Assignee
PHARMACIA & UPJOHN SPA
IT·99 granted patents·3 pending applications·1,827 citations·filing 1987–2002
Top patents by PatentIndex Score
102 records- 0197US6335342B1Azaindole derivatives, process for their preparation, and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 2000·Granted Jan 1, 2002·149 cites·172 claims
- 0297US6218418B13(5)-amino-pyrazole derivatives, process for their preparation and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 2000·Granted Apr 17, 2001·145 cites·25 claims
- 0396US6414013B1Thiophene compounds, process for preparing the same, and pharmaceutical compositions containing the same background of the inventionPHARMACIA & UPJOHN SPA·Filed 2000·Granted Jul 2, 2002·106 cites·45 claims
- 0492US6114365AArylmethyl-carbonylamino-thiazole derivatives, process for their preparation, and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 1999·Granted Sep 5, 2000·94 cites·21 claims
- 0591US5700788AUreido derivatives of naphthalenephosphonic acidsPHARMACIA & UPJOHN SPA·Filed 1995·Granted Dec 23, 1997·106 cites·16 claims
- 0690US5856496ACombinatorial solid phase synthesis of a library of indole derivativesPHARMACIA & UPJOHN SPA·Filed 1997·Granted Jan 5, 1999·62 cites·6 claims
- 0787US6863647B22-Ureido-thiazole derivatives, process for their preparation, and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 1999·Granted Mar 8, 2005·63 cites·3 claims
- 0887US6194451B1Matrix metalloproteinase inhibitorsPHARMACIA & UPJOHN SPA·Filed 1998·Granted Feb 27, 2001·116 cites·19 claims
- 0987US5919955ACombinatorial solid phase synthesis of a library of benzofuran derivativesPHARMACIA & UPJOHN SPA·Filed 1997·Granted Jul 6, 1999·52 cites·4 claims
- 1082US6495534B2Stabilized aqueous suspensions for parenteral usePHARMACIA & UPJOHN SPA·Filed 2000·Granted Dec 17, 2002·17 cites·21 claims
- 1182US5719265APolymer-bound paclitaxel derivativesPHARMACIA & UPJOHN SPA·Filed 1995·Granted Feb 17, 1998·40 cites·1 claims
- 1280US5945454A2-(4-substituted)-benzylamino-2-methyl-propanamide derivativesPHARMACIA & UPJOHN SPA·Filed 1996·Granted Aug 31, 1999·49 cites·12 claims
- 1379US5691334APyrrolydenemethyl-derivatives and process for their preparationPHARMACIA & UPJOHN SPA·Filed 1994·Granted Nov 25, 1997·27 cites·40 claims
- 1478US7037929B12-amino-thiazole derivatives, process for their preparation, and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 1999·Granted May 2, 2006·43 cites·13 claims
- 1578US5731313AUse of anthracyclinone derivatives in amyloidosisPHARMACIA & UPJOHN SPA·Filed 1995·Granted Mar 24, 1998·18 cites·10 claims
- 1676US6387900B13(5)-ureido-pyrazole derivatives process for their preparation and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 1999·Granted May 14, 2002·41 cites·28 claims
- 1776US6284887B1Process for preparing carboxamido-4-azasteroidsPHARMACIA & UPJOHN SPA·Filed 2000·Granted Sep 4, 2001·7 cites·7 claims
- 1876US5849710ASubstituted indolylmethylene-oxindole analogues as tyrosine kinase inhibitorsPHARMACIA & UPJOHN SPA·Filed 1996·Granted Dec 15, 1998·43 cites·12 claims
- 1976US5593976ANew ureido derivatives of poly-4-amino-2-carboxy-1-methyl compoundsPHARMACIA & UPJOHN SPA·Filed 1995·Granted Jan 14, 1997·32 cites·4 claims
- 2074US6403563B1Antitumor composition containing a synergistic combination of an anthracycline derivative with a camptothecin derivatePHARMACIA & UPJOHN SPA·Filed 1999·Granted Jun 11, 2002·36 cites·10 claims
- 2174US5912183APeptide inhibitors of mitogenesis and motogenesisPHARMACIA & UPJOHN SPA·Filed 1996·Granted Jun 15, 1999·26 cites·14 claims
- 2272US6528301B1Paclitaxel production by actinomycetesPHARMACIA & UPJOHN SPA·Filed 1999·Granted Mar 4, 2003·28 cites·6 claims
- 2371US6750215B2Substituted benzoxazines as integrin antagonistsPHARMACIA & UPJOHN SPA·Filed 2001·Granted Jun 15, 2004·2 cites·19 claims
