Inventor
GUSTAFSON GARY
US45 patents
⚠️ This page may combine multiple inventors who share the name “GUSTAFSON GARY”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
FORMA THERAPEUTICS INC
28 patentsUS10208052B1Feb 19, 2019
Compositions for activating pyruvate kinase
FORMA THERAPEUTICS INC36 citations97
US10675274B2Jun 9, 2020
Activating pyruvate kinase R
FORMA THERAPEUTICS INC12 citations94
US10550098B2Feb 4, 2020
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC17 citations94
US10414752B2Sep 17, 2019
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC19 citations94
US10005734B2Jun 26, 2018
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC25 citations94
US9834539B2Dec 5, 2017
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC28 citations94
US9815817B2Nov 14, 2017
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC24 citations94
US9771349B2Sep 26, 2017
Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC27 citations94
US9624175B2Apr 18, 2017
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC25 citations94
US9624216B2Apr 18, 2017
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC26 citations94
US10472371B2Nov 12, 2019
Compositions for activating pyruvate kinase
FORMA THERAPEUTICS INC13 citations92
US11649242B2May 16, 2023
Pyrrolopyrrole compositions as pyruvate kinase (PKR) activators
FORMA THERAPEUTICS INC5 citations85
US11396513B2Jul 26, 2022
Compositions for activating pyruvate kinase
FORMA THERAPEUTICS INC6 citations85
US11498913B2Nov 15, 2022
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC4 citations84
US11071725B2Jul 27, 2021
Activating pyruvate kinase R
FORMA THERAPEUTICS INC8 citations84
US11014927B2May 25, 2021
Pyrrolopyrrole compositions as pyruvate kinase (PKR) activators
FORMA THERAPEUTICS INC6 citations84
US10889567B2Jan 12, 2021
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC5 citations84
US10836771B2Nov 17, 2020
Compositions for activating pyruvate kinase
FORMA THERAPEUTICS INC7 citations84
US10550099B2Feb 4, 2020
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC4 citations84
US11161848B2Nov 2, 2021
Purinones as ubiquitin-specific protease 1 inhibitors
FORMA THERAPEUTICS INC1 citations73
US11001588B2May 11, 2021
Activating pyruvate kinase R and mutants thereof
FORMA THERAPEUTICS INC3 citations73
US10807976B2Oct 20, 2020
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC2 citations73
US10577329B2Mar 3, 2020
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC4 citations73
US10407419B2Sep 10, 2019
Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC5 citations73
US10399980B2Sep 3, 2019
Purinones as ubiquitin-specific protease 1 inhibitors
FORMA THERAPEUTICS INC2 citations73
US10189841B2Jan 29, 2019
Purinones as ubiquitin-specific protease 1 inhibitors
FORMA THERAPEUTICS INC3 citations73
US12275715B2Apr 15, 2025
Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA THERAPEUTICS INC0 citations63
US12043623B2Jul 23, 2024
Purinones as ubiquitin-specific protease 1 inhibitors
FORMA THERAPEUTICS INC0 citations62
NOVO NORDISK HEALTHCARE AG
6 patentsUS11980611B2May 14, 2024
Treating sickle cell disease with a pyruvate kinase R activating compound
NOVO NORDISK HEALTHCARE AG3 citations85
US11844787B2Dec 19, 2023
Activating pyruvate kinase R
NOVO NORDISK HEALTHCARE AG5 citations85
US12122778B2Oct 22, 2024
Activating pyruvate kinase R
NOVO NORDISK HEALTHCARE AG0 citations62
US12071440B2Aug 27, 2024
Pyrrolopyrrole compositions as pyruvate kinase (PKR) activators
NOVO NORDISK HEALTHCARE AG0 citations62
US12053458B2Aug 6, 2024
Treating sickle cell disease with a pyruvate kinase R activating compound
NOVO NORDISK HEALTHCARE AG0 citations62
US12128035B2Oct 29, 2024
Activating pyruvate kinase R
NOVO NORDISK HEALTHCARE AG1 citations57
FORMA TM2 INC
4 patentsUS10280150B2May 7, 2019
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors
FORMA TM2 INC19 citations93
US10266495B2Apr 23, 2019
Phenyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA TM2 INC19 citations93
US10253015B2Apr 9, 2019
Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA TM2 INC20 citations93
US10294206B2May 21, 2019
Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
FORMA TM2 INC7 citations83