Inventor
DUTHEUIL GUILLAUME
BE23 patents
⚠️ This page may combine multiple inventors who share the name “DUTHEUIL GUILLAUME”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
OGEDA SA
13 patentsUS10836768B2Nov 17, 2020
N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
OGEDA SA1 citations72
US10787458B2Sep 29, 2020
Chiral synthesis of N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-A]pyrazines
OGEDA SA2 citations72
US10183948B2Jan 22, 2019
N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
OGEDA SA1 citations72
US9987274B2Jun 5, 2018
N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
OGEDA SA4 citations72
US9969745B2May 15, 2018
N-acyl-(3-substituted)-(8-methyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders
OGEDA SA2 citations72
US10683295B2Jun 16, 2020
Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-A]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof
OGEDA SA1 citations67
US12162849B2Dec 10, 2024
Synthesis of 3-methyl-1,2,4-thiadiazole-5-carbohydrazide or of the methyl-d3 deuterated form thereof
OGEDA SA0 citations62
US11731974B2Aug 22, 2023
N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
OGEDA SA0 citations62
US10941151B2Mar 9, 2021
Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof
OGEDA SA0 citations58
US10214533B2Feb 26, 2019
N-acyl-(3-substituted)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders
OGEDA SA0 citations51
US9926325B2Mar 27, 2018
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders
OGEDA SA0 citations51
US10544150B2Jan 28, 2020
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders
OGEDA SA0 citations49
US10065960B2Sep 4, 2018
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders
OGEDA SA0 citations40
EUROSCREEN SA
7 patentsUS9422299B2Aug 23, 2016
Substituted [1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
EUROSCREEN SA17 citations91
US8871761B2Oct 28, 2014
NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders
EUROSCREEN SA15 citations90
US9475814B2Oct 25, 2016
Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof
EUROSCREEN SA7 citations80
US9969738B2May 15, 2018
N-acyl-(3-substituted)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders
EUROSCREEN SA2 citations72
US10065961B2Sep 4, 2018
Chiral N-acyl-5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof
EUROSCREEN SA2 citations68
US10030025B2Jul 24, 2018
Substituted [1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
EUROSCREEN SA1 citations51
US9840508B2Dec 12, 2017
N-acyl-(3-substituted)-(8-methyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a] pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders
EUROSCREEN SA0 citations51
EPICS THERAPEUTICS
3 patentsUS12528769B2Jan 20, 2026
Synthesis of (2S,5R)-5-(2-chlorophenyl)-1-(2′-methoxy-[1,1′-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid
EPICS THERAPEUTICS0 citations60
US12054457B2Aug 6, 2024
Polymorphs of (2S,5R)-5-(2-chlorophenyl)-1-(2′-methoxy-[1,1′-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid and preparation processes thereof
EPICS THERAPEUTICS0 citations60
US12091400B2Sep 17, 2024
Piperidine derivatives as METTL3 inhibitors
EPICS THERAPEUTICS0 citations36