Inventor
XUE CHU-BIAO
US59 patents
⚠️ This page may combine multiple inventors who share the name “XUE CHU-BIAO”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
INCYTE CORP
29 patentsUS9999619B2Jun 19, 2018
Piperidin-4-yl azetidine derivatives as JAK1 inhibitors
INCYTE CORP38 citations98
US9464088B2Oct 11, 2016
Piperidin-4-yl azetidine derivatives as JAK1 inhibitors
INCYTE CORP57 citations98
US9200004B2Dec 1, 2015
Thiazolecarboxamides and pyridinecarboxamide compounds useful as Pim kinase inhibitors
INCYTE CORP25 citations96
US11285140B2Mar 29, 2022
Piperidin-4-yl azetidine derivatives as JAK1 inhibitors
INCYTE CORP14 citations94
US10695337B2Jun 30, 2020
Piperidin-4-yl azetidine derivatives as JAK1 inhibitors
INCYTE CORP21 citations94
US9278950B2Mar 8, 2016
Bicyclic aromatic carboxamide compounds useful as Pim kinase inhibitors
INCYTE CORP24 citations94
US10265307B2Apr 23, 2019
Thiazolecarboxamides and pyridinecarboxamide compounds useful as Pim kinase inhibitors
INCYTE CORP10 citations93
US9849120B2Dec 26, 2017
Thiazolecarboxamides and pyridinecarboxamide compounds useful as Pim kinase inhibitors
INCYTE CORP12 citations93
US9676750B2Jun 13, 2017
Bicyclic aromatic carboxamide compounds useful as pim kinase inhibitors
INCYTE CORP18 citations93
US9550765B2Jan 24, 2017
Thiazolecarboxamides and pyridinecarboxamide compounds useful as Pim kinase inhibitors
INCYTE CORP19 citations93
US9556197B2Jan 31, 2017
Furo- and thieno-pyridine carboxamide compounds useful as pim kinase inhibitors
INCYTE CORP19 citations92
US10828290B2Nov 10, 2020
Thiazolecarboxamides and pyridinecarboxamide compounds useful as pim kinase inhibitors
INCYTE CORP3 citations84
US10517858B2Dec 31, 2019
Thiazolecarboxamides and pyridinecarboxamide compounds useful as PIM kinase inhibitors
INCYTE CORP6 citations84
US10000507B2Jun 19, 2018
Furo- and thieno-pyridine carboxamide compounds useful as pim kinase inhibitors
INCYTE CORP12 citations84
US7511050B2Mar 31, 2009
Purinone derivatives as HM74A agonists
INCYTE CORP14 citations84
US7307086B2Dec 11, 2007
3-(4-heteroarylcyclohexylamino)cyclopentanecarboxamides as modulators of chemokine receptors
INCYTE CORP21 citations84
US7576089B2Aug 18, 2009
3-cycloalkylaminopyrrolidine derivatives as modulators of chemokine receptors
INCYTE CORP8 citations83
US7985730B2Jul 26, 2011
3-aminopyrrolidine derivatives as modulators of chemokine receptors
INCYTE CORP6 citations74
US7834021B2Nov 16, 2010
3-aminopyrrolidine derivatives as modulators of chemokine receptors
INCYTE CORP4 citations74
US7678798B2Mar 16, 2010
Piperazinylpiperidine derivatives as chemokine receptor antagonists
INCYTE CORP5 citations74
US7462624B2Dec 9, 2008
Purinone derivatives as HM74a agonists
INCYTE CORP8 citations74
US11229631B2Jan 25, 2022
Thiazolecarboxamides and pyridinecarboxamide compounds useful as Pim kinase inhibitors
INCYTE CORP0 citations63
US7902205B2Mar 8, 2011
Purinone derivatives as HM74A agonists
INCYTE CORP3 citations63
US7700624B2Apr 20, 2010
3-aminocyclopentanecrboxamides as modulators of chemokine receptors
INCYTE CORP6 citations63
US7618970B2Nov 17, 2009
3-aminocyclopentanecarboxamides as modulators of chemokine receptors
INCYTE CORP5 citations63
US8362003B2Jan 29, 2013
3-aminopyrrolidine derivatives as modulators of chemokine receptors
INCYTE CORP2 citations62
US9067921B2Jun 30, 2015
Piperazinylpiperidine derivatives as chemokine receptor antagonists
INCYTE CORP0 citations52
US8039478B2Oct 18, 2011
Purinone derivatives as HM74A agonists
INCYTE CORP1 citations52
US7863285B2Jan 4, 2011
Purinone derivatives as HM74A agonists
INCYTE CORP1 citations52
BRISTOL MYERS SQUIBB PHARMA CO
9 patentsUS6429213B1Aug 6, 2002
Cyclic hydroxamic acids as metalloproteinase inhibitors
BRISTOL MYERS SQUIBB PHARMA CO95 citations97
US6858626B2Feb 22, 2005
Cyclic hydroxamic acid as metalloproteinase inhibitors
BRISTOL MYERS SQUIBB PHARMA CO66 citations96
US6906053B2Jun 14, 2005
Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme (TACE)
BRISTOL MYERS SQUIBB PHARMA CO33 citations91
US6890915B2May 10, 2005
Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme (TACE)
BRISTOL MYERS SQUIBB PHARMA CO32 citations91
US6689771B2Feb 10, 2004
Amide derivatives as inhibitors of matrix metalloproteinases, TNF-α, and aggrecanase
BRISTOL MYERS SQUIBB PHARMA CO14 citations84
US6984648B2Jan 10, 2006
Cyclic β-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-α
BRISTOL MYERS SQUIBB PHARMA CO15 citations82
US6743807B2Jun 1, 2004
Cyclic β-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-α
BRISTOL MYERS SQUIBB PHARMA CO15 citations82
US6825215B2Nov 30, 2004
1,1-disubstituted cyclic inhibitors of matrix metalloproteases and TNF-α
BRISTOL MYERS SQUIBB PHARMA CO5 citations63
US6642255B2Nov 4, 2003
1,2,-Disubstituted cyclic inhibitors of matrix metalloproteases and TNF-alpha
BRISTOL MYERS SQUIBB PHARMA CO5 citations61
DU PONT MERCK PHARMA
4 patentsUS5849736ADec 15, 1998
Isoxazoline and isoxazole fibrinogen receptor antagonists
DU PONT MERCK PHARMA70 citations94
US5563158AOct 8, 1996
Aromatic compounds containing basic and acidic termini useful as fibrinogen receptor antagonists
DU PONT MERCK PHARMA26 citations92
US5703092ADec 30, 1997
Hydroxamic acid compounds as metalloprotease and TNF inhibitors
DU PONT MERCK PHARMA58 citations90
US5691329ANov 25, 1997
Compounds containing basic and acidic termini useful as fibrinogen receptor antagonists
DU PONT MERCK PHARMA13 citations73
DU PONT PHARM CO
3 patentsUS6268379B1Jul 31, 2001
Substituted aryl hydroxamic acids as metalloproteinase inhibitors
DU PONT PHARM CO71 citations96
US6376665B1Apr 23, 2002
Amide derivatives as inhibitors of matrix metalloproteinases, TNF-α, and aggrecanase
DU PONT PHARM CO23 citations93
US6114328ASep 5, 2000
Isoxazoline and isoxazole fibrogen receptor antagonists
DU PONT PHARM CO27 citations90
HUANG TAISHENG
1 patentPFIZER
1 patentXUE CHU-BIAO
1 patentBRISTOL MYERS SQUIBB CO
1 patentZHENG CHANGSHENG
1 patentShowing the top 50 of 59 patents by PatentIndex Score.