Inventor
MACDONALD GREGOR JAMES
GB69 patents
⚠️ This page may combine multiple inventors who share the name “MACDONALD GREGOR JAMES”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
CID-NUNEZ JOSE MARIA
11 patentsUS8937060B2Jan 20, 2015
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of prevention of neurological and psychiatric disorders
CID-NUNEZ JOSE MARIA39 citations97
US8252937B2Aug 28, 2012
1,3-disubstituted 4-(aryl-X-phenyl)-1H-pyridin-2-ones
CID-NUNEZ JOSE MARIA28 citations90
US8299101B2Oct 30, 2012
1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive mGluR2-receptor modulators
CID-NUNEZ JOSE MARIA29 citations89
US8946205B2Feb 3, 2015
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
CID-NUNEZ JOSE MARIA4 citations71
US8748621B2Jun 10, 2014
1,3-disubstituted 4-(aryl-X-phenyl)-1H-pyridin-2-ones
CID-NUNEZ JOSE MARIA4 citations71
US8716480B2May 6, 2014
7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
CID-NUNEZ JOSE MARIA4 citations71
US8906939B2Dec 9, 2014
3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
CID-NUNEZ JOSE MARIA2 citations62
US9114138B2Aug 25, 2015
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyridinyl-2′-ones
CID-NUNEZ JOSE MARIA2 citations61
US9067891B2Jun 30, 2015
1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of mGluR2-receptors
CID-NUNEZ JOSE MARIA2 citations61
US8841323B2Sep 23, 2014
1, 4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of MGLUR2-receptors
CID-NUNEZ JOSE MARIA2 citations58
US8691813B2Apr 8, 2014
Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
CID-NUNEZ JOSE MARIA1 citations52
GLAXO GROUP LTD
9 patentsUS7538121B2May 26, 2009
Vanilloid receptor modulators
GLAXO GROUP LTD59 citations96
US7262188B2Aug 28, 2007
Phenyl sulfone derivatives and their use in the treatment of CNS disorders
GLAXO GROUP LTD19 citations93
US7601837B2Oct 13, 2009
Quinoline derivatives and their use as 5-HT6 ligands
GLAXO GROUP LTD15 citations92
US7452888B2Nov 18, 2008
Quinoline derivatives and their use as 5-ht6 ligands
GLAXO GROUP LTD23 citations92
US7977337B2Jul 12, 2011
Quinoline derivatives and their use as 5-HT6 ligands
GLAXO GROUP LTD11 citations91
US7799774B2Sep 21, 2010
Quinoline derivatives and their use as 5-HT6 ligands
GLAXO GROUP LTD11 citations91
US7964602B2Jun 21, 2011
Biaryl compounds useful as agonists of the Gpr38 receptor
GLAXO GROUP LTD10 citations83
US7531558B2May 12, 2009
Carboxamide derivatives
GLAXO GROUP LTD11 citations82
US7439245B2Oct 21, 2008
Compounds
GLAXO GROUP LTD0 citations52
JANSSEN PHARMACEUTICALS INC
6 patentsUS11071729B2Jul 27, 2021
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyridinyl-2′-ones
JANSSEN PHARMACEUTICALS INC1 citations72
US9737533B2Aug 22, 2017
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of prevention of neurological and psychiatric disorders
JANSSEN PHARMACEUTICALS INC3 citations72
US9226930B2Jan 5, 2016
1,2,4-triazolo [4,3-a] pyridine derivatives and their use for the treatment of prevention of neurological and psychiatric disorders
JANSSEN PHARMACEUTICALS INC3 citations72
US9132122B2Sep 15, 2015
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyridinyl-2′-ones
JANSSEN PHARMACEUTICALS INC2 citations59
US9266834B2Feb 23, 2016
1, 4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of MGLUR2-receptors
JANSSEN PHARMACEUTICALS INC2 citations57
US9085577B2Jul 21, 2015
7-aryl-1,2,4-triazolo[4,3-A]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
JANSSEN PHARMACEUTICALS INC1 citations51
MACDONALD GREGOR JAMES
5 patentsUS8791120B2Jul 29, 2014
Fast-dissociating dopamine 2 receptor antagonists
MACDONALD GREGOR JAMES2 citations60
US8778974B2Jul 15, 2014
Trisubstituted 1,2,4 triazoles
MACDONALD GREGOR JAMES2 citations57
US9174953B2Nov 3, 2015
Bicyclic thiazoles as allosteric modulators of mGluR5 receptors
MACDONALD GREGOR JAMES0 citations50
US8933101B2Jan 13, 2015
Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists
MACDONALD GREGOR JAMES0 citations50
US8906921B2Dec 9, 2014
4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists
MACDONALD GREGOR JAMES0 citations50
CONN P JEFFREY
4 patentsUS8592422B2Nov 26, 2013
Bicyclic triazole and pyrazole lactams as allosteric modulators of mGluR5 receptors
CONN P JEFFREY5 citations71
US8710074B2Apr 29, 2014
Dihydronaphthyridinyl(organo)methanone analogs as positive allosteric mGluR5 modulators
CONN P JEFFREY2 citations58
US9090632B2Jul 28, 2015
Bicyclic oxazole and thiazole compounds and their use as allosteric modulators of mGluR5 receptors
CONN P JEFFREY1 citations51
US8865725B2Oct 21, 2014
Substituted imidazopyrimidin-5(6H)-ones as allosteric modulators of MGLUR5 receptors
CONN P JEFFREY1 citations50
CID-NÚÑEZ JOSÉ MARIA
3 patentsUS9012448B2Apr 21, 2015
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of MGLUR2 receptors
CID-NÚÑEZ JOSÉ MARIA17 citations81
US9271967B2Mar 1, 2016
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
CID-NÚÑEZ JOSÉ MARIA4 citations70
US8993591B2Mar 31, 2015
1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positive allosteric modulators of MGLUR2 receptors
CID-NÚÑEZ JOSÉ MARIA4 citations70
JANSSEN PHARMACEUTICA NV
3 patentsUS9468640B2Oct 18, 2016
Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating dopamine 2 receptor antagonists
JANSSEN PHARMACEUTICA NV1 citations61
US9751860B2Sep 5, 2017
Piperidin-4YL-pyridazin-3-ylamine derivatives as fast dissociating dopamine 2 receptor antagonists
JANSSEN PHARMACEUTICA NV0 citations50
US9422296B2Aug 23, 2016
Fast-dissociating dopamine 2 receptor antagonists
JANSSEN PHARMACEUTICA NV0 citations50
THURING JOHANNES WILHELMUS JOHN F
2 patentsGIJSEN HENRICUS JACOBUS MARIA
2 patentsUS8546440B2Oct 1, 2013
Substituted bicyclic imidazole derivatives as gamma secretase modulators
GIJSEN HENRICUS JACOBUS MARIA5 citations71
US8772504B2Jul 8, 2014
Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators
GIJSEN HENRICUS JACOBUS MARIA2 citations60
AHMED MAHMOOD
1 patentSMITHKLINE BEECHAM PLC
1 patentPASTOR-FERNÁNDEZ JOAQUIN
1 patentBARTOLOMÉ-NEBREDA JOSÉ MANUEL
1 patentDE BRUYN MARCEL FRANS LEOPOLD
1 patentShowing the top 50 of 69 patents by PatentIndex Score.