Inventor
MEERPOEL LIEVEN
BE97 patents
⚠️ This page may combine multiple inventors who share the name “MEERPOEL LIEVEN”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
JANSSEN PHARMACEUTICA NV
31 patentsUS7615553B2Nov 10, 2009
Inhibitors of histone deacetylase
JANSSEN PHARMACEUTICA NV61 citations99
US7709487B2May 4, 2010
Sulfonyl-derivatives as novel inhibitors of histone deacetylase
JANSSEN PHARMACEUTICA NV53 citations97
US8343988B2Jan 1, 2013
Inhibitors of histone deacetylase
JANSSEN PHARMACEUTICA NV24 citations96
US7501417B2Mar 10, 2009
Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase
JANSSEN PHARMACEUTICA NV47 citations96
US7704998B2Apr 27, 2010
Sulfonyl-derivatives as novel inhibitors or histone deacetylase
JANSSEN PHARMACEUTICA NV39 citations95
US7205304B2Apr 17, 2007
Sulfonyl-Derivatives as novel inhibitors of histone deacetylase
JANSSEN PHARMACEUTICA NV54 citations94
US6878724B2Apr 12, 2005
Polyarylcarboxamides useful as lipid lowering agents
JANSSEN PHARMACEUTICA NV14 citations92
US5985878ANov 16, 1999
Angiogenesis inhibiting pyridazinamines
JANSSEN PHARMACEUTICA NV50 citations89
US7816360B2Oct 19, 2010
MTP inhibiting aryl piperidines or piperazines substituted with 5-membered heterocycles
JANSSEN PHARMACEUTICA NV9 citations83
US7504400B2Mar 17, 2009
MTP inhibiting aryl piperydines or piperazines substituted with 5-membered heterocycles
JANSSEN PHARMACEUTICA NV8 citations83
US11059850B2Jul 13, 2021
Spirobicyclic analogues
JANSSEN PHARMACEUTICA NV8 citations81
US10653711B2May 19, 2020
6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors
JANSSEN PHARMACEUTICA NV6 citations81
US9150560B2Oct 6, 2015
Inhibitors of histone deacetylase
JANSSEN PHARMACEUTICA NV3 citations74
US7244848B2Jul 17, 2007
Biphenylcarboxamides useful as lipid lowering agents
JANSSEN PHARMACEUTICA NV5 citations71
US11702441B2Jul 18, 2023
Spirobicyclic analogues
JANSSEN PHARMACEUTICA NV2 citations70
US11318157B2May 3, 2022
6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors
JANSSEN PHARMACEUTICA NV1 citations70
US10077261B2Sep 18, 2018
Imidazolin-5-one derivative useful as FASN inhibitors for the treatment of cancer
JANSSEN PHARMACEUTICA NV7 citations70
US10501469B2Dec 10, 2019
Substituted thiohydantoin derivatives as androgen receptor antagonists
JANSSEN PHARMACEUTICA NV1 citations69
US10138246B2Nov 27, 2018
Deuterated triazolopyridazine as a kinase modulator
JANSSEN PHARMACEUTICA NV2 citations67
US7202240B2Apr 10, 2007
Antifungal 4-substituted 5,6-dihydro-4h-pyrrolo[1,2-a][1,4] benzodiazepines
JANSSEN PHARMACEUTICA NV9 citations67
US7253157B2Aug 7, 2007
Polyarylcarboxamides useful as lipid lowering agents
JANSSEN PHARMACEUTICA NV2 citations62
US7169796B2Jan 30, 2007
Polyarylcarboxamides useful as lipid lowering agents
JANSSEN PHARMACEUTICA NV2 citations62
US6262052B1Jul 17, 2001
Amino acid ester containing azole antifungals
JANSSEN PHARMACEUTICA NV2 citations62
US11883367B2Jan 30, 2024
6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors
JANSSEN PHARMACEUTICA NV0 citations60
US9688696B2Jun 27, 2017
Piperidine/piperazine derivatives
JANSSEN PHARMACEUTICA NV1 citations60
US7135586B2Nov 14, 2006
Biphenylcarboxamides useful as lipid lowering agents
JANSSEN PHARMACEUTICA NV3 citations60
US12145961B2Nov 19, 2024
Spirobicyclic analogues
JANSSEN PHARMACEUTICA NV0 citations59
US11993614B2May 28, 2024
Monocyclic and bicyclic ring system substituted carbanucleoside analogues for use as PRMT5 inhibitors
JANSSEN PHARMACEUTICA NV0 citations59
US11267804B2Mar 8, 2022
(R)-8-(1-((3-fluorophenyl)amino)ethyl)-N-(2-hydroxyethyl)-2-morpholinoquinoxaline-6-carboxamide for inhibiting phosphoinositide-3-kinase activity
JANSSEN PHARMACEUTICA NV0 citations59
US11098062B2Aug 24, 2021
Monocyclic and bicyclic ring system substituted carbanucleoside analogues for use as PRMT5 inhibitors
JANSSEN PHARMACEUTICA NV0 citations59
US10981926B2Apr 20, 2021
Substituted thiohydantoin derivatives as androgen receptor antagonists
JANSSEN PHARMACEUTICA NV0 citations58
ASTEX THERAPEUTICS LTD
8 patentsUS9309242B2Apr 12, 2016
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD26 citations94
US9303029B2Apr 5, 2016
Substituted quinoxalines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD25 citations94
US9464071B2Oct 11, 2016
Pyrazolyl quinoxaline kinase inhibitors
ASTEX THERAPEUTICS LTD24 citations93
US9850228B2Dec 26, 2017
Pyrazolyl quinoxaline kinase inhibitors
ASTEX THERAPEUTICS LTD17 citations91
US10052320B2Aug 21, 2018
Substituted quinoxalines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD11 citations84
US10045982B2Aug 14, 2018
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD11 citations84
US9493426B2Nov 15, 2016
Quinazolinone derivatives useful as FGFR kinase modulators
ASTEX THERAPEUTICS LTD20 citations84
US10519137B2Dec 31, 2019
Pyrazolyl quinoxaline kinase inhibitors
ASTEX THERAPEUTICS LTD6 citations83
EMELEN KRISTOF VAN
5 patentsUS8865720B2Oct 21, 2014
Sulfonyl-derivatives as novel inhibitors of histone deacetylase
EMELEN KRISTOF VAN6 citations83
US8455498B2Jun 4, 2013
Inhibitors of histone deacetylase
EMELEN KRISTOF VAN3 citations73
US8114999B2Feb 14, 2012
Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase
EMELEN KRISTOF VAN3 citations70
US8097611B2Jan 17, 2012
Sulfonyl-derivatives as novel or histone deacetylase
EMELEN KRISTOF VAN3 citations62
US8557825B2Oct 15, 2013
Sulfonyl-derivatives as novel inhibitors of histone deacetylase
EMELEN KRISTOF VAN1 citations60
(unassigned)
2 patentsMEERPOEL LIEVEN
2 patentsANGIBAUD PATRICK RENE
1 patentSAXTY GORDON
1 patentShowing the top 50 of 97 patents by PatentIndex Score.