B2Jan 4, 2005
Substituted urea retinoid agonists
SYNTEX LLC19 citations84
US6984637B2Jan 10, 2006
Cyclic amine derivatives-CCR-3 receptor antagonists
SYNTEX LLC12 citations83
US6903086B2Jun 7, 2005
Alkoxycarbonylamino benzoic acid or alkoxycarbonylamino tetrazolyl phenyl derivatives as IP antagonists
SYNTEX LLC16 citations83
US6635658B2Oct 21, 2003
Amino-tetralin derivatives as muscarinic receptor antagonists
SYNTEX LLC14 citations83
US6444696B1Sep 3, 2002
Pyrazole derivatives P38 MAP kinase inhibitors
SYNTEX LLC17 citations83
US6339087B1Jan 15, 2002
Cyclic amine derivatives-CCR-3 receptor antagonists
SYNTEX LLC16 citations83
US7186841B2Mar 6, 2007
Antiinflammation agents
SYNTEX LLC11 citations82
US6649377B1Nov 18, 2003
Human aggrecanase and nucleic acid compositions encoding the same
SYNTEX LLC23 citations82
US6355641B1Mar 12, 2002
Oxazolone derivatives and uses thereof
SYNTEX LLC14 citations82
US6900220B2May 31, 2005
Quinazolone derivatives as alpha 1A/B adrenergic receptor antagonists
SYNTEX LLC14 citations81
US6900336B2May 31, 2005
8-aza-11-deoxy prostaglandin analogues
SYNTEX LLC12 citations78
US6559138B1May 6, 2003
3-Desoxy-vitamin D3 analog esters
SYNTEX LLC7 citations74
US6376500B2Apr 23, 2002
Substituted 2-(4-piperidyl)-4(3H)-quinazolinones and 2-(4-piperidyl)-4(3H)-azaquinazolinones
SYNTEX LLC7 citations74
US6309858B1Oct 30, 2001
T-type calcium channel variants; compositions thereof; and uses
SYNTEX LLC12 citations74
US6258819B1Jul 10, 2001
Substituted 2(4-piperidyl)-4(3H)-quinazolinones and 2-(4-piperidyl)-4(3H)-azaquinazolinones
SYNTEX LLC7 citations74
US6861423B2Mar 1, 2005
Methods of treating p38 kinase-mediated disorders with pyrido[2,3-d]pyrimidin-7-one compounds
SYNTEX LLC11 citations73
US6777418B2Aug 17, 2004
Retinoid compounds (I)
SYNTEX LLC12 citations73
US6630485B2Oct 7, 2003
p38 map kinase inhibitors
SYNTEX LLC6 citations73
US6500822B2Dec 31, 2002
Benzocycloalkylenylamine derivatives as muscarinic receptor antagonists
SYNTEX LLC7 citations73
US6376527B1Apr 23, 2002
Pyrazole derivatives-p38 map kinase inhibitors
SYNTEX LLC13 citations73
US6316466B1Nov 13, 2001
Pyrazole derivatives P-38 MAP kinase inhibitors
SYNTEX LLC14 citations73
US6770650B2Aug 3, 2004
Cyclic amine derivatives-CCR-3 receptor antagonists
SYNTEX LLC10 citations72
US6753427B2Jun 22, 2004
7-oxo-pyridopyrimidines (II)
SYNTEX LLC9 citations72
US6667301B2Dec 23, 2003
Heterocyclylalkylamines as muscarinic receptor antagonists
SYNTEX LLC5 citations72
US6642241B1Nov 4, 2003
Alkylamino-substituted bicyclic nitrogen heterocycles
SYNTEX LLC9 citations72
US6492353B1Dec 10, 2002
1,3-dihydroxy-20,20-cycloalkyl-vitamin D3analogs
SYNTEX LLC9 citations72
US7056903B2Jun 6, 2006
Carboxylic acid derivatives as IP antagonists
SYNTEX LLC8 citations71
Showing the top 50 of 97 patents by PatentIndex Score.