Inventor
KYBURZ EMILIO
CH75 patents
Patents
50 patentsUS4407752AOct 4, 1983
Azeto-imidazo-diazepines
HOFFMANN LA ROCHE65 citations96
US4405517ASep 20, 1983
Azeto-diazepines
HOFFMANN LA ROCHE64 citations96
US4405516ASep 20, 1983
Benzodiazepine derivatives
HOFFMANN LA ROCHE66 citations96
US4386028AMay 31, 1983
Imidazo[1,5a][1,4]benzodiazepines
HOFFMANN LA ROCHE67 citations96
US4382032AMay 3, 1983
Diazepine derivatives
HOFFMANN LA ROCHE64 citations96
US4353827AOct 12, 1982
Diazepine derivatives
HOFFMANN LA ROCHE73 citations96
US4316839AFeb 23, 1982
Imidazodiazepine derivatives
HOFFMANN LA ROCHE70 citations96
US4775671AOct 4, 1988
Imidazodiazepines
HOFFMANN LA ROCHE38 citations93
US4764522AAug 16, 1988
Ethylenediamine monoamides
HOFFMANN LA ROCHE33 citations92
US5011849AApr 30, 1991
Compounds for treating and preventing cognitive diseases and depression and methods of making same
HOFFMANN LA ROCHE50 citations91
US5387585AFeb 7, 1995
Imidazodiazepine derivatives
HOFFMANN LA ROCHE53 citations90
US4476308AOct 9, 1984
1-Pyrrolidine acetamides
HOFFMANN LA ROCHE18 citations82
US4369139AJan 18, 1983
1-(P-Methoxy p-hydroxy, and p-benzyloxy benzoyl)-2-pyrrolidinones
HOFFMANN LA ROCHE21 citations82
US4352815AOct 5, 1982
Imidazo-benzodiazepines and their use
HOFFMANN LA ROCHE22 citations82
US4352818AOct 5, 1982
Diazepine derivatives and their use
HOFFMANN LA ROCHE22 citations82
US4236010ANov 25, 1980
Phenyl-quinolizidines
HOFFMANN LA ROCHE13 citations82
US4359420ANov 16, 1982
Thieno-1,4-diazepin-5-ones and benzo-1,4-diazepin-5-ones
HOFFMANN LA ROCHE11 citations81
US4489003ADec 18, 1984
Imidazobenzodiazepines
HOFFMANN LA ROCHE17 citations74
US4391978AJul 5, 1983
Phenyl-quinolizidines
HOFFMANN LA ROCHE5 citations74
US4362732ADec 7, 1982
Diazepine derivatives and their use
HOFFMANN LA ROCHE9 citations74
US4352817AOct 5, 1982
Imidazo-diazepines and their use
HOFFMANN LA ROCHE16 citations74
US4352816AOct 5, 1982
Azeto-imidazo-diazepines and their use
HOFFMANN LA ROCHE11 citations74
US4044010AAug 23, 1977
Dibenzo[b,f] thiepins bearing piperazinyl substitution
HOFFMANN LA ROCHE8 citations74
US3966737AJun 29, 1976
Fluoro-substituted dibenso[b,f] thiepins
HOFFMANN LA ROCHE8 citations74
US3954764AMay 4, 1976
Dibenzo [b,f]thiepins bearing piperazinyl substitution
HOFFMANN LA ROCHE13 citations74
US5034402AJul 23, 1991
Methods and pharmaceutical compositions using pyrrolidine derivatives
HOFFMANN LA ROCHE12 citations73
US4749791AJun 7, 1988
Benzo[f]quinoline intermediates
HOFFMANN LA ROCHE10 citations73
US4732979AMar 22, 1988
Benzazecine derivatives for cognitive and memory functions
HOFFMANN LA ROCHE5 citations73
US4650878AMar 17, 1987
2-(2-oxo-1-pyrrolidinyl) acetic acids
HOFFMANN LA ROCHE12 citations73
US4452807AJun 5, 1984
(R,S)-1-(3-Hydroxy-4-methoxybenzoyl)-3-hydroxy-2-pyrrolidinone intermediates therefor and use for treating cerebral insufficiency
HOFFMANN LA ROCHE9 citations73
US4363762ADec 14, 1982
Process for preparing imidazodiazepines
HOFFMANN LA ROCHE4 citations73
US4346030AAug 24, 1982
Imidazodiazepine derivatives
HOFFMANN LA ROCHE6 citations73
US4346036AAug 24, 1982
Process for preparing imidazodiazepine derivatives
HOFFMANN LA ROCHE4 citations73
US4346032AAug 24, 1982
Imidazodiazepine derivatives
HOFFMANN LA ROCHE4 citations73
US4346034AAug 24, 1982
Process for preparing imidazodiazepines
HOFFMANN LA ROCHE4 citations73
US4346031AAug 24, 1982
Process for preparing imidazodiazepines
HOFFMANN LA ROCHE4 citations73
US4346035AAug 24, 1982
Process for preparing imidazodiazepines
HOFFMANN LA ROCHE4 citations73
US4346033AAug 24, 1982
Thienodiazepinone and benzodiazepinone intermediates
HOFFMANN LA ROCHE3 citations73
US4239770ADec 16, 1980
Substituted 2-pyrrolidinones for counteracting cerebral insufficiency
HOFFMANN LA ROCHE5 citations73
US4863920ASep 5, 1989
Imidazodiazepine derivatives for treatment of disorders of the central nervous system
HOFFMANN LA ROCHE10 citations70
US5238962AAug 24, 1993
Benzamide derivatives
HOFFMANN LA ROCHE10 citations65
US5017608AMay 21, 1991
Hydrocinnamic acid derivatives
HOFFMANN LA ROCHE4 citations63
US4338444AJul 6, 1982
Phenyl-hexahydro-2H-quinolizines
HOFFMANN LA ROCHE1 citations63
US4329467AMay 11, 1982
Phenyl-quinolizidines
HOFFMANN LA ROCHE1 citations63
US4316030AFeb 16, 1982
Phenyl-quinolizidines
HOFFMANN LA ROCHE1 citations63
US4306067ADec 15, 1981
Precursors of phenyl-quinolizidines
HOFFMANN LA ROCHE1 citations63
US4272627AJun 9, 1981
Phenyl-quinolizinones
HOFFMANN LA ROCHE2 citations63
US4118572AOct 3, 1978
Dibenz(b,f)oxepin derivatives
HOFFMANN LA ROCHE1 citations63
US4105664AAug 8, 1978
Dibenz[b,f]oxepin derivatives
HOFFMANN LA ROCHE2 citations63
US4100173AJul 11, 1978
Dibenz[b,f]oxepin derivatives
HOFFMANN LA ROCHE3 citations63
Showing the top 50 of 75 patents by PatentIndex Score.