Inventor
SARGES REINHARD
US47 patents
Patents
47 patentsUS5998463ADec 7, 1999
Glycogen phosphorylase inhibitors
PFIZER98 citations98
US4130714ADec 19, 1978
Hydantoin therapeutic agents
PFIZER71 citations96
US4117230ASep 26, 1978
Hydantoin derivatives as therapeutic agents
PFIZER62 citations96
US4980357ADec 25, 1990
Azolidinedione derivatives
PFIZER29 citations93
US4147795AApr 3, 1979
Hydantoin derivatives as therapeutic agents
PFIZER31 citations93
US4127665ANov 28, 1978
Thienohydantoin derivatives
PFIZER33 citations93
US4210667AJul 1, 1980
Pharmaceutical preparations containing coumarin carboxylic acid derivatives
PFIZER50 citations92
US3991207ANov 9, 1976
Combination therapy for Parkinson's disease
PFIZER35 citations87
US5064852ANov 12, 1991
Indolinone derivatives
PFIZER21 citations82
US4307108ADec 22, 1981
Method for lowering sorbitol levels using spiro-imides
PFIZER23 citations82
US4248882AFeb 3, 1981
Treating diabetes-associated complications with hydantoin amines
PFIZER18 citations82
US4181729AJan 1, 1980
Phenyl or phenoxy substituted spiro-imidazolidinedione derivatives
PFIZER23 citations82
US4045488AAug 30, 1977
Aminophenyltetralin compounds
PFIZER20 citations82
US4029731AJun 14, 1977
Aminophenyltetralin compounds
PFIZER24 citations82
US5011840AApr 30, 1991
Imidazolidinedione derivatives in diabetes treatment
PFIZER11 citations74
US4940708AJul 10, 1990
4-arylsulfonyl-3,4-dihydro-2(1H)-quinoxalinone-1-alkanoic acids, esters, and salts
PFIZER8 citations74
US4623725ANov 18, 1986
[1,2,4]Triazolo[4,3-a]quinoxaline-4-amine derivatives
PFIZER10 citations74
US4623728ANov 18, 1986
Intermediates for 1,3-disubstituted piperidine compounds as neuroleptic agents
PFIZER12 citations74
US4593037AJun 3, 1986
1,3-disubstituted piperidine compounds as neuroleptic agents
PFIZER9 citations74
US4547501AOct 15, 1985
Method of using [1,2,4]triazolo[4,3-a]quinoxaline-4-amine derivatives as antidepressant and antifatigue agents
PFIZER9 citations74
US4495187AJan 22, 1985
Method of using [1,2,4]triazolo[4,3-a]quinoxaline-4-amine derivatives as antidepressant and antifatigue agents
PFIZER13 citations74
US4348526ASep 7, 1982
Intermediates in the preparation of chiral hydantoins
PFIZER11 citations74
US4286098AAug 25, 1981
Process for the preparation of chiral hydantoins
PFIZER15 citations74
US4235911ANov 25, 1980
Hydantoin derivatives
PFIZER11 citations74
US4209630AJun 24, 1980
Hydantoin derivatives as therapeutic agents
PFIZER11 citations74
US4209527AJun 24, 1980
Benzimidazolone derivatives
PFIZER11 citations74
US4977178ADec 11, 1990
Method of treating anxiety and depression with 1-phenyl-2(1H,3H)-indolone psycho-therapeutic agents
PFIZER11 citations73
US4960785AOct 2, 1990
Indolinone derivatives
PFIZER11 citations73
US4181728AJan 1, 1980
Spiro-polycyclicimidazolidinedione derivatives
PFIZER16 citations73
US4147797AApr 3, 1979
Spiro-furanohydantoin derivatives
PFIZER12 citations70
US4474967AOct 2, 1984
8-Deutero and 8-tritio-substituted derivatives of D-4S-6-fluoro-spiro-[chroman-4,4'-imidazolidine]-2',5'-dione
PFIZER3 citations63
US4419521ADec 6, 1983
6-Halo-4-chromanamines useful as intermediates to make chiral hydantoins
PFIZER2 citations63
US4273775AJun 16, 1981
Hydantoin derivatives, anti-diabetic compositions thereof, and method of use thereof
PFIZER3 citations63
US4258054AMar 24, 1981
Hydantoin derivatives as therapeutic agents
PFIZER6 citations63
US4210756AJul 1, 1980
Tetrahydroquinoline hydantoins for chronic diabetic complications
PFIZER4 citations63
US4177282ADec 4, 1979
Hydantoin therapeutic agents
PFIZER5 citations63
US3961065AJun 1, 1976
Benzenesulfonylurea derivatives
PFIZER2 citations63
US4879391ANov 7, 1989
1-Phenyl-2(1H,3H)-indolone psychotherapeutic agents
PFIZER5 citations62
US4861880AAug 29, 1989
1-phenyl-2(1H,3H)-indolone psycho-therapeutic agents
PFIZER3 citations62
US4476307AOct 9, 1984
Heteroylidene indolone compounds
PFIZER6 citations62
US4471124ASep 11, 1984
Spiro-imide derivatives
PFIZER3 citations62
US4442114AApr 10, 1984
Imide derivatives
PFIZER4 citations62
US4283409AAug 11, 1981
Imidazolone derivatives
PFIZER3 citations62
US5362743ANov 8, 1994
Aminoquinoline derivatives
PFIZER5 citations61
US3987172AOct 19, 1976
Piperidinesulfonylurea derivatives
PFIZER3 citations60
US3944524AMar 16, 1976
4-Substituted-1-piperidinesulfonamides
PFIZER3 citations60
US3961067AJun 1, 1976
Composition comprising a benzenesulfonylurea hypoglycemic agent and method of treatment
PFIZER0 citations50