Inventor
SANTILLI ARTHUR A
44 patents
⚠️ This page may combine multiple inventors who share the name “SANTILLI ARTHUR A”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
AMERICAN HOME PROD
32 patentsUS5998402ADec 7, 1999
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
AMERICAN HOME PROD172 citations99
US6369056B1Apr 9, 2002
Cyclic urea and cyclic amide derivatives
AMERICAN HOME PROD61 citations96
US6306851B1Oct 23, 2001
Cyclocarbamate and cyclic amide derivatives
AMERICAN HOME PROD65 citations96
US4284768AAug 18, 1981
1,2-Dihydro-4-amino-2-oxo-3-quinoline-carboxylic acid derivatives
AMERICAN HOME PROD65 citations96
US6380178B1Apr 30, 2002
Cyclic regimens using cyclocarbamate and cyclic amide derivatives
AMERICAN HOME PROD45 citations92
US6232307B1May 15, 2001
Tissue selective compounds in the treatment of ovarian cancer
AMERICAN HOME PROD18 citations92
US6225308B1May 1, 2001
Tissue selective compounds in the treatment of prostate cancer or benign prostate hypertrophy
AMERICAN HOME PROD16 citations92
US4215123AJul 29, 1980
Antisecretory 4-oxy-3-carboxy or cyano-1,2-dihydro-2-oxo-1,8-naphthyridine derivatives
AMERICAN HOME PROD45 citations92
US6291451B1Sep 18, 2001
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
AMERICAN HOME PROD12 citations82
US6127404AOct 3, 2000
Tissue selective compounds in the treatment of endometrial proliferation
AMERICAN HOME PROD14 citations82
US4452985AJun 5, 1984
2-Guanyl-4-(substituted phenyl) thiazole derivatives
AMERICAN HOME PROD22 citations82
US4215216AJul 29, 1980
7,8-Dihydro-2,5,8-trisubstituted-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives
AMERICAN HOME PROD24 citations82
US4148801AApr 10, 1979
3-[(Chlorophenylsulfonyl)methyl]-1,2,4-oxadiazole-5-carboxylic acid derivatives
AMERICAN HOME PROD25 citations82
US3974162AAug 10, 1976
4-Pyrimidinylthioacetic acid derivatives
AMERICAN HOME PROD23 citations78
US6326367B1Dec 4, 2001
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
AMERICAN HOME PROD5 citations74
US5081253AJan 14, 1992
Imidazo(4,5-c)pyridines as antiosteoporotic agents
AMERICAN HOME PROD9 citations74
US4324893AApr 13, 1982
4-Amino-3-carboxy or cyano-1,2-dihydro-2-oxo-1,8-naphthyridine derivatives
AMERICAN HOME PROD15 citations74
US4301281ANov 17, 1981
7,8-Dihydro-2,5,8-trisubstituted-7-oxo-pyrido[2,3-d]-pyrimidine-6-carboxylic acid amides
AMERICAN HOME PROD15 citations74
US4236004ANov 25, 1980
2-Alkylsulphonyl-7,8-dihydro-5-hydroxy-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives
AMERICAN HOME PROD5 citations74
US3940395AFeb 24, 1976
4-Amino-2-phenyl-6-thiopryimidines
AMERICAN HOME PROD10 citations74
US4743692AMay 10, 1988
N-(pyridinylalkyl)-thieno-or benzo-isothiazol-3-amine derivatives
AMERICAN HOME PROD10 citations73
US5288871AFeb 22, 1994
Antiosteoporotic imidazo[4,5-c]pyridines
AMERICAN HOME PROD7 citations68
US4350817ASep 21, 1982
4-Cl, Br or I-3-Carboxy or cyano-1,2-dihydro-2-oxo-1,8-naphthyridine derivatives
AMERICAN HOME PROD4 citations63
US4255568AMar 10, 1981
2H-Pyrimido[4,5-d][1,3]oxazine-2,4(1H)-dione derivatives
AMERICAN HOME PROD4 citations63
US4245094AJan 13, 1981
5-Amino-2,8-dialkyl-7,8-dihydro-7-oxo-pyrido-[2,3-d]pyrimidine-6 carboxylic acid derivatives
AMERICAN HOME PROD4 citations63
US6380185B1Apr 30, 2002
N-substituted benzoyl indoles as estrogenic agents
AMERICAN HOME PROD2 citations62
US3988335AOct 26, 1976
1-Substituted-6-(2-substituted aminoethoxy)xanthen-9-ones
AMERICAN HOME PROD5 citations62
US4621142ANov 4, 1986
Precursors of benzo- and thieno-fused heterocyclic anti-ulcer agents
AMERICAN HOME PROD1 citations52
US4537968AAug 27, 1985
Thiophene derivatives with antisecretory activity
AMERICAN HOME PROD1 citations52
US4266050AMay 5, 1981
1,2-Dihydro-4-hydroxy-2-imino-N-substituted-3-quinolinecarboxamide derivatives
AMERICAN HOME PROD0 citations52
US4233446ANov 11, 1980
5-Chloro-7,8-dihydro-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives
AMERICAN HOME PROD0 citations52
US3950339AApr 13, 1976
Substituted-2-(pyrimidinylthio)acetamidoximes and acetonitriles
AMERICAN HOME PROD1 citations52
WYETH CORP
11 patentsUS6924281B2Aug 2, 2005
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP12 citations92
US6835729B2Dec 28, 2004
2-phenyl-1-[4(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP14 citations92
US6787538B2Sep 7, 2004
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP13 citations92
US6441019B2Aug 27, 2002
Cyclocarbamate and cyclic amide derivatives
WYETH CORP47 citations92
US6399593B1Jun 4, 2002
Cyclic regimens using cyclic urea and cyclic amide derivatives
WYETH CORP47 citations92
US7132417B2Nov 7, 2006
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP9 citations82
US7041663B2May 9, 2006
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP10 citations82
US7678787B2Mar 16, 2010
Pyrrolobenzodiazepine pyridine carboxamides and derivatives as follicle-stimulating hormone receptor antagonists
WYETH CORP15 citations79
US7247624B2Jul 24, 2007
2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP3 citations74
US6951852B2Oct 4, 2005
2-Phenyl-1-[4-(2-Aminoethoxy)-Benzyl]-Indoles as estrogenic agents
WYETH CORP4 citations74
US7449455B2Nov 11, 2008
2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
WYETH CORP1 citations63