Inventor
GRAPPERHAUS MARGARET L
US37 patents
⚠️ This page may combine multiple inventors who share the name “GRAPPERHAUS MARGARET L”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
PHARMACIA CORP
18 patentsUS6723753B2Apr 20, 2004
Substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP22 citations96
US6723752B2Apr 20, 2004
(R)-chiral halogenated substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP53 citations96
US6710089B2Mar 23, 2004
Substituted N-fused-phenyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP23 citations96
US6683099B2Jan 27, 2004
Substituted N,N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP19 citations96
US6677375B2Jan 13, 2004
Substituted N,N-bis-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP19 citations96
US6677341B2Jan 13, 2004
(R)-Chiral halogenated substituted heteroaryl benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP13 citations93
US6586433B2Jul 1, 2003
Substituted N-heteroaryl-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP13 citations93
US6521607B1Feb 18, 2003
(R)-chiral halogenated substituted N-phenoxy N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP17 citations93
US7119203B2Oct 10, 2006
Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
PHARMACIA CORP11 citations83
US6696472B2Feb 24, 2004
Substituted N-phenoxy-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP11 citations82
US6696435B2Feb 24, 2004
Substituted N,N-disubstituted fused-heterocyclo amino compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP7 citations82
US6683113B2Jan 27, 2004
(R)-chiral halogenated substituted N,N-Bis-benzyl aminioalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP11 citations82
US6677353B2Jan 13, 2004
Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP12 citations82
US6677379B2Jan 13, 2004
Substituted N,N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP12 citations82
US6677380B2Jan 13, 2004
Substituted N, N-disubstituted mercapto amino compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP11 citations82
US6583183B2Jun 24, 2003
Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP11 citations82
US6677382B1Jan 13, 2004
Substituted N,N-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PHARMACIA CORP10 citations74
US6465686B2Oct 15, 2002
Halogenated 2-amino-5,6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
PHARMACIA CORP10 citations72
SEARLE & CO
12 patentsUS6458803B1Oct 1, 2002
Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO48 citations97
US6476075B1Nov 5, 2002
Use of substituted N, N-bis-benzyl aminoalcohol compounds inhibiting cholesteryl ester transfer protein activity
SEARLE & CO29 citations96
US6462092B1Oct 8, 2002
Use of substituted N, N-disubstituted reverse aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO23 citations96
US6455519B1Sep 24, 2002
Use of substituted N, N-disubstituted fused-heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO17 citations96
US6451830B1Sep 17, 2002
Use of substituted N,N-disubstituted non-fused heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO17 citations96
US6451823B1Sep 17, 2002
Use of substituted N-phenoxy-N-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO18 citations96
US6448295B1Sep 10, 2002
Use of substituted N-fused-phenyl-N-benzyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO17 citations96
US6544974B2Apr 8, 2003
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO13 citations93
US6479552B2Nov 12, 2002
Use of substituted N, N-disubstituted diamino compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO15 citations93
US6476057B1Nov 5, 2002
Use of substituted N, N-disubstituted cycloalkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO12 citations82
US6458849B1Oct 1, 2002
use of substituted N,N-disubstituted mercapto amino compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO12 citations82
US6458852B1Oct 1, 2002
Use of substituted N, N-bis-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
SEARLE & CO10 citations82
PFIZER
6 patentsUS6803388B2Oct 12, 2004
(R)-Chiral halogenated substituted n,n-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PFIZER15 citations93
US6765023B2Jul 20, 2004
Use of substituted N, N-disubstituted reverse aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PFIZER14 citations93
US6787570B2Sep 7, 2004
Substituted N-cycloalkyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
PFIZER13 citations84
US7253211B2Aug 7, 2007
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity
PFIZER0 citations52
US7122536B2Oct 17, 2006
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity
PFIZER0 citations52
US7700658B2Apr 20, 2010
(R)-chiral halogenated substituted fused heterocyclic amino compounds useful for inhibiting cholesterol ester transfer protein activity
PFIZER0 citations51