Inventor
MATHIAS JOHN PAUL
US30 patents
⚠️ This page may combine multiple inventors who share the name “MATHIAS JOHN PAUL”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
PFIZER
23 patentsUS6916927B2Jul 12, 2005
Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3′,5′-monophosphate phosphodiesterase (cGMP-PDE5) for the treatment of sexual dysfunction
PFIZER113 citations97
US9879022B2Jan 30, 2018
Bicyclic-fused heteroaryl or aryl compounds
PFIZER19 citations93
US9458168B2Oct 4, 2016
Bicyclic-fused heteroaryl or aryl compounds
PFIZER17 citations92
US6670366B1Dec 30, 2003
Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction
PFIZER36 citations92
US6458951B2Oct 1, 2002
Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction
PFIZER39 citations92
US6407114B1Jun 18, 2002
Pyrazolopyrimidinone CGMP PDE5 inhibitors for the treatment of sexual dysfunction
PFIZER28 citations92
US6333330B1Dec 25, 2001
Pyrazolopyrimidinone CGMP PDE5 inhibitors for the treatment of sexual dysfunction
PFIZER39 citations92
US6251904B1Jun 26, 2001
Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction
PFIZER35 citations92
US6677335B1Jan 13, 2004
Pharmaceutically active compounds
PFIZER28 citations90
US11702424B2Jul 18, 2023
Bicyclic-fused heteroaryl or aryl compounds
PFIZER4 citations85
US7153870B2Dec 26, 2006
Nicotinamide derivatives useful as PDE4 inhibitors
PFIZER11 citations84
US6723719B1Apr 20, 2004
Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3′,5′—monophosphate phosphodiesterase (cGMP PDE5) for the treatment of sexual dysfunction
PFIZER14 citations84
US10793579B2Oct 6, 2020
Bicyclic-fused heteroaryl or aryl compounds
PFIZER3 citations83
US10329302B2Jun 25, 2019
Bicyclic-fused heteroaryl or aryl compounds
PFIZER3 citations83
US7511057B2Mar 31, 2009
Triazolopyridinylsulfanyl derivatives as p38 MAP kinase inhibitors
PFIZER11 citations83
US10316018B2Jun 11, 2019
Bicyclic-fused heteroaryl or aryl compounds as IRAK4 modulators
PFIZER2 citations72
US10174000B2Jan 8, 2019
Bicyclic-fused heteroaryl or aryl compounds as IRAK4 modulators
PFIZER5 citations72
US6936619B2Aug 30, 2005
Quinazolinone compounds useful in therapy
PFIZER7 citations70
US10308615B2Jun 4, 2019
Heterocyclic compounds as inhibitors of Vanin-1 enzyme
PFIZER3 citations68
US7056934B2Jun 6, 2006
Nicotinamide derivatives useful as PDE4 inhibitors
PFIZER2 citations63
US12202836B2Jan 21, 2025
Bicyclic-fused heteroaryl or aryl compounds
PFIZER0 citations62
US7176311B2Feb 13, 2007
Process for preparing pharmaceutically active compounds
PFIZER2 citations60
US7557121B2Jul 7, 2009
Tetrahydronaphthyridine derivatives
PFIZER3 citations59
CYSTIC FIBROSIS FOUND THERAPEUTICS INC
4 patentsUS10208053B2Feb 19, 2019
Bicyclic heteroaryl derivatives as CFTR potentiators
CYSTIC FIBROSIS FOUND THERAPEUTICS INC31 citations92
US10131670B2Nov 20, 2018
Bicyclic heteroaryl derivatives as CFTR potentiators
CYSTIC FIBROSIS FOUND THERAPEUTICS INC27 citations92
US10377762B2Aug 13, 2019
Bicyclic heteroaryl derivatives as CFTR potentiators
CYSTIC FIBROSIS FOUND THERAPEUTICS INC1 citations71
US10301315B2May 28, 2019
Pyrrolopyrimidines as CFTR potentiators
CYSTIC FIBROSIS FOUND THERAPEUTICS INC1 citations61