Inventor
COMBS ANDREW P
US117 patents
⚠️ This page may combine multiple inventors who share the name “COMBS ANDREW P”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
INCYTE CORP
41 patentsUS8741895B2Jun 3, 2014
Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors
INCYTE CORP84 citations99
US8053433B2Nov 8, 2011
Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors
INCYTE CORP107 citations99
US7335667B2Feb 26, 2008
Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-4-yl-amines as Janus kinase inhibitors
INCYTE CORP149 citations99
US9707233B2Jul 18, 2017
Heterocyclylamines as PI3K inhibitors
INCYTE CORP23 citations98
US9624241B2Apr 18, 2017
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP27 citations98
US9540368B2Jan 10, 2017
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins
INCYTE CORP35 citations98
US9434746B2Sep 6, 2016
Pyrimidinones as PI3K inhibitors
INCYTE CORP32 citations98
US9227985B2Jan 5, 2016
Tricyclic heterocycles as bet protein inhibitors
INCYTE CORP40 citations98
US9090611B2Jul 28, 2015
Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors
INCYTE CORP60 citations98
US8993605B2Mar 31, 2015
1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase
INCYTE CORP34 citations98
US8034953B2Oct 11, 2011
Modulators of indoleamine 2,3-dioxygenase and methods of using the same
INCYTE CORP45 citations98
US8835423B2Sep 16, 2014
Azepine inhibitors of janus kinases
INCYTE CORP71 citations97
US8822511B2Sep 2, 2014
1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase
INCYTE CORP24 citations96
US11059821B2Jul 13, 2021
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins
INCYTE CORP13 citations94
US10781209B2Sep 22, 2020
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins
INCYTE CORP12 citations94
US10618910B2Apr 14, 2020
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP12 citations94
US10472358B2Nov 12, 2019
1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins
INCYTE CORP19 citations94
US10464947B2Nov 5, 2019
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP17 citations94
US10227359B2Mar 12, 2019
Tricyclic heterocycles as bet protein inhibitors
INCYTE CORP20 citations94
US10138248B2Nov 27, 2018
Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-γ inhibitors
INCYTE CORP36 citations94
US10092570B2Oct 9, 2018
Heterocyclylamines as PI3K inhibitors
INCYTE CORP17 citations94
US10077277B2Sep 18, 2018
Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
INCYTE CORP22 citations94
US9957268B2May 1, 2018
1H-pyrrolo[2,3,c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins
INCYTE CORP23 citations94
US9938294B2Apr 10, 2018
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP24 citations94
US9918990B2Mar 20, 2018
Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors
INCYTE CORP23 citations94
US9850257B2Dec 26, 2017
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP22 citations94
US9834565B2Dec 5, 2017
Tricyclic heterocycles as bet protein inhibitors
INCYTE CORP23 citations94
US9737516B2Aug 22, 2017
Bicyclic heterocycles as bet protein inhibitors
INCYTE CORP25 citations94
US9730939B2Aug 15, 2017
Heterocyclylamines as PI3K inhibitors
INCYTE CORP23 citations94
US9533997B2Jan 3, 2017
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP29 citations94
US9527848B2Dec 27, 2016
N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
INCYTE CORP25 citations94
US9527864B2Dec 27, 2016
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP31 citations94
US9399640B2Jul 26, 2016
Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors
INCYTE CORP37 citations94
US9315501B2Apr 19, 2016
Bicyclic heterocycles as BET protein inhibitors
INCYTE CORP33 citations94
US9309251B2Apr 12, 2016
Bicyclic azaheterocyclobenzylamines as PI3K inhibitors
INCYTE CORP25 citations94
US9290514B2Mar 22, 2016
Tricyclic heterocycles as BET protein inhibitors
INCYTE CORP33 citations94
US10646492B2May 12, 2020
Heterocyclylamines as PI3K inhibitors
INCYTE CORP9 citations93
US10428087B2Oct 1, 2019
Pyrimidinones as PI3K inhibitors
INCYTE CORP13 citations93
US10376513B2Aug 13, 2019
Heterocyclylamines as PI3K inhibitors
INCYTE CORP12 citations93
US10034864B2Jul 31, 2018
1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase
INCYTE CORP8 citations93
US9975907B2May 22, 2018
Pyrimidinones as PI3K inhibitors
INCYTE CORP14 citations93
LI YUN-LONG
4 patentsUS9199982B2Dec 1, 2015
Heterocyclylamines as PI3K inhibitors
LI YUN-LONG52 citations98
US9096600B2Aug 4, 2015
N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
LI YUN-LONG47 citations98
US8680108B2Mar 25, 2014
Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors
LI YUN-LONG62 citations98
US9062055B2Jun 23, 2015
Fused pyrrole derivatives as PI3K inhibitors
LI YUN-LONG28 citations94
COMBS ANDREW P
3 patentsUS8088803B2Jan 3, 2012
1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase
COMBS ANDREW P64 citations99
US8759359B2Jun 24, 2014
Substituted heteroaryl fused derivatives as PI3K inhibitors
COMBS ANDREW P64 citations98
US9108984B2Aug 18, 2015
Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors
COMBS ANDREW P32 citations94
RODGERS JAMES D
1 patentARVANITIS ARGYRIOS G
1 patentShowing the top 50 of 117 patents by PatentIndex Score.