Inventor
GEORGE PASCAL
FR56 patents
⚠️ This page may combine multiple inventors who share the name “GEORGE PASCAL”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SYNTHELABO
41 patentsUS4460592AJul 17, 1984
6-Methyl-2-(4-methylthiophenyl)-imidazo[1,2-a]-pyridine-3-N,N-dimethylacetamide
SYNTHELABO55 citations96
US4382938AMay 10, 1983
Imidazo[1,2-a] pyridine derivatives and their application as pharmaceuticals
SYNTHELABO107 citations96
US4808594AFeb 28, 1989
Imidopyridines useful in therapy
SYNTHELABO47 citations93
US4977159ADec 11, 1990
2-[(4-piperidyl)methyl]-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole derivatives, and their application in treating depressive state, anxiety state or hypertension
SYNTHELABO46 citations92
US4492695AJan 8, 1985
Therapeutically useful imidazo[1,2-a]pyridine derivatives
SYNTHELABO28 citations92
US6075021AJun 13, 2000
1H-pyrido[3,4-b]indole-4-carboxamide derivatives, preparation and application thereof in therapeutics
SYNTHELABO30 citations91
US5663183ASep 2, 1997
N-(3-Aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide derivatives, their preparation and their therapeutic use
SYNTHELABO18 citations91
US5512590AApr 30, 1996
5,6-dihydro-4h-imidazo 2',1':2,3!imidazo- 4,5,1-ij!quinoline and 4,5-dihydroimidazo- 1,2-a!pyrolo 1,2,3-cd!benzimidazole derivatives, their preparation and application in therapeutics
SYNTHELABO20 citations91
US5447928ASep 5, 1995
Benzoxazine derivatives and their application in therapy
SYNTHELABO26 citations91
US5244901ASep 14, 1993
4-pyrimidinecarboxamide derivatives, their preparation and their application in therapy
SYNTHELABO27 citations91
US4650796AMar 17, 1987
3-acylaminomethylimidazo[1,2-a]pyridine derivatives and pharmaceutical compositions containing them
SYNTHELABO39 citations87
US4501745AFeb 26, 1985
Anxiolytic imidazo[1,2-a]pyridine derivatives
SYNTHELABO24 citations82
US4767755AAug 30, 1988
3-(acylaminomethyl)imidazo[1,2-a]pyridine derivatives and pharmaceutical compositions
SYNTHELABO19 citations80
US5272157ADec 21, 1993
Derivatives of 4-(aminomethyl) piperidine, their preparation and their therapeutic application
SYNTHELABO6 citations74
US5179108AJan 12, 1993
Derivatives of 4-(aminomethyl) piperidine, their preparation and their therapeutic application
SYNTHELABO17 citations74
US5254560AOct 19, 1993
2-piperidinylpyrimidine-4-carboxamide derivatives, and their use in therapeutics
SYNTHELABO7 citations73
US5244894ASep 14, 1993
2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
SYNTHELABO16 citations73
US5210086AMay 11, 1993
2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapy
SYNTHELABO15 citations73
US5164397ANov 17, 1992
2-aminopyrimidine-4-carboxamide derivatives, their preparation and their application in urinary therapeutics
SYNTHELABO11 citations73
US5550125AAug 27, 1996
3-(2-aminomethyl)-4-[3-trifluoromethyl)benzoyl]-3-4 dihydro-2h-1,4-benzoxazine derivatives and their therapeutic application
SYNTHELABO9 citations72
US5229392AJul 20, 1993
2-aminopyrimidine-4-carboxamide derivatives, their preparaton and their application in therapy
SYNTHELABO10 citations72
US5096900AMar 17, 1992
(4-piperidyl)methyl-2,3-dihydro-1h-isoindole and -2,3,4,5-tetrahydro-1h-benzazepine derivatives, their preparation and their application in therapy
SYNTHELABO9 citations72
US4891371AJan 2, 1990
3-(Acylaminomethyl)imidazo[1,2-a]pyridine derivatives, their preparation and their application in therapy
SYNTHELABO9 citations72
US5550162AAug 27, 1996
N-(-3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydro-naphthalene-2-carboxamide derivatives, their preparation and their therapeutic use
SYNTHELABO6 citations71