- 2471US6458768B1Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor agentsPHARMACIA & UPJOHN SPA·Filed 1999·Granted Oct 1, 2002·15 cites·7 claims
- 2571US6153642ABenzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agentsPHARMACIA & UPJOHN SPA·Filed 1997·Granted Nov 28, 2000·16 cites·10 claims
- 2670US6562562B2Procedure for partial liver resection in nonhuman primatesPHARMACIA & UPJOHN SPA·Filed 2001·Granted May 13, 2003·9 cites·8 claims
- 2770US6177408B1Distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agentsPHARMACIA & UPJOHN SPA·Filed 1997·Granted Jan 23, 2001·14 cites·6 claims
- 2870US5965563AAryl and heteroaryl purine compoundsPHARMACIA & UPJOHN SPA·Filed 1996·Granted Oct 12, 1999·27 cites·7 claims
- 2969US6096888AAnthracyclinone derivatives and their use in amyloidosisPHARMACIA & UPJOHN SPA·Filed 1999·Granted Aug 1, 2000·10 cites·6 claims
- 3069US5847127AProcess for the preparation of 2,2'-bipyrrolyl-pyrromethene (prodigiosins) derivativesPHARMACIA & UPJOHN SPA·Filed 1997·Granted Dec 8, 1998·17 cites·6 claims
- 3168US6210930B1Process for preparing doxorubicinPHARMACIA & UPJOHN SPA·Filed 1998·Granted Apr 3, 2001·15 cites·16 claims
- 3268US5856333ASubstituted camptothecin derivatives and process for their preparationPHARMACIA & UPJOHN SPA·Filed 1996·Granted Jan 5, 1999·13 cites·13 claims
- 3364US6369096B1Benzyloxy prodigiosine compoundsPHARMACIA & UPJOHN SPA·Filed 1999·Granted Apr 9, 2002·9 cites·14 claims
- 3464US5695966ADNA encoding daunorubicin 14-hyroxylase and method for preparing doxorubicinPHARMACIA & UPJOHN SPA·Filed 1995·Granted Dec 9, 1997·11 cites·18 claims
- 3564US5602141ACamptothecin derivatives and process for their preparationPHARMACIA & UPJOHN SPA·Filed 1995·Granted Feb 11, 1997·18 cites·6 claims
- 3663US5776458AAnthracycline-conjugatesPHARMACIA & UPJOHN SPA·Filed 1995·Granted Jul 7, 1998·29 cites·6 claims
- 3763US5614628AProcess for the preparation of 9-amino camptothecinPHARMACIA & UPJOHN SPA·Filed 1994·Granted Mar 25, 1997·14 cites·8 claims
- 3862US5798097AImmunogobulin conjugatesPHARMACIA & UPJOHN SPA·Filed 1995·Granted Aug 25, 1998·21 cites·12 claims
- 3960US6048896A4-phenyl-4-oxo-2-butenoic acid derivatives with kynurenine-3-hydroxylase inhibiting activityPHARMACIA & UPJOHN SPA·Filed 1996·Granted Apr 11, 2000·16 cites·7 claims
- 4060US5998615AAnthracyclinone derivativesPHARMACIA & UPJOHN SPA·Filed 1997·Granted Dec 7, 1999·13 cites·7 claims
- 4160US5912242AN-(4-substituted-benzyl)-2-aminolactam derivativesPHARMACIA & UPJOHN SPA·Filed 1996·Granted Jun 15, 1999·15 cites·9 claims
- 4259US6071947AIndolyl-pyrrolydenemethylpyrrole derivatives and process for their preparationPHARMACIA & UPJOHN SPA·Filed 1998·Granted Jun 6, 2000·16 cites·18 claims
- 4358US6794385B2Benzoxazine derivatives useful as integrin receptor antagonistsPHARMACIA & UPJOHN SPA·Filed 2001·Granted Sep 21, 2004·1 cites·27 claims
- 4457US6121449AProcess for preparing carboxamido-4-azasteroidsPHARMACIA & UPJOHN SPA·Filed 1998·Granted Sep 19, 2000·11 cites·8 claims
- 4555US6093721AAmidino-camptothecin derivativesPHARMACIA & UPJOHN SPA·Filed 1998·Granted Jul 25, 2000·5 cites·11 claims
- 4654US6482827B1Matrix metalloproteinase inhibitorsPHARMACIA & UPJOHN SPA·Filed 1998·Granted Nov 19, 2002·13 cites·18 claims
- 4752US5985887AAza-anthracyclinone derivativesPHARMACIA & UPJOHN SPA·Filed 1996·Granted Nov 16, 1999·8 cites·13 claims
- 4852US5905149ASubstituted quinolymethylen-oxindole analogues as tyrosine kinase inhibitorsPHARMACIA & UPJOHN SPA·Filed 1997·Granted May 18, 1999·5 cites·7 claims
- 4951US6323240B14-phenyl-4-oxo-butanoic acid derivatives with kynurenine-3-hydroxylase inhibiting activityPHARMACIA & UPJOHN SPA·Filed 1996·Granted Nov 27, 2001·9 cites·14 claims
- 5051US6133302A5-(3-Phenyl-3-oxo-propyl)-1H-tetrazole derivativesPHARMACIA & UPJOHN SPA·Filed 1998·Granted Oct 17, 2000·9 cites·7 claims
Showing the top 50 of 102 patent records by PatentIndex Score.
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