Inventor
METCALF ANDREW T
US25 patents
⚠️ This page may combine multiple inventors who share the name “METCALF ANDREW T”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
ARRAY BIOPHARMA INC
22 patentsUS10208024B2Feb 19, 2019
2-aryl- and 2-heteroaryl-substituted 2-pyridazin-3(2H)-one compounds as inhibitors of FGFR tyrosine kinases
ARRAY BIOPHARMA INC32 citations94
US10112942B2Oct 30, 2018
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC29 citations94
US10137124B2Nov 27, 2018
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC12 citations92
US10584124B2Mar 10, 2020
Crystalline forms
ARRAY BIOPHARMA INC12 citations86
US10953005B1Mar 23, 2021
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC4 citations84
US10555944B2Feb 11, 2020
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC10 citations84
US10172851B2Jan 8, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC8 citations84
US10172845B2Jan 8, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC4 citations83
US10144734B2Dec 4, 2018
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC6 citations83
US10881652B2Jan 5, 2021
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC2 citations72
US10441581B2Oct 15, 2019
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC2 citations72
US10154995B2Dec 18, 2018
Serine/threonine kinase inhibitors
ARRAY BIOPHARMA INC3 citations72
US9763942B2Sep 19, 2017
Serine/threonine kinase inhibitors
ARRAY BIOPHARMA INC5 citations72
US9670208B2Jun 6, 2017
Serine/threonine kinase inhibitors
ARRAY BIOPHARMA INC4 citations71
US11998545B2Jun 4, 2024
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations62
US11648243B2May 16, 2023
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations62
US11247990B1Feb 15, 2022
Bicyclic fused pyridine compounds as inhibitors of TAM kinases
ARRAY BIOPHARMA INC1 citations62
US11524963B2Dec 13, 2022
Substituted pyrazolo[3,4-d]pyrimidines as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations60
US10766881B2Sep 8, 2020
2-aryl- and 2-heteroaryl-substituted 2-pyridazin-3(2H)-one compounds as inhibitors of FGFR tyrosine kinases
ARRAY BIOPHARMA INC0 citations52
US11603374B2Mar 14, 2023
Substituted pyrrolo[2,3-d]pyrimidines compounds as ret kinase inhibitors
ARRAY BIOPHARMA INC0 citations50
US11472802B2Oct 18, 2022
Substituted pyrazolyl[4,3-c]pyridine compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations50
US11964988B2Apr 23, 2024
Fused heterocyclic compounds as RET kinase inhibitors
ARRAY BIOPHARMA INC0 citations49
LOXO ONCOLOGY INC
3 patentsUS10745419B2Aug 18, 2020
Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-carbonitrile
LOXO ONCOLOGY INC2 citations70
US11807651B2Nov 7, 2023
Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-carbonitrile
LOXO ONCOLOGY INC0 citations59
US11098064B2Aug 24, 2021
Process for the preparation of 6-(2-hydroxy-2-methylpropoxy)-4-(6-(6-((6-methoxypyridin-3-yl)methyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)pyridin-3-yl)pyrazolo[1,5-a]pyridine-3-carbontrile
LOXO ONCOLOGY INC1 citations59