US5543421AAug 6, 1996
Method of treatment of peripheral neuropathies and central neurodegenerative diseases
SYNTHELABO8 citations71
US4675323AJun 23, 1987
Imidazo(1,2-a)quinoline derivatives useful as anxiolytic agents
SYNTHELABO12 citations71
US5466706ANov 14, 1995
9H-imidazo[1,2-A]benzimidazole-3-acetamide derivatives, their preparation and their therapeutic application
SYNTHELABO13 citations70
US4847263AJul 11, 1989
Imidazopyridine derivatives and compositions containing them
SYNTHELABO16 citations69
US5420130AMay 30, 1995
2-aminopyrazine-5-carboxamide derivatives, their preparation and their application in therapeutics
SYNTHELABO6 citations63
US4945096AJul 31, 1990
Treatment of a depressive state with 2-[(4-piperidyl)methyl]-1,2,3,4-tetrahydroisoquinoline derivates
SYNTHELABO4 citations63
US5922739AJul 13, 1999
5-Naphthalen-1-yl-1,3-dioxane derivatives, preparation and therapeutical use thereof
SYNTHELABO6 citations62
US5330985AJul 19, 1994
2-amino-N-[[4-(aminocarbonyl)pyrimidin-2-yl]amino]-alkyl]pyrimidine-4-carboxamide derivatives, their preparation and pharmaceutical compositions containing them
SYNTHELABO6 citations62
US5246939ASep 21, 1993
2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
SYNTHELABO5 citations62
US4925850AMay 15, 1990
Derivatives of 2-((4-piperidinyl)methyl)-1,2,3,4-tetrahydroisoquinoline, their preparation and their application in therapeutics
SYNTHELABO6 citations62
US5081128AJan 14, 1992
2,3-dihydro-1h-isoindole derivatives and their application in therapy
SYNTHELABO3 citations61
US4990506AFeb 5, 1991
3-(acylaminomethyl)imidazo[1,2-a]pyridine derivatives and their application in therapy
SYNTHELABO2 citations61
US5929078AJul 27, 1999
1- 2-(2,3-Dihydro-1H-inden-1-yl)ethyl!-4-(naphthalen-1-yl) piperazine, derivatives, preparation thereof and therapeutical use thereof
SYNTHELABO2 citations60
US5064836ANov 12, 1991
Imidazopyridine for use as an anaesthetic
SYNTHELABO2 citations59
US4810711AMar 7, 1989
1-(acylaminomethyl)imidazo(1,2-A)quinoline derivatives, their preparation and their application in therapy
SYNTHELABO2 citations59
US4931449AJun 5, 1990
2-((4-piperidyl)methyl)benzofuro(2,3-C)pyridine derivatives, and their application in therapy
SYNTHELABO1 citations51
US5418248AMay 23, 1995
2-thienylimidazo[2,1-β]benzothiazole-3-acetic acid derivatives, their preparation and their use
SYNTHELABO0 citations50
SANOFI AVENTIS
3 patentsUS7476756B2Jan 13, 2009
Alkyl-, alkenyl- and alkynylcarbamate derivatives, their preparation and their application in therapeutics
SANOFI AVENTIS36 citations92
US7507743B2Mar 24, 2009
Substituted 8′-pyridinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a] pyrimidin-6-one and 8′-pyrimidinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a] pyrimidin-6-one derivatives
SANOFI AVENTIS1 citations52
US7294632B2Nov 13, 2007
Substituted 8′-pyridinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a]pyrimidin-6-one and 8′-pyrimidinyl-dihydrospiro-[cycloalkyl]-pyrimido[1,2-a]pyrimidin-6-one derivatives
SANOFI AVENTIS0 citations52
STEP PHARMA S A S
3 patentsUS11505547B2Nov 22, 2022
Compounds
STEP PHARMA S A S3 citations70
US12466810B2Nov 11, 2025
N-(5-(6-ethoxypyrazin-2-yl)pyridin-2-yl)-4-(2-(methylsulfonamido)pyrimidin-4-yl) tetrahydro-2H-pyran-4-carboxamide derivatives and related compounds as human CTPS1 inhibitors for the treatment of proliferative diseases
STEP PHARMA S A S0 citations58
US11655246B2May 23, 2023
Aminothiazole compounds as inhibitors of CTPS1
STEP PHARMA S A S1 citations56
GEORGE PASCAL
1 patentSANOFI SYNTHELABO
1 patentSANOFI SA
1 patentShowing the top 50 of 56 patents by PatentIndex Score.