Inventor
GIJSEN HENRICUS JACOBUS MARIA
NL39 patents
⚠️ This page may combine multiple inventors who share the name “GIJSEN HENRICUS JACOBUS MARIA”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
JANSSEN PHARMACEUTICA NV
23 patentsUS6544997B1Apr 8, 2003
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders
JANSSEN PHARMACEUTICA NV60 citations94
US9453002B2Sep 27, 2016
Substituted imidazoles as N-type calcium channel blockers
JANSSEN PHARMACEUTICA NV18 citations90
US9751886B2Sep 5, 2017
4-amino-6-phenyl-6,7-dihydro[1,2,3]triazolo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE)
JANSSEN PHARMACEUTICA NV2 citations72
US9284303B2Mar 15, 2016
Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group
JANSSEN PHARMACEUTICA NV4 citations70
US7635706B2Dec 22, 2009
5HT4-antagonistic 4-(aminomethyl)-piperidine benzamides
JANSSEN PHARMACEUTICA NV2 citations62
US7652040B2Jan 26, 2010
Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT4-antagonists
JANSSEN PHARMACEUTICA NV5 citations61
US7205410B2Apr 17, 2007
4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders
JANSSEN PHARMACEUTICA NV4 citations60
US11053248B2Jul 6, 2021
[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitors
JANSSEN PHARMACEUTICA NV0 citations59
US10947239B2Mar 16, 2021
[1,2,4]triazolo[1,5-a]pyrimidin-7-yl compound
JANSSEN PHARMACEUTICA NV0 citations55
US9834559B2Dec 5, 2017
4-Amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2H)-one derivatives as inhibitors of beta-secretase (BACE)
JANSSEN PHARMACEUTICA NV1 citations51
US10653673B2May 19, 2020
Substituted imidazoles as N-type calcium channel blockers
JANSSEN PHARMACEUTICA NV0 citations50
US9974775B2May 22, 2018
Substituted imidazoles as N-type calcium channel blockers
JANSSEN PHARMACEUTICA NV1 citations50
US9828350B2Nov 28, 2017
5,6-dihydro-2H-[1,4]oxazin-3-yl-amine derivatives useful as inhibitors of beta-secretase (BACE)
JANSSEN PHARMACEUTICA NV1 citations49
US11319321B2May 3, 2022
[1,2,4]triazolo[1,5-a]pyrimidine compounds as PDE2 inhibitors
JANSSEN PHARMACEUTICA NV0 citations48
US10106524B2Oct 23, 2018
2,3,4,5-tetrahydropyridin-6-amine and 3,4-dihydro-2H-pyrrol-5-amine compound inhibitors of beta-secretase
JANSSEN PHARMACEUTICA NV1 citations47
US10947242B2Mar 16, 2021
[1,2,4]triazolo[1,5and#8208;A]pyrimidine compounds as PDE2 inhibitors
JANSSEN PHARMACEUTICA NV0 citations46
US9580433B2Feb 28, 2017
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-A]pyrazine derivatives as inhibitors of beta-secretase (BACE)
JANSSEN PHARMACEUTICA NV0 citations41
US7638535B2Dec 29, 2009
4-(aminomethyl)-piperidine benzamides as 5HT4-antagonists
JANSSEN PHARMACEUTICA NV0 citations41
US7732464B2Jun 8, 2010
Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5HT4-antagonists
JANSSEN PHARMACEUTICA NV0 citations40
US7498347B2Mar 3, 2009
Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT4 antagonists
JANSSEN PHARMACEUTICA NV0 citations40
US10112943B2Oct 30, 2018
Substituted imidazoles as gamma secretase modulators
JANSSEN PHARMACEUTICA NV0 citations39
US10562897B2Feb 18, 2020
Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators
JANSSEN PHARMACEUTICA NV0 citations37
US10246454B2Apr 2, 2019
Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators
JANSSEN PHARMACEUTICA NV0 citations37
GIJSEN HENRICUS JACOBUS MARIA
6 patentsUS8546440B2Oct 1, 2013
Substituted bicyclic imidazole derivatives as gamma secretase modulators
GIJSEN HENRICUS JACOBUS MARIA5 citations71
US8772504B2Jul 8, 2014
Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators
GIJSEN HENRICUS JACOBUS MARIA2 citations60
US8461145B2Jun 11, 2013
Dibenzoazepine and dibenzooxazepine TRPA1 agonists
GIJSEN HENRICUS JACOBUS MARIA3 citations59
US8524757B2Sep 3, 2013
Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group
GIJSEN HENRICUS JACOBUS MARIA0 citations48
US8946426B2Feb 3, 2015
Substituted bicyclic heterocyclic compounds as gamma secretase modulators
GIJSEN HENRICUS JACOBUS MARIA0 citations39
US8193369B2Jun 5, 2012
Benzimidazole cannabinoid agonists
GIJSEN HENRICUS JACOBUS MARIA0 citations39
TRABANCO-SUÁREZ ANDRÉS AVELINO
2 patentsUS9840507B2Dec 12, 2017
5,6-dihydro-imidazo[1,2-a]pyrazin-8-ylamine derivatives useful as inhibitors of beta-secretase (BACE)
TRABANCO-SUÁREZ ANDRÉS AVELINO0 citations34
US9346811B2May 24, 2016
6,7-dihydro-pyrazolo[1,5-a]pyrazin-4-ylamine derivatives useful as inhibitors of beta-secretase (BACE)
TRABANCO-SUÁREZ ANDRÉS AVELINO0 citations34