Inventor · disambiguated record
Alfred Jonczyk
Also filed as: JONCZYK ALFRED · JONCZYK ALFRED DR
45 granted patents·13 pending applications·506 citations·filing 1985–2016
98Inventor score
Top patents by PatentIndex Score
58 records- 0190US8846694B2Pyrrolidone derivatives for use as MetAP-2 inhibitorsHEINRICH TIMO·Filed 2009·Granted Sep 30, 2014·35 cites·2 claims
- 0290US8791113B22,4-diaryl-substituted [1,8] naphthyridines as kinase inhibitors for use against cancerDORSCH DIETER·Filed 2011·Granted Jul 29, 2014·17 cites·20 claims
- 0388US6001961ACyclic adhesion inhibitorsMERCK PATENT GMBH·Filed 1996·Granted Dec 14, 1999·88 cites·5 claims
- 0482US9051318B2Pyrido [2, 3-B] pyrazine compounds and their therapeutical uses such as for inhibiting ATP consuming proteins and treating diseases associated therewithDORSCH DIETER·Filed 2012·Granted Jun 9, 2015·6 cites·19 claims
- 0582US8987301B2Heteroarylaminoquinolines as TGF-beta receptor kinase inhibitorsJONCZYK ALFRED·Filed 2010·Granted Mar 24, 2015·7 cites·19 claims
- 0682US8846931B2Bipyridyl derivativesHOELZEMANN GUENTER·Filed 2011·Granted Sep 30, 2014·6 cites·12 claims
- 0782US7138417B2Inhibitors of integrin αvβ6MERCK PATENT GMBH·Filed 2003·Granted Nov 21, 2006·17 cites·20 claims
- 0881US7470702B2BenzimidazolesMERCK PATENT GMBH·Filed 2004·Granted Dec 30, 2008·14 cites·13 claims
- 0979US8003657B2Heterocyclic substituted bisarylurea derivativesMERCK PATENT GMBH·Filed 2005·Granted Aug 23, 2011·4 cites·12 claims
- 1078US5849692ACyclic peptides containing Arg-Gly-Asp, and derivatives thereof, as adhesion inhibitorsMERCK PATENT GMBH·Filed 1996·Granted Dec 15, 1998·44 cites·18 claims
- 1176US10179777B23-(1H-benzimidazol-2-yl)-1H-pyridin-2-one derivativesMERCK PATENT GMBH·Filed 2016·Granted Jan 15, 2019·2 cites·17 claims
- 1276US9051307B2Bipyridyl derivativesMERCK PATENT GMBH·Filed 2014·Granted Jun 9, 2015·2 cites·9 claims
- 1376US8614226B2Hetaryl-[1,8]naphthyridine derivativesJONCZYK ALFRED·Filed 2010·Granted Dec 24, 2013·3 cites·11 claims
- 1476US5866540ACyclic adhesion inhibitorsMERCK PATENT GMBH·Filed 1995·Granted Feb 2, 1999·42 cites·3 claims
- 1575US8912216B2Hetaryl-[1,8]naphthyridine derivativesMERCK PATENT GMBH·Filed 2013·Granted Dec 16, 2014·2 cites·15 claims
- 1675US7547695B2PyridopyrimidinonesMERCK PATENT GMBH·Filed 2004·Granted Jun 16, 2009·11 cites·13 claims
- 1775US5705481ACyclopeptidesMERCK PATENT GMBH·Filed 1995·Granted Jan 6, 1998·32 cites·23 claims
- 1874US9382244B27-azaindole-2,7-naphthyridine derivative for the treatment of tumoursMERCK PATENT GMBH·Filed 2013·Granted Jul 5, 2016·1 cites·8 claims
- 1974US7846927B2N,N′-diphenylurea derivatives suitable as kinase inhibitorsMERCK PATENT GMBH·Filed 2005·Granted Dec 7, 2010·2 cites·16 claims
- 2073US6576637B1β-alanine derivativesMERCK PATENT GMBH·Filed 2000·Granted Jun 10, 2003·10 cites·10 claims
- 2171US8815893B2HetarylaminonaphthyridinesJONCZYK ALFRED·Filed 2011·Granted Aug 26, 2014·2 cites·20 claims
- 2271US6645991B1αvβ3 integrin inhibitorsMERCK PATENT GMBH·Filed 2000·Granted Nov 11, 2003·5 cites·16 claims
- 2370US6822074B1Process for the preparation of cyclo(Asp-DPhe-NMeVal-Arg-Gly)MERCK PATENT GMBH·Filed 2000·Granted Nov 23, 2004·7 cites·13 claims
- 2470US5693612ACyclopeptides of the formula IMERCK PATENT GMBH·Filed 1995·Granted Dec 2, 1997·32 cites·9 claims
