Inventor
PARUCH KAMIL
US50 patents
⚠️ This page may combine multiple inventors who share the name “PARUCH KAMIL”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SCHERING CORP
33 patentsUS6919341B2Jul 19, 2005
Imidazopyrazines as cyclin dependent kinase inhibitors
SCHERING CORP65 citations96
US7605155B2Oct 20, 2009
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
SCHERING CORP28 citations92
US7601724B2Oct 13, 2009
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
SCHERING CORP22 citations92
US7645762B2Jan 12, 2010
Substituted pyrazolo[1,5-a] pyrimidines as protein kinase inhibitors
SCHERING CORP8 citations84
US7642266B2Jan 5, 2010
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
SCHERING CORP11 citations84
US7205308B2Apr 17, 2007
Trisubstituted 7-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP12 citations84
US7196092B2Mar 27, 2007
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP15 citations84
US7776865B2Aug 17, 2010
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
SCHERING CORP9 citations83
US7563798B2Jul 21, 2009
Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
SCHERING CORP11 citations83
US7576085B2Aug 18, 2009
Imidazopyrazines as cyclin dependent kinase inhibitors
SCHERING CORP10 citations82
US7038045B2May 2, 2006
Pyrazolotriazines as kinase inhibitors
SCHERING CORP10 citations74
US6992080B2Jan 31, 2006
Imidazopyridines as cyclin dependent kinase inhibitors
SCHERING CORP7 citations74
US7468372B2Dec 23, 2008
Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP7 citations72
US7700773B2Apr 20, 2010
4-cyano, 4-amino, and 4-aminomethyl derivatives of pyrazolo[1,5-a]pyridines, pyrazolo[1,5-c]pyrimidines and 2H-indazole compounds and 5-cyano, 5-amino, and 5-aminomethyl derivatives of imidazo[1,2-a]pyridines, and imidazo[1,5-a]pyrazines as cyclin dependent kinase inhibitors
SCHERING CORP3 citations63
US7452902B2Nov 18, 2008
Imidazopyridines as cyclin dependent kinase inhibitors
SCHERING CORP2 citations63
US7186740B2Mar 6, 2007
Imidazopyrazines as cyclin dependent kinase inhibitors
SCHERING CORP7 citations63
US6969718B2Nov 29, 2005
17-β hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
SCHERING CORP2 citations63
US7557104B2Jul 7, 2009
Imidazopyrazines as protein kinase inhibitors
SCHERING CORP2 citations62
US7309705B2Dec 18, 2007
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP2 citations62
US7138396B2Nov 21, 2006
17 β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
SCHERING CORP3 citations62
US6903102B2Jun 7, 2005
17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
SCHERING CORP3 citations62
US7476681B2Jan 13, 2009
17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
SCHERING CORP1 citations52
US7470695B2Dec 30, 2008
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP0 citations52
US7432265B2Oct 7, 2008
Imidazopyrazines as cyclin dependent kinase inhibitors
SCHERING CORP0 citations52
US7354921B2Apr 8, 2008
Pyrazolotriazines as kinase inhibitors
SCHERING CORP0 citations52
US7166602B2Jan 23, 2007
Pyrazolotriazines as kinase inhibitors
SCHERING CORP1 citations52
US7074795B2Jul 11, 2006
17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
SCHERING CORP0 citations52
US7807683B2Oct 5, 2010
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP0 citations51
US7514442B2Apr 7, 2009
Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP1 citations51
US7511049B2Mar 31, 2009
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
SCHERING CORP0 citations51
US7432268B2Oct 7, 2008
17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
SCHERING CORP1 citations51
US7449488B2Nov 11, 2008
Pyrazolopyrimidines as protein kinase inhibitors
SCHERING CORP0 citations42
US7151104B2Dec 19, 2006
Pyrazolopyridines as cyclin dependent kinase inhibitors
SCHERING CORP0 citations42
PHARMACOPEIA DRUG DISCOVERY
6 patentsUS7161003B1Jan 9, 2007
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
PHARMACOPEIA DRUG DISCOVERY32 citations91
US7119200B2Oct 10, 2006
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
PHARMACOPEIA DRUG DISCOVERY45 citations91
US7078525B2Jul 18, 2006
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
PHARMACOPEIA DRUG DISCOVERY15 citations84
US7084271B2Aug 1, 2006
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
PHARMACOPEIA DRUG DISCOVERY9 citations73
US7074924B2Jul 11, 2006
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
PHARMACOPEIA DRUG DISCOVERY2 citations62
US7067661B2Jun 27, 2006
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
PHARMACOPEIA DRUG DISCOVERY5 citations61
GUZI TIMOTHY J
5 patentsUS8586576B2Nov 19, 2013
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors
GUZI TIMOTHY J15 citations91
US8580782B2Nov 12, 2013
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors
GUZI TIMOTHY J14 citations83
US8211854B2Jul 3, 2012
Methods for inhibiting protein kinases
GUZI TIMOTHY J12 citations83
US8673924B2Mar 18, 2014
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors
GUZI TIMOTHY J11 citations81
US8603998B2Dec 10, 2013
Modulators of cell cycle checkpoints and their use in combination with checkpoint kinase inhibitors
GUZI TIMOTHY J5 citations71
UNIV MASARYKOVA
5 patentsUS11584742B2Feb 21, 2023
Substituted aminothiazoles as inhibitors of nucleases
UNIV MASARYKOVA0 citations39
US11453663B2Sep 27, 2022
Substituted propanamides as inhibitors of nucleases
UNIV MASARYKOVA0 citations38
US11498920B2Nov 15, 2022
4-(1H-imidazol-5-yl)-1H-pyrrolo[2, 3-b] pyridines for use in the treatment of leukaemias, lymphomas and solid tumors
UNIV MASARYKOVA0 citations35
US9969741B2May 15, 2018
Pyrazolotriazines as inhibitors of nucleases
UNIV MASARYKOVA0 citations29
US9902733B2Feb 27, 2018
Furopyridines as inhibitors of protein kinases
UNIV MASARYKOVA0 citations28