P

Inventor

JANSSENS FRANS E

BE38 patents

Patents

38 patents
US5258380ANov 2, 1993

(4-piperidinylmethyl and -hetero)purines

JANSSEN PHARMACEUTICA NV122 citations98
US5041448AAug 20, 1991

(4-piperidinylmethyl and -hetero) purines

JANSSEN PHARMACEUTICA NV128 citations98
US4695575ASep 22, 1987

4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines

JANSSEN PHARMACEUTICA NV113 citations96
US5360807ANov 1, 1994

Substituted thiazolyl and substituted pyridinyl derivatives

JANSSEN PHARMACEUTICA NV22 citations92
US4835161AMay 30, 1989

Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines

JANSSEN PHARMACEUTICA NV32 citations92
US4634704AJan 6, 1987

Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines

JANSSEN PHARMACEUTICA NV33 citations92
US4588722AMay 13, 1986

N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives

JANSSEN PHARMACEUTICA NV38 citations92
US5468743ANov 21, 1995

Imidazo[2,1-b]benzazepine derivatives, compositions and method of use

JANSSEN PHARMACEUTICA NV32 citations91
US4988689AJan 29, 1991

((Pharmacologically active bicyclic heterocyclic)methyl and -heteroatom) substituted hexahydro-1H-azepines and pyrrolidines

JANSSEN PHARMACEUTICA NV31 citations90
US4695569ASep 22, 1987

Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines

JANSSEN PHARMACEUTICA NV29 citations89
USRE37886EOct 15, 2002

1-(1,2-Disubstituted piperidinyl)-4-substituted piperazine derivatives

JANSSEN PHARMACEUTICA NV30 citations88
US5086056AFeb 4, 1992

2-(heterocyclylalkyl)imidazopyridines

JANSSEN PHARMACEUTICA NV16 citations81
US4946843AAug 7, 1990

2-(heterocyclylalkyl)imidazopyridines

JANSSEN PHARMACEUTICA NV22 citations81
US4556660ADec 3, 1985

N-(Bicyclic heterocyclyl)-4-piperidinamines

JANSSEN PHARMACEUTICA NV23 citations81
US4943580AJul 24, 1990

Anti-histaminic benzimidazole, imidazopyridine and purine derivatives

JANSSEN PHARMACEUTICA NV8 citations73
US4861785AAug 29, 1989

Benzoxazol-and benzothiazolamine derivatives, useful as anti-anoxic agents

JANSSEN PHARMACEUTICA NV12 citations73
US4839374AJun 13, 1989

4-((Bicyclic heterocyclyl)-methyl and -hetero)-piperidines

JANSSEN PHARMACEUTICA NV11 citations73
US5629308AMay 13, 1997

Imidazo [1,2-A] (pyrrolo, thieno or furano) [2,3-D] azepine derivatives

JANSSEN PHARMACEUTICA NV7 citations72
US5272150ADec 21, 1993

Hydroxyalkylfuranyl derivatives

JANSSEN PHARMACEUTICA NV14 citations72
US4826848AMay 2, 1989

Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines

JANSSEN PHARMACEUTICA NV10 citations72
US4689330AAug 25, 1987

Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines

JANSSEN PHARMACEUTICA NV20 citations72
US5217980AJun 8, 1993

Oxazolyl and piperidinyl substituted benimidazolyl compounds

JANSSEN PHARMACEUTICA NV11 citations71
US5151424ASep 29, 1992

Pharmacologically active (Bicyclic heterocyclyl)methyl and -hetero) substituted hexahydro-1H-azepines and pyrrolidines

JANSSEN PHARMACEUTICA NV11 citations71
US5126339AJun 30, 1992

Anti-allergic bicyclic heterocyclyl-containing N-(bicyclic heterocyclyl)-4-piperidinamines

JANSSEN PHARMACEUTICA NV3 citations62
US5011842AApr 30, 1991

2-(heterocyclylalkyl)imidazopyridines for treating allergic diseases

JANSSEN PHARMACEUTICA NV4 citations62
US5010198AApr 23, 1991

Intermediates for the synthesis of benzoxazol- and benzothiazolamine derivatives, useful as anti-anoxic agents

JANSSEN PHARMACEUTICA NV3 citations62
US4897401AJan 30, 1990

N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives useful in treating allergic diseases

JANSSEN PHARMACEUTICA NV5 citations62
US4888426ADec 19, 1989

1-(5-methyl-furan-2-ylmethyl)-N-(4-piperidinyl)imidazo [4,5-6]pyridine-2-amine

JANSSEN PHARMACEUTICA NV2 citations62
US4820822AApr 11, 1989

Novel N-(bicyclic heterocyclyl)-4-piperidinamines

JANSSEN PHARMACEUTICA NV2 citations62
US5461050AOct 24, 1995

Imidazo[1,2-a](pyrrolo, thieno or furano) [3,2a-d]azepine derivatives, compositions and methods of use

JANSSEN PHARMACEUTICA NV6 citations61
US5008268AApr 16, 1991

2-aminopyrimidinone derivatives

JANSSEN PHARMACEUTICA NV4 citations61
US4749702AJun 7, 1988

Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines

JANSSEN PHARMACEUTICA NV4 citations61
US5278165AJan 11, 1994

Oxazolyl imidazol[4,5-b]pyridin and pyrimidine compounds

JANSSEN PHARMACEUTICA NV5 citations60
US5071846ADec 10, 1991

Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines

JANSSEN PHARMACEUTICA NV3 citations60
US4760074AJul 26, 1988

Novel-N-(bicyclic heterocyclyl)-4-piperidinamines

JANSSEN PHARMACEUTICA NV2 citations57
US5595988AJan 21, 1997

Triazolo(pyrrolo, thieno or furano)azepine derivatives

JANSSEN PHARMACEUTICA NV4 citations51
US5025014AJun 18, 1991

Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines as pharmaceuticals

JANSSEN PHARMACEUTICA NV2 citations47
US5006527AApr 9, 1991

Pharmacologically active N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives

JANSSEN PHARMACEUTICA NV0 citations34