Inventor
GRAUERT MATTHIAS
DE74 patents
⚠️ This page may combine multiple inventors who share the name “GRAUERT MATTHIAS”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
BOEHRINGER INGELHEIM INT
24 patentsUS7241889B2Jul 10, 2007
6-formyl-tetrahydropteridines, process for their manufacture and use thereof as medicaments
BOEHRINGER INGELHEIM INT70 citations98
US7371753B2May 13, 2008
Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions
BOEHRINGER INGELHEIM INT77 citations97
US7332491B2Feb 19, 2008
Dihydropteridione derivatives, process for their manufacture and their use as medicament
BOEHRINGER INGELHEIM INT62 citations97
US7241769B2Jul 10, 2007
Pyrimidines as PLK inhibitors
BOEHRINGER INGELHEIM INT71 citations97
US7700769B2Apr 20, 2010
Dihydropteridione derivatives, process for their manufacture and their use as medicament
BOEHRINGER INGELHEIM INT32 citations96
US7629460B2Dec 8, 2009
Dihydropteridione derivatives, process for their manufacture and their use as medicament
BOEHRINGER INGELHEIM INT42 citations96
US7439358B2Oct 21, 2008
Specific salt, anhydrous and crystalline form of a dihydropteridione derivative
BOEHRINGER INGELHEIM INT50 citations96
US7414053B2Aug 19, 2008
Dihydropteridione derivatives, process for their manufacture and their use as medicament
BOEHRINGER INGELHEIM INT50 citations96
USRE47636EOct 8, 2019
Substituted spirocycles
BOEHRINGER INGELHEIM INT18 citations94
US9879026B2Jan 30, 2018
Substituted spirocycles
BOEHRINGER INGELHEIM INT17 citations94
US10238633B2Mar 26, 2019
Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C
BOEHRINGER INGELHEIM INT18 citations93
US7807831B2Oct 5, 2010
Dihydropteridione derivatives, process for their manufacture and their use as medicament
BOEHRINGER INGELHEIM INT30 citations93
US7723517B2May 25, 2010
Dihydropteridione derivatives, process for their manufacture and their use as medicament
BOEHRINGER INGELHEIM INT31 citations93
US9713606B2Jul 25, 2017
Methods for treating pulmonary emphysema using substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C
BOEHRINGER INGELHEIM INT20 citations92
US7759347B2Jul 20, 2010
2-benzylaminodihydropteridinones, process for their manufacture and use thereof as medicaments
BOEHRINGER INGELHEIM INT32 citations92
US7625899B2Dec 1, 2009
Pyridodihydropyraziones, process for their manufacture and use thereof as medicaments
BOEHRINGER INGELHEIM INT42 citations92
US7547780B2Jun 16, 2009
Dihydropteridione intermediate compounds
BOEHRINGER INGELHEIM INT44 citations91
US7517995B2Apr 14, 2009
Thiazolyl-dihydro-cyclopentapyrazole
BOEHRINGER INGELHEIM INT10 citations83
US10154990B2Dec 18, 2018
Medicaments for the treatment or prevention of fibrotic diseases
BOEHRINGER INGELHEIM INT15 citations82
US9440960B2Sep 13, 2016
Substituted oxetanes and their use as inhibitors of cathepsin C
BOEHRINGER INGELHEIM INT17 citations81
US9540373B2Jan 10, 2017
Substituted spirocycles
BOEHRINGER INGELHEIM INT4 citations73
US7691888B2Apr 6, 2010
Thiazolyl-dihydro-indazole
BOEHRINGER INGELHEIM INT7 citations71
US7902183B2Mar 8, 2011
Thiazolyl-dihydro-indazole
BOEHRINGER INGELHEIM INT4 citations61
US7691868B2Apr 6, 2010
Thiazolyl-dihydro-quinazoline
BOEHRINGER INGELHEIM INT3 citations61
