Assignee
ARIAD PHARMA INC
US·49 granted patents·28 pending applications·655 citations·filing 1994–2023
Top patents by PatentIndex Score
77 records- 0195US9493470B2Crystalline forms of 3-(imidazo[1,2-B] pyridazin-3-ylethynyl)-4-methyl-N-{4-[(4-methylpiperazin-1-yl) methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2013·Granted Nov 15, 2016·16 cites·17 claims
- 0294US9611283B1Methods for inhibiting cell proliferation in ALK-driven cancersARIAD PHARMA INC·Filed 2014·Granted Apr 4, 2017·16 cites·17 claims
- 0394US9273077B2Phosphorus derivatives as kinase inhibitorsARIAD PHARMA INC·Filed 2013·Granted Mar 1, 2016·13 cites·51 claims
- 0493US9029533B2Substituted acetylenic imidazo[1,2-A]pyridazines as kinase inhibitorsARIAD PHARMA INC·Filed 2013·Granted May 12, 2015·14 cites·17 claims
- 0593US6150527ASynthetic multimerizing agentsARIAD PHARMA INC·Filed 1997·Granted Nov 21, 2000·78 cites·51 claims
- 0692US10227342B2Heteroaryl compounds for kinase inhibitionARIAD PHARMA INC·Filed 2015·Granted Mar 12, 2019·7 cites·14 claims
- 0791US9796712B2Heteroaryl compounds for kinase inhibitionARIAD PHARMA INC·Filed 2017·Granted Oct 24, 2017·6 cites·15 claims
- 0891US9278971B2Substituted acetylenic pyrazolo[1,5-a]pyrimidines as kinase inhibitorsARIAD PHARMA INC·Filed 2014·Granted Mar 8, 2016·10 cites·11 claims
- 0991US8778942B2Substituted acetylenic imidazo[1,2-A]pyrazine compounds as kinase inhibitorsARIAD PHARMA INC·Filed 2013·Granted Jul 15, 2014·11 cites·19 claims
- 1091US6420384B2Proton pump inhibitorsARIAD PHARMA INC·Filed 2000·Granted Jul 16, 2002·32 cites·9 claims
- 1190US6878697B2Phenylamino-pyrimidines and uses thereofARIAD PHARMA INC·Filed 2002·Granted Apr 12, 2005·26 cites·68 claims
- 1290US6015709ATranscriptional activators, and compositions and uses related theretoARIAD PHARMA INC·Filed 1997·Granted Jan 18, 2000·108 cites·44 claims
- 1389US10125136B2Crystalline forms of 3-(imidazo[1,2-B] pyridazin-3-ylethynyl)-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2016·Granted Nov 13, 2018·3 cites·12 claims
- 1488US10662197B2Crystalline forms of 3-(imidazo[1,2-b)pyridazin-3-ylethynyl)-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2018·Granted May 26, 2020·4 cites·11 claims
- 1586US6713462B2Quinolinones and uses thereofARIAD PHARMA INC·Filed 2002·Granted Mar 30, 2004·16 cites·75 claims
- 1685US9834571B2Compounds for inhibiting cell proliferation in EGFR-driven cancersARIAD PHARMA INC·Filed 2016·Granted Dec 5, 2017·2 cites·16 claims
- 1785US5710129AInhibitors of SH2-mediated processesARIAD PHARMA INC·Filed 1995·Granted Jan 20, 1998·61 cites·8 claims
- 1884US9834521B2Choline kinase inhibitorsARIAD PHARMA INC·Filed 2014·Granted Dec 5, 2017·4 cites·1 claims
- 1984US6482852B2Bicyclic signal transduction inhibitors, compositions containing them & uses thereofARIAD PHARMA INC·Filed 2001·Granted Nov 19, 2002·20 cites·81 claims
- 2084US2024083902A1Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2023·Application pending·0 cites
- 2183US6573295B2Bicyclic signal transduction inhibitors, compositions containing them & uses thereofARIAD PHARMA INC·Filed 2001·Granted Jun 3, 2003·17 cites·81 claims
- 2283US6207397B1In vitro fluorescence polarization assayARIAD PHARMA INC·Filed 1997·Granted Mar 27, 2001·80 cites·11 claims
- 2380US7709020B2Implantable device comprising phosphorus-containing macrolidesARIAD PHARMA INC·Filed 2007·Granted May 4, 2010·2 cites·4 claims
- 2480US2022081440A1Substituted acetylenic pyrazolo[1,5-a]pyridine compounds as kinase inhibitorsARIAD PHARMA INC·Filed 2021·Application pending·0 cites
- 2579US11192896B2Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2021·Granted Dec 7, 2021·0 cites·18 claims
