Inventor
PONTICELLO GERALD S
68 patents
Patents
50 patentsUS5837719ANov 17, 1998
2,5-substituted aryl pyrroles, compositions containing such compounds and methods of use
MERCK & CO INC77 citations96
US5792778AAug 11, 1998
2-substituted aryl pyrroles, compositions containing such compounds and methods of use
MERCK & CO INC63 citations96
US5633247AMay 27, 1997
Nitrogen-containing spirocycles
MERCK & CO INC73 citations96
US5215989AJun 1, 1993
Nitrogen-containing heterocyclic compounds as class III antiarrhythmic agents
MERCK & CO INC108 citations96
US5206240AApr 27, 1993
Nitrogen-containing spirocycles
MERCK & CO INC77 citations96
US5032598AJul 16, 1991
Nitrogens containing heterocyclic compounds as class III antiarrhythmic agents
MERCK & CO INC58 citations96
US4797413AJan 10, 1989
Thieno thiopyran sulfonamide derivatives, pharmaceutical compositions and use
MERCK & CO INC103 citations96
US5475109ADec 12, 1995
Dioxobutanoic acid derivatives as inhibitors of influenza endonuclease
MERCK & CO INC56 citations95
US5112824AMay 12, 1992
Benzofuran compounds as class III antiarrhythmic agents
MERCK & CO INC25 citations92
US4863922ASep 5, 1989
Substituted aromatic sulfonamides as antiglaucoma agents, compositions and use
MERCK & CO INC52 citations92
US4602093AJul 22, 1986
Novel substituted imidazoles, their preparation and use
MERCK & CO INC34 citations92
US5872138AFeb 16, 1999
Thrombin inhibitors
MERCK & CO INC47 citations91
US4677115AJun 30, 1987
Antiglaucoma thieno-thiopyran and thieno-thiepin sulfonamide derivatives, compositions, and method of use thereof
MERCK & CO INC24 citations82
US4176183ANov 27, 1979
Novel naphthyridines
MERCK & CO INC21 citations82
US4064139ADec 20, 1977
Substituted 9,10-dihydroanthracen-9,10-imines
MERCK & CO INC25 citations82
US4052508AOct 4, 1977
Heterocyclic dihydroanthracen imines
MERCK & CO INC22 citations82
US5403846AApr 4, 1995
Spirocycles
MERCK & CO INC18 citations74
US5032604AJul 16, 1991
Class III antiarrhythmic agents
MERCK & CO INC18 citations74
US4853383AAug 1, 1989
β-blocking substituted imidazoles
MERCK & CO INC18 citations74
US4735961AApr 5, 1988
Oxazoles and thiazoles containing an aminohydroxypropoxyphenyl moiety
MERCK & CO INC15 citations74
US4642311AFeb 10, 1987
β-adrenergic blocking imidazolylphenoxy propanolamines
MERCK & CO INC12 citations74
US4616017AOct 7, 1986
Aminohydroxypropoxy substituted aryl compounds
MERCK & CO INC16 citations74
US4562184ADec 31, 1985
Substituted-aminohydroxypropoxy-thiadiazoles, β-blocking compositions and use
MERCK & CO INC12 citations74
US4539318ASep 3, 1985
Tertiary aminohydroxypropoxy substituted thiadiazoles, pharmaceutical compositions and use
MERCK & CO INC10 citations74
US4294969AOct 13, 1981
Process for producing 2-bromo-3,5-disubstituted pyridines
MERCK & CO INC7 citations74
US4260609AApr 7, 1981
Di- and tri- substituted thiazoles
MERCK & CO INC10 citations74
US4259341AMar 31, 1981
Di- and tri-substituted thiazoles
MERCK & CO INC10 citations74
US4144343AMar 13, 1979
Heterocycle substituted (3-loweralkylamino-2-R1 O-propoxy)pyridines
MERCK & CO INC13 citations74
US5618830AApr 8, 1997
Dioxobutanoic acid derivatives as inhibitors of influenza endonuclease
MERCK & CO INC13 citations73
US4803286AFeb 7, 1989
Amino-2-hydroxypropyloximinoheterocycle α-blockers
MERCK & CO INC6 citations73
US4593039AJun 3, 1986
1-aryloxy-3-(substituted aminoalkylamino)-2-propanols
MERCK & CO INC8 citations73
US5441722AAug 15, 1995
Short synthesis of 5,6-dihydro-(S)-4-(ethylamino)-(S)-6-[C3 H3 ]-4[2,3-b]thiopyran-2-sulfonamide 7,7-dioxide and related non radioactive compounds
MERCK & CO INC14 citations72
US4847289AJul 11, 1989
Thiophene sulfonamide antiglaucoma agents
MERCK & CO INC13 citations71
US4820848AApr 11, 1989
Substituted aromatic sulfonamides as antiglaucoma agents
MERCK & CO INC8 citations71
US4824968AApr 25, 1989
Substituted aromatic sulfonamides as antiglaucoma agents
MERCK & CO INC7 citations66
US6350744B1Feb 26, 2002
Compounds having cytokine inhibitory activity
MERCK & CO INC2 citations63
US5439914AAug 8, 1995
Spirocycles
MERCK & CO INC5 citations63
US5334591AAug 2, 1994
Tricyclic thienothiopyran carbonic anhydrase inhibitors
MERCK & CO INC2 citations63
US5235059AAug 10, 1993
Tricyclic thienothiopyran carbonic anhydrase inhibitors
MERCK & CO INC4 citations63
US5175284ADec 29, 1992
Tricyclic thienothiopyrans as pharmaceutical intermediates
MERCK & CO INC2 citations63
US5120757AJun 9, 1992
Substituted aromatic sulfonamides as antiglaucoma agents
MERCK & CO INC5 citations63
US5091409AFeb 25, 1992
4-alkylamino-6-(C3-5 -hydrocarbyl)thieno[2,3-B]thiopyran-2-sulfonamide-7,7-dioxides
MERCK & CO INC5 citations63
US5045561ASep 3, 1991
Substituted furan sulfonamides as antiglaucoma agents
MERCK & CO INC4 citations63
US4883814ANov 28, 1989
1-aryloxy-3-(substituted alkylamino)-2-propanols and use as β-blocker
MERCK & CO INC3 citations63
US4574127AMar 4, 1986
Oxazoles and thiazoles containing an aminohydroxypropoxyphenyl moiety
MERCK & CO INC5 citations63
US4539317ASep 3, 1985
4-Substituted amino-3-[3-alkylindoloamino-2-hydroxypropoxy] thiadiazoles, compositions and pharmaceutical use
MERCK & CO INC2 citations63
US4329351AMay 11, 1982
2-Substituted propoxy-3-cyano-5-RO-pyridines and intermediates
MERCK & CO INC2 citations63
US4279913AJul 21, 1981
Polysubstituted-2-(3-loweralkylamino-2-R1 O-propoxy)pyridines
MERCK & CO INC5 citations63
US5952351ASep 14, 1999
Alpha 1a adrenergic receptor antagonists
MERCK & CO INC2 citations62
US5308863AMay 3, 1994
Substituted aromatic sulfonamides as antiglaucoma agents
MERCK & CO INC3 citations62
Showing the top 50 of 68 patents by PatentIndex Score.