Assignee
XENOPORT INC
US117 patents
Top patents by PatentIndex Score
US7227028B2Jun 5, 2007
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
XENOPORT INC93 citations98
US7101912B2Sep 5, 2006
Carbidopa prodrugs and derivatives, and compositions and uses thereof
XENOPORT INC98 citations98
US6818787B2Nov 16, 2004
Prodrugs of GABA analogs, compositions and uses thereof
XENOPORT INC99 citations98
US7265096B2Sep 4, 2007
Gemcitabine prodrugs, pharmaceutical compositions and uses thereof
XENOPORT INC62 citations97
US7563821B2Jul 21, 2009
Levodopa prodrug mesylate, compositions thereof, and uses thereof
XENOPORT INC30 citations96
US7351740B2Apr 1, 2008
Acyloxyalkyl carbamate prodrugs of tranexamic acid, methods of synthesis and use
XENOPORT INC43 citations96
US7232924B2Jun 19, 2007
Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
XENOPORT INC53 citations96
US6777239B2Aug 17, 2004
Epitope-captured antibody display
XENOPORT INC36 citations96
US7109239B2Sep 19, 2006
Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
XENOPORT INC61 citations95
US7186855B2Mar 6, 2007
Prodrugs of GABA analogs, compositions and uses thereof
XENOPORT INC51 citations94
US6972341B2Dec 6, 2005
Prodrugs of GABA analogs, compositions and uses thereof
XENOPORT INC59 citations94
US8344028B2Jan 1, 2013
Gamma-amino-butyric acid derivatives as GABAB receptor ligands
XENOPORT INC43 citations93
US7601706B2Oct 13, 2009
Bile-acid conjugates providing for sustained systemic concentration of drugs
XENOPORT INC17 citations93
US7241807B2Jul 10, 2007
Prodrugs of propofol, compositions and uses thereof
XENOPORT INC16 citations93
US7192720B2Mar 20, 2007
Array-based epitope-captured antibody display
XENOPORT INC15 citations93
US7144877B2Dec 5, 2006
Bile-acid derived compounds for enhancing oral absorption and systemic bioavailability of drugs
XENOPORT INC37 citations93
US7026351B2Apr 11, 2006
Cyclic 1-(acyloxy)-alkyl prodrugs of GABA analogs, compositions and uses thereof
XENOPORT INC17 citations93
US6992076B2Jan 31, 2006
Bile-acid derived compounds for providing sustained systemic concentrations of drugs after oral administration
XENOPORT INC21 citations93
US6984634B2Jan 10, 2006
Bile-acid conjugates for providing sustained systemic concentrations of drugs
XENOPORT INC18 citations93
US6900192B2May 31, 2005
Bile-acid conjugates for providing sustained systemic concentrations of drugs
XENOPORT INC14 citations93
US6833140B2Dec 21, 2004
Orally administered dosage forms of GABA analog prodrugs having reduced toxicity
XENOPORT INC34 citations93
US7893105B2Feb 22, 2011
Levodopa prodrug mesylate, compositions thereof, and uses thereof
XENOPORT INC29 citations92
US7829592B2Nov 9, 2010
Catechol protected levodopa diester prodrugs, compositions, and methods of use
XENOPORT INC21 citations92
US7803785B2Sep 28, 2010
Gemcitabine prodrugs, pharmaceutical compositions and uses thereof
XENOPORT INC13 citations92
US7749985B2Jul 6, 2010
Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
XENOPORT INC28 citations92
US7709527B2May 4, 2010
Levodopa dimethyl-substituted diester prodrugs compositions, and methods of use
XENOPORT INC15 citations92
US7671089B2Mar 2, 2010
Levodopa prodrugs, and compositions and uses thereof
XENOPORT INC24 citations92
US7534813B2May 19, 2009
Levodopa prodrugs, and compositions and uses thereof
XENOPORT INC33 citations92
US7511158B2Mar 31, 2009
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
XENOPORT INC29 citations92
US7423169B2Sep 9, 2008
Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
XENOPORT INC17 citations92
US7413536B1Aug 19, 2008
Substrates and screening methods for transport proteins
XENOPORT INC38 citations92
US7342131B2Mar 11, 2008
Levodopa prodrugs, and compositions and uses thereof
XENOPORT INC32 citations92
US7323585B2Jan 29, 2008
Levodopa prodrugs, and compositions and uses thereof
XENOPORT INC26 citations92
US7300956B2Nov 27, 2007
Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
XENOPORT INC25 citations92
US8952006B2Feb 10, 2015
Morpholinoalkyl fumarate compounds, pharmaceutical compositions, and methods of use
XENOPORT INC15 citations84
US7968597B2Jun 28, 2011
Levodopa prodrug mesylate, compositions thereof, and uses thereof
XENOPORT INC10 citations84
US7956212B2Jun 7, 2011
Levodopa prodrugs, and compositions and uses thereof
XENOPORT INC11 citations84
US7868043B2Jan 11, 2011
Mesophasic forms of (3S)-aminomethyl-5-methyl-hexanoic acid prodrugs and methods of use
XENOPORT INC7 citations84
US7700652B2Apr 20, 2010
Treating urinary incontinence using prodrugs of GABA analogs
XENOPORT INC13 citations84
US7662987B2Feb 16, 2010
Methods for synthesis of acyloxyalkyl compounds
XENOPORT INC13 citations84
US7592369B2Sep 22, 2009
Acyloxyalkyl carbamate prodrugs of tranexamic acid, methods of synthesis and use
XENOPORT INC10 citations84
US7462459B2Dec 9, 2008
LAT1 transporters expressed in blood brain barrier cells
XENOPORT INC14 citations84
US7230003B2Jun 12, 2007
Aromatic prodrugs of propofol, compositions and uses thereof
XENOPORT INC14 citations84
US7053076B2May 30, 2006
Bile-acid derived compounds for enhancing oral absorption and systemic bioavailability of drugs
XENOPORT INC12 citations84
US7049305B2May 23, 2006
Bile-acid conjugates providing for sustained systemic concentration of drugs
XENOPORT INC11 citations84
US9302977B2Apr 5, 2016
Method of making monomethyl fumarate
XENOPORT INC12 citations83
US8378137B2Feb 19, 2013
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
XENOPORT INC5 citations83
US7994218B2Aug 9, 2011
Simple pantoic acid ester neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use
XENOPORT INC14 citations83
US7531572B2May 12, 2009
Acyloxyalkyl carbamate prodrugs of α-amino acids, methods of synthesis and use
XENOPORT INC8 citations83
US7645792B2Jan 12, 2010
Prodrugs of propofol, compositions and uses thereof
XENOPORT INC8 citations82
Showing the top 50 of 117 patents by PatentIndex Score.