Inventor
FREYNE EDDY JEAN EDGARD
BE50 patents
⚠️ This page may combine multiple inventors who share the name “FREYNE EDDY JEAN EDGARD”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
JANSSEN PHARMACEUTICA NV
26 patentsUS7514445B2Apr 7, 2009
Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors)
JANSSEN PHARMACEUTICA NV117 citations97
US7799772B2Sep 21, 2010
Pyrido-and pyrimidopyrimidine derivatives as anti-profilerative agents
JANSSEN PHARMACEUTICA NV16 citations92
US6583141B1Jun 24, 2003
4,5-dihydro-isoxazole derivatives and their pharmaceutical use
JANSSEN PHARMACEUTICA NV18 citations89
US6403805B1Jun 11, 2002
1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one derivatves
JANSSEN PHARMACEUTICA NV20 citations87
US7648975B2Jan 19, 2010
Macrocyclic quinazoline derivatives as antiproliferative agents
JANSSEN PHARMACEUTICA NV12 citations83
US7560458B2Jul 14, 2009
Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
JANSSEN PHARMACEUTICA NV9 citations83
US5994376ANov 30, 1999
1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one compounds and their use for treating allergic, atopic or inflammatory diseases
JANSSEN PHARMACEUTICA NV17 citations83
US7655642B2Feb 2, 2010
3-cyano-quinoline derivatives with antiproliferative activity
JANSSEN PHARMACEUTICA NV13 citations82
US7449465B2Nov 11, 2008
Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
JANSSEN PHARMACEUTICA NV12 citations82
US6051718AApr 18, 2000
PDE IV inhibiting 2-cyanoiminoimidazole derivatives
JANSSEN PHARMACEUTICA NV15 citations71
US5952510ASep 14, 1999
1,3-dihydro-1-(phenylalkenyl)-2H-imidazol-2-one derivatives having PDE IV and cytokine inhibiting activity
JANSSEN PHARMACEUTICA NV3 citations61
US5869515AFeb 9, 1999
1,3-dihydro-2H-imidazol-2-one compounds
JANSSEN PHARMACEUTICA NV5 citations61
US7947695B2May 24, 2011
5-membered annelated heterocyclic pyrimidines as kinase inhibitors
JANSSEN PHARMACEUTICA NV4 citations60
US7947694B2May 24, 2011
Substituted pyrazolo[3,4-D]pyrimidines as cell cycle kinase inhibitors
JANSSEN PHARMACEUTICA NV2 citations60
US6803364B1Oct 12, 2004
Il-5 inhibiting 6-azauracil derivatives
JANSSEN PHARMACEUTICA NV2 citations60
US7241763B2Jul 10, 2007
3-furanyl analogs of toxoflavine as kinase inhibitors
JANSSEN PHARMACEUTICA NV2 citations57
US10208062B2Feb 19, 2019
Macrocyclic quinazole derivatives and their use as MTKI
JANSSEN PHARMACEUTICA NV0 citations51
US9688691B2Jun 27, 2017
Macrocyclic quinazole derivatives and their use as MTKI
JANSSEN PHARMACEUTICA NV0 citations51
US9365517B2Jun 14, 2016
3-cyano-quinoline derivatives with antiproliferative activity
JANSSEN PHARMACEUTICA NV0 citations51
US9273013B2Mar 1, 2016
Quinazoline derivatives
JANSSEN PHARMACEUTICA NV0 citations51
US9040511B2May 26, 2015
3-cyano-quinoline derivatives with antiproliferative activity
JANSSEN PHARMACEUTICA NV0 citations51
US7414048B2Aug 19, 2008
4,5-dihydro-isoxazole derivatives and their pharmaceutical use
JANSSEN PHARMACEUTICA NV0 citations48
US6743792B2Jun 1, 2004
6-azauracil derivatives as IL-5 inhibitors
JANSSEN PHARMACEUTICA NV1 citations47
US6894046B2May 17, 2005
IL-5 inhibiting 6-azauracil derivatives
JANSSEN PHARMACEUTICA NV0 citations41
US6867207B2Mar 15, 2005
IL-5 inhibiting 6-azauracil derivatives
JANSSEN PHARMACEUTICA NV0 citations41
US6498158B1Dec 24, 2002
Il-5 inhibiting 6-azauracil derivatives
JANSSEN PHARMACEUTICA NV0 citations35
FREYNE EDDY JEAN EDGARD
9 patentsUS8476289B2Jul 2, 2013
Aza-bicyclohexyl substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylace
FREYNE EDDY JEAN EDGARD12 citations84
US8148388B2Apr 3, 2012
2,4 (4,6) pyrimidine derivatives
FREYNE EDDY JEAN EDGARD6 citations83
US8394786B2Mar 12, 2013
Quinazoline derivatives
FREYNE EDDY JEAN EDGARD5 citations82
US8168644B2May 1, 2012
Quinazolinone derivatives as tubulin polymerization inhibitors
FREYNE EDDY JEAN EDGARD2 citations61
US8394955B2Mar 12, 2013
2,4 (4,6) pyrimidine derivatives
FREYNE EDDY JEAN EDGARD0 citations51
US8772272B2Jul 8, 2014
Pyrido-and pyrimidopyrimidine derivatives as anti-proliferative agents
FREYNE EDDY JEAN EDGARD0 citations49
US8778920B2Jul 15, 2014
3-cyano-quinoline derivatives with antiproliferative activity
FREYNE EDDY JEAN EDGARD0 citations47
US6951857B2Oct 4, 2005
6-Azauracil derivatives as IL-5 inhibitors
FREYNE EDDY JEAN EDGARD0 citations47
US7183288B2Feb 27, 2007
Amide derivatives as glycogen synthase kinase 3-β inhibitors
FREYNE EDDY JEAN EDGARD0 citations33
ASTEX THERAPEUTICS LTD
3 patentsSAXTY GORDON
3 patentsUS8895601B2Nov 25, 2014
Pyrazolyl quinoxaline kinase inhibitors
SAXTY GORDON25 citations91
US8481531B2Jul 9, 2013
Bicyclic heterocyclyl derivatives as FGFR kinase inhibitors for therapeutic use
SAXTY GORDON9 citations82
US8722687B2May 13, 2014
Imidazo [1,2-A]pyridine derivatives as FGFR kinase inhibitors for use in therapy
SAXTY GORDON0 citations38