- 2566US8765684B2Solid materials of {[(2S,5R,8S,11S)-5-benzyl-11-(3-guanidino-propyl)-8-isopropyl-7-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentaaza-cyclopentadec-2-yl]-acetic acid} and methods for obtaining themMERCK PATENT GMBH·Filed 2013·Granted Jul 1, 2014·1 cites·18 claims
- 2665US5962638APeptides and synthetic cell membranesMERCK PATENT GMBH·Filed 1995·Granted Oct 5, 1999·21 cites·16 claims
- 2763US8242128B21,3-benzoxazolyl derivatives as kinase inhibitorsSTAEHLE WOLFGANG·Filed 2004·Granted Aug 14, 2012·1 cites·18 claims
- 2862US7632951B2Inhibitors of integrin ανβ6MERCK PATENT GMBH·Filed 2002·Granted Dec 15, 2009·1 cites·26 claims
- 2962US6127335ACyclic adhesion inhibitorsMERCK PATENT GMBH·Filed 1997·Granted Oct 3, 2000·18 cites·5 claims
- 3062US4755592AStatine-containing peptides useful in medicamentsMERCK PATENT GMBH·Filed 1986·Granted Jul 5, 1988·11 cites·24 claims
- 3160US6995238B2Cyclopeptide derivativesBIOMET DEUTCHLAND GMBH·Filed 2002·Granted Feb 7, 2006·2 cites·15 claims
- 3258US2009082404A1BenzimidazolesMERCK PATENT GMBH·Filed 2008·Application pending·0 cites
- 3357US2011027209A1Compositions Containing Cyclic Peptides And Methods Of UseMERCK PATENT GMBH·Filed 2009·Application pending·0 cites
- 3454US6683051B1Pharmaceutical preparation containing a cyclopeptide and a chemotherapeutic agent or an angiogenesis inhibitorMERCK PATENT GMBH·Filed 1999·Granted Jan 27, 2004·15 cites·14 claims
- 3554US6610826B1Cyclopeptide derivatives with integrin inhibitor propertiesMERCK PATENT DEPT·Filed 1998·Granted Aug 26, 2003·13 cites·24 claims
- 3649US6169072B1Cyclic adhesion inhibitorsMERCK PATENT GMBH·Filed 1998·Granted Jan 2, 2001·8 cites·10 claims
- 3748US6534478B1Cyclic azapeptides with angiogenic effectMERCK PATENT GMBH·Filed 1998·Granted Mar 18, 2003·8 cites·8 claims
- 3848US2012220611A11,3-benzoxazolyl derivatives as kinase inhibitorsSTAEHLE WOLFGANG·Filed 2012·Application pending·0 cites
- 3947US4709010APeptides useful for inhibition of reninMERCK PATENT GMBH·Filed 1985·Granted Nov 24, 1987·4 cites·19 claims
- 4046US2007021456A1Aminobenzimidazole derivativesMERCK PATENT GMBH·Filed 2004·Application pending·0 cites
- 4145US2009124633A1N-oxides of heterocyclic substituted bisarylureas for treating kinase-mediated diseasesJONCZYK ALFRED·Filed 2007·Application pending·0 cites
- 4244US2007117849A1Alfavbeta3 and alfavbet6 integrin antagonists as antifibrotic agentsGOODMAN SIMON·Filed 2004·Application pending·0 cites
- 4343US7759302B2Peptidic sulfonamidesMERCK PATENT GMBH·Filed 2004·Granted Jul 20, 2010·0 cites·9 claims
- 4443US2007066606A1Benzylbenzimidazolyl derivativesSTAHLE WOLFGANG·Filed 2004·Application pending·0 cites
- 4543US2008045529A1Use Of ThienopyrimidinesMERCK PATENT GMBH·Filed 2004·Application pending·0 cites
- 4642US10278911B2Compositions containing cyclic peptides and methods of useMERCK PATENT GMBH·Filed 2015·Granted May 7, 2019·0 cites·23 claims
- 4742US7528139B2SulfonamidesMERCK PATENT GMBH·Filed 2005·Granted May 5, 2009·0 cites·21 claims
- 4842US2006241301A1Urea derivatives and their use as tyrosinkinase inhibitorsHOELZEMANN GUNTER·Filed 2004·Application pending·0 cites
- 4942US2008214582A1Purine Derivatives as Inhibitors of Receptor Tyrosine Kinase ActivityHOELZEMANN GUENTER·Filed 2006·Application pending·0 cites
- 5041US7135587B2Urea and urethane derivatives as integrin inhibitorsMERCK PATENT GMBH·Filed 2001·Granted Nov 14, 2006·0 cites·18 claims
Showing the top 50 of 58 patent records by PatentIndex Score.
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