- 2678US11192895B2Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2021·Granted Dec 7, 2021·0 cites·24 claims
- 2778US11192897B2Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2021·Granted Dec 7, 2021·0 cites·23 claims
- 2877US11384086B2Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1- yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2021·Granted Jul 12, 2022·0 cites·19 claims
- 2977US11001580B2Aminothiazole compounds as c-Kit inhibitorsARIAD PHARMA INC·Filed 2017·Granted May 11, 2021·1 cites·14 claims
- 3077US2024208960A1Aminothiazole compounds as c-kit inhibitorsARIAD PHARMA INC·Filed 2023·Application pending·0 cites
- 3176US11117883B2Benzimidazole compounds as c-Kit inhibitorsARIAD PHARMA INC·Filed 2017·Granted Sep 14, 2021·1 cites·7 claims
- 3275US11180482B2Anilinopyrimidines as haematopoietic progenitor kinase 1 (HPK1) inhibitorsARIAD PHARMA INC·Filed 2017·Granted Nov 23, 2021·2 cites·12 claims
- 3375US2020231588A1Bicyclic Heteroaryl CompoundsARIAD PHARMA INC·Filed 2019·Application pending·0 cites
- 3474US11279705B2Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride saltARIAD PHARMA INC·Filed 2020·Granted Mar 22, 2022·0 cites·3 claims
- 3573US2020317705A1Phosphorous derivatives as kinase inhibitorsARIAD PHARMA INC·Filed 2019·Application pending·0 cites
- 3672US11427605B2Crystalline forms of 5-chloro-N4-[-2-(dimethylphosphoryl) phenyl]-N2-{2-methoxy-4-[4-(4-methylpiperazin-1-yl) piperidin-1-yl] phenyl} pyrimidine-2,4-diamineARIAD PHARMA INC·Filed 2020·Granted Aug 30, 2022·0 cites·8 claims
- 3771US11753404B2Aminothiazole compounds as c-Kit inhibitorsARIAD PHARMA INC·Filed 2021·Granted Sep 12, 2023·0 cites·4 claims
- 3871US7132427B2Quinazolines and uses thereofARIAD PHARMA INC·Filed 2002·Granted Nov 7, 2006·5 cites·22 claims
- 3970US6960572B2Indolinones and uses thereofARIAD PHARMA INC·Filed 2002·Granted Nov 1, 2005·6 cites·30 claims
- 4070US6706699B2Quinolines and uses thereofARIAD PHARMA INC·Filed 2002·Granted Mar 16, 2004·5 cites·44 claims
- 4169US7115589B2Purine derivativesARIAD PHARMA INC·Filed 2000·Granted Oct 3, 2006·4 cites·20 claims
- 4269US2019031656A1Substituted acetylenic pyrazolo[1,5-a]pyridine compounds as kinase inhibitorsARIAD PHARMA INC·Filed 2018·Application pending·0 cites
- 4367US6576766B1Signal transduction inhibitors, compositions containing themARIAD PHARMA INC·Filed 1998·Granted Jun 10, 2003·12 cites·73 claims
- 4467US6251620B1Three dimensional structure of a ZAP tyrosine protein kinase fragment and modeling methodsARIAD PHARMA INC·Filed 1997·Granted Jun 26, 2001·30 cites·7 claims
- 4566US10934317B2Crystalline forms of 5-chloro-N4-[-2-(dimethylphosphoryl) phenyl]-N2-{2-methoxy-4-[4-(4-methylpiperazin-1-yl) piperidin-1-yl] phenyl} pyrimidine-2,4-diamineARIAD PHARMA INC·Filed 2019·Granted Mar 2, 2021·0 cites·13 claims
- 4666US2021186994A1Pharmaceutical formulations comprising 5-Chloro-N4-[2-(dimethylphosphoryl)phenyl]-N2-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineARIAD PHARMA INC·Filed 2021·Application pending·0 cites
- 4765US2019218212A1Heteroaryl compounds for kinase inhibitionARIAD PHARMA INC·Filed 2019·Application pending·0 cites
- 4864US2022064144A1Benzimidazole compounds as c-kit inhibitorsARIAD PHARMA INC·Filed 2021·Application pending·0 cites
- 4964US2020048288A1Phosphorous derivatives as kinase inhibitorsARIAD PHARMA INC·Filed 2019·Application pending·0 cites
- 5063US9573934B2Methods and compositions for the synthesis of multimerizing agentsARIAD PHARMA INC·Filed 2015·Granted Feb 21, 2017·0 cites·20 claims
Showing the top 50 of 77 patent records by PatentIndex Score.
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