Inventor
SIFFERLEN THIERRY
CH41 patents
⚠️ This page may combine multiple inventors who share the name “SIFFERLEN THIERRY”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
IDORSIA PHARMACEUTICALS LTD
13 patentsUS11241431B2Feb 8, 2022
N-substituted indole derivatives as PGE2 receptor modulators
IDORSIA PHARMACEUTICALS LTD6 citations83
US9732075B2Aug 15, 2017
Benzimidazole-proline derivatives
IDORSIA PHARMACEUTICALS LTD8 citations82
US11325899B2May 10, 2022
Benzofurane and benzothiophene derivatives as PGE2 receptor modulators
IDORSIA PHARMACEUTICALS LTD6 citations73
US10329287B2Jun 25, 2019
Benzimidazole-proline derivatives
IDORSIA PHARMACEUTICALS LTD3 citations72
US10023560B2Jul 17, 2018
Crystalline salt form of (S)-(2-(6 chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist
IDORSIA PHARMACEUTICALS LTD3 citations72
US9914720B2Mar 13, 2018
Crystalline form of (S)-(2-(6-chloro-7-methyl-1H-benzo[D]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone and its use as orexin receptor antagonists
IDORSIA PHARMACEUTICALS LTD3 citations72
US9790208B2Oct 17, 2017
Crystalline salt form of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist
IDORSIA PHARMACEUTICALS LTD4 citations72
US11712438B2Aug 1, 2023
Phenyl derivatives as PGE2 receptor modulators
IDORSIA PHARMACEUTICALS LTD2 citations71
US11446298B2Sep 20, 2022
Pyrimidine derivatives
IDORSIA PHARMACEUTICALS LTD5 citations71
US9914721B2Mar 13, 2018
Use of benzimidazole-proline derivatives
IDORSIA PHARMACEUTICALS LTD4 citations71
US12011444B2Jun 18, 2024
N-substituted indole derivatives as PGE2 receptor modulators
IDORSIA PHARMACEUTICALS LTD2 citations70
US11839613B2Dec 12, 2023
Pyrimidine derivatives as PGE2 receptor modulators
IDORSIA PHARMACEUTICALS LTD1 citations61
US11040966B2Jun 22, 2021
Benzimidazole-proline derivatives
IDORSIA PHARMACEUTICALS LTD0 citations60
ACTELION PHARMACEUTICALS LTD
12 patentsUS7994336B2Aug 9, 2011
Azetidine compounds as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD23 citations92
US8003654B2Aug 23, 2011
N-glycinsulfonamide derivatives and uses as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD7 citations84
US7834028B2Nov 16, 2010
Pyrazolo-tetrahydro pyridine derivatives as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD9 citations84
US7435815B2Oct 14, 2008
Sulfonylamino-acetic acid derivatives
ACTELION PHARMACEUTICALS LTD10 citations84
US7279578B2Oct 9, 2007
Sulfonylamino-acetic acid derivatives
ACTELION PHARMACEUTICALS LTD11 citations84
US7192950B2Mar 20, 2007
Benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD15 citations84
US7538109B2May 26, 2009
Quinoxalin-3-one derivatives as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD7 citations74
US9493446B2Nov 15, 2016
Orexin receptor antagonists which are [ortho bi-(hetero-)aryl]-[2-(meta bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone derivatives
ACTELION PHARMACEUTICALS LTD6 citations73
US9211279B2Dec 15, 2015
Proline sulfonamide derivatives as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD3 citations62
US7915259B2Mar 29, 2011
Diazabicyclononene derivatives and use thereof
ACTELION PHARMACEUTICALS LTD3 citations62
US9403813B2Aug 2, 2016
Azetidine amide derivatives as orexin receptor antagonists
ACTELION PHARMACEUTICALS LTD1 citations52
US7799805B2Sep 21, 2010
Piperidine carboxylic acid amide derivatives
ACTELION PHARMACEUTICALS LTD1 citations51
AISSAOUI HAMED
11 patentsUS8288411B2Oct 16, 2012
Pyrrolidines and piperidines as orexin receptor antagonists
AISSAOUI HAMED14 citations84
US8236964B2Aug 7, 2012
Thiazolidine derivatives as orexin receptor antagonists
AISSAOUI HAMED13 citations84
US8106215B2Jan 31, 2012
3-aza-bicyclo[3.3.0]octane compounds
AISSAOUI HAMED13 citations84
US8288429B2Oct 16, 2012
2-aza-bicyclo[3.3.0]octane derivatives
AISSAOUI HAMED15 citations83
US8288435B2Oct 16, 2012
2-aza-bicyclo[3.1.0]hexane derivatives as orexin receptor antagonists
AISSAOUI HAMED11 citations83
US8063099B2Nov 22, 2011
Trans-3-aza-bicyclo[3.1.0]hexane derivatives
AISSAOUI HAMED7 citations82
US9242970B2Jan 26, 2016
Lactam derivatives useful as orexin receptor antagonists
AISSAOUI HAMED3 citations72
US8236801B2Aug 7, 2012
2-aza-bicyclo[2.2.1]heptane derivatives
AISSAOUI HAMED6 citations72
US8133901B2Mar 13, 2012
3-heteroaryl (amino or amido)-1-(biphenyl or phenylthiazolyl) carbonylpiperidine derivatives as orexin receptor inhibitors
AISSAOUI HAMED4 citations62
US8329706B2Dec 11, 2012
Oxazolidinone derivatives
AISSAOUI HAMED1 citations51
US7067519B2Jun 27, 2006
7,8,9,10-tetrahydro-6H-azepino, 6,7,8,9-tetrahydro-pyrido and 2,3-dihydro-2H-pyrrolo[2,1-b]-quinazolinone derivatives
AISSAOUI HAMED0 citations41