BOEHRINGER INGELHEIM PHARMA
11 patentsUS7816530B2Oct 19, 2010
Piperazinyl compounds
BOEHRINGER INGELHEIM PHARMA49 citations98
US6861422B2Mar 1, 2005
Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions
BOEHRINGER INGELHEIM PHARMA115 citations98
US7750152B2Jul 6, 2010
Intermediate compounds for making dihydropteridinones useful as pharmaceutical compositions and processes of making the same
BOEHRINGER INGELHEIM PHARMA47 citations96
US6806272B2Oct 19, 2004
Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions
BOEHRINGER INGELHEIM PHARMA128 citations96
US8003786B2Aug 23, 2011
Dihydropteridinone compounds
BOEHRINGER INGELHEIM PHARMA34 citations95
US6696462B2Feb 24, 2004
Anticholinergics, processes for the preparation thereof, and pharmaceutical compositions
BOEHRINGER INGELHEIM PHARMA37 citations92
US7786299B2Aug 31, 2010
Methods for treating diseases or conditions using dihydropteridinone compounds
BOEHRINGER INGELHEIM PHARMA19 citations91
US6455538B1Sep 24, 2002
1,2,3,4,5,6-Hexahydro-2,6-methano-3-benzazocin-10-ols
BOEHRINGER INGELHEIM PHARMA10 citations72
US7094788B2Aug 22, 2006
Esters of hydroxyl-substituted nitrogen heterocycles, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions
BOEHRINGER INGELHEIM PHARMA2 citations62
US6770636B2Aug 3, 2004
Phenyl-and phenylalkyl-substituted ethanolamines and ethylenediamines
BOEHRINGER INGELHEIM PHARMA5 citations62
US6245777B1Jun 12, 2001
N-(5-phenyl-tetrahydrofuranyl)methyl- and N-(6-phenyl-tetrahydropyranyl)methyl-substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-10-ols
BOEHRINGER INGELHEIM PHARMA2 citations62
BOEHRINGER INGELHEIM KG
5 patentsUS5731318AMar 24, 1998
Benzomorphan derivatives
BOEHRINGER INGELHEIM KG15 citations73
US5196454AMar 23, 1993
Method of treating disorders of the dopaminergic systems using 2,5-diaminotetralines
BOEHRINGER INGELHEIM KG14 citations73
US5945535AAug 31, 1999
Method of preparing norbenzomorphanes
BOEHRINGER INGELHEIM KG8 citations72
US5053430AOct 1, 1991
Use of 2,7-diamino-1,2,3,4-tetrahydronaphthalenes as medicaments, new 2,7-diamino-1,2,3,4-tetrahydronaphthalenes and processes for their preparation
BOEHRINGER INGELHEIM KG5 citations62
US6054604AApr 25, 2000
Method of preparing norbenzomorphane as an intermediate
BOEHRINGER INGELHEIM KG1 citations61
ANDERSKEWITZ RALF
3 patentsUS8987249B2Mar 24, 2015
Substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C
ANDERSKEWITZ RALF48 citations97
US9073869B2Jul 7, 2015
Method of using substituted 2-Aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C
ANDERSKEWITZ RALF20 citations92
US8877775B2Nov 4, 2014
Substituted 2-aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C
ANDERSKEWITZ RALF21 citations92
GRAUERT MATTHIAS
3 patentsUS8889708B2Nov 18, 2014
Substituted bicyclic 1-carboxylic-acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C
GRAUERT MATTHIAS19 citations83
US8889677B2Nov 18, 2014
Substituted triazoles useful as mGlu5 receptor modulators
GRAUERT MATTHIAS8 citations83
US8642774B2Feb 4, 2014
Compounds
GRAUERT MATTHIAS5 citations71
BOEHRINGER SOHN INGELHEIM
1 patentLINZ GUENTER
1 patentHOFFMANN MATTHIAS
1 patentBOEHRINGER INGELHIEM PHARMA GM
1 patentShowing the top 50 of 74 patents by PatentIndex Score.