Inventor

BURKHART JOSEPH P

US30 patents

⚠️ This page may combine multiple inventors who share the name “BURKHART JOSEPH P”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.

BURKHART JOSEPH P

MERRELL PHARMA INC

Peptidase inhibitors

Peptidase inhibitors

Peptidase inhibitors

Orally-active elastase inhibitors

Prolyl endopeptidase inhibitors

.increment.16 unsaturated C17 heterocyclic steroids useful as steroid C17-20 lyase inhibitors

16 unsaturated C17 heterocyclic steroids useful as steroid C17-20 lyase inhibitors

Acylated enol derivatives as prodrugs of elastase inhibitors

2,19-methyleneoxy and 2,19-methylenethio bridged steroids as aromatase, 19-hydroxylase inhibitors and methods of their use in the treatment of estrogen mediated disorders

Orally-active elastase inhibitors

Acylated enol derivatives as prodrugs of elastase inhibitors

Methods and compositions using Δ16 unsaturated C17 heterocyclic steroids useful as steroid C17-20 lyase inhibitors

MERRELL DOW PHARMA

Orally-active elastase inhibitors

2,19-methyleneoxy and 2,19-methylenethio bridged steroids as aromatase, 19-hydroxylaser inhibitors and methods of their use in the treatment of estrogen mediated disorders

4-amino-Δ4-steroids and their use as 5α-reductase inhibitors

Haloethyl-substituted steroid enzyme inhibitors

2β,19-methyleneamino bridged steroids as aromatase inhibitors

4-amino-4-ene-steroids and their use as 5α-reductase inhibitors

2,19-methyleneoxy and 2,19-methylenethio bridged steroids as aromatase and 19-hydroxylase inhibitors

Method of using 4-amino-Δ4 -steroids in the treatment of benign prostatic hyperplasia

2β,19-ethylene bridged steroids as aromatase inhibitors

Synthesis for the preparation of 4-amino-4,5-dihydro-2-furancarboxylic acid

Intermediates for the synthesis of 4-amino-4,5-dihydro-2-furancarboxylic acid

AVENTIS PHARMA INC

Elastase inhibitors

Acylated enol derivative of α-ketoesters and α-ketoamides

20-fluoro-17(20)-vinyl steroids

3-mercaptoacetylamino-1,5-substituted-2-oxo-azepan derivatives useful as inhibitors of matrix metalloproteinase

HOECHST MARION ROUSSEL INC

Acylated enol derivatives of α-ketoesters and α-ketoamides

Perfluoroalkyl ketone inhibitors of elastase and processes for making the same

Polyfluoroalkyl tryptophan tripeptide thrombin inhibitors