Inventor
GRAHAM DONALD W
US44 patents
⚠️ This page may combine multiple inventors who share the name “GRAHAM DONALD W”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK & CO INC
35 patentsUS6849636B2Feb 1, 2005
Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1
MERCK & CO INC52 citations95
US5710275AJan 20, 1998
7β-substituted-4-aza-5α-androstan-3-ones as 5α-reductase inhibitors
MERCK & CO INC22 citations92
US5693809ADec 2, 1997
Substituted 4-aza-5α-androstan-ones as 5α-reductase inhibitors
MERCK & CO INC37 citations92
US5516779AMay 14, 1996
17β-substituted-6-azasteroid derivatives useful as 5α-reductase inhibitors
MERCK & CO INC35 citations92
US5510351AApr 23, 1996
Delta-17 and delta-20 olefinic and saturated 17 beta-substituted 4-aza-5 alpha-androstan-ones as 5 alpha reductase inhibitors useful in the prevention and treatment of hyperandrogenic disorders
MERCK & CO INC25 citations92
US5510485AApr 23, 1996
17-ester, amide, and ketone derivatives of 3-oxo-4-azasteroids as 5A-reductase inhibitors
MERCK & CO INC25 citations92
US5147868ASep 15, 1992
Thienamycin renal peptidase inhibitors
MERCK & CO INC36 citations92
US6090836AJul 18, 2000
Benzisoxazole-derived antidiabetic compounds
MERCK & CO INC24 citations91
US5595996AJan 21, 1997
7-substituted 4-aza cholanic acid derivatives and their use
MERCK & CO INC33 citations90
US4847271AJul 11, 1989
Antihypercholesterolemic β-lactones
MERCK & CO INC41 citations90
US7625937B2Dec 1, 2009
1H-benzo[F]indazol-5-YL derivatives as selective glucocorticoid receptor modulators
MERCK & CO INC11 citations83
US4806564AFeb 21, 1989
Antihypercholesterolemic beta-lactones
MERCK & CO INC22 citations82
US4407802AOct 4, 1983
6-Amidino-9-substituted benzyl purines
MERCK & CO INC13 citations74
US7282591B2Oct 16, 2007
1h-benzo{f}indazol-5-yl derivatives as selective glucocorticoid receptor modulators
MERCK & CO INC5 citations73
US5760045AJun 2, 1998
Delta-17 and delta-20 olefinic and saturated 17β-substituted-4-aza-5α-androstan-3-ones as 5α-reductase inhibitors useful in the prevention and treatment of hyperandrogenic disorders
MERCK & CO INC6 citations73
US5438061AAug 1, 1995
7-substituted-δ4-6-azasteroid derivatives as 5α-reductase inhibitors
MERCK & CO INC9 citations73
US5047420ASep 10, 1991
1,3-diaryl cyclopentanes and derivatives thereof as PAF antagonists
MERCK & CO INC18 citations73
US4816477AMar 28, 1989
Antihypercholesterolemic β-lactones
MERCK & CO INC15 citations73
US4173631ANov 6, 1979
7-Methyl-8-methylamino-10-(1'-D-ribityl)isoalloxazine
MERCK & CO INC10 citations73
US5741795AApr 21, 1998
16-substituted-6-aza-androsten-4-ene-3-ones as 5-α-reductase inhibitors
MERCK & CO INC14 citations71
US4094976AJun 13, 1978
Anticoccidial cyclicamino ethanols and esters thereof
MERCK & CO INC7 citations71
US5843953ADec 1, 1998
7-substituted 4-aza cholanic acid derivatives and their use
MERCK & CO INC6 citations70
US5621104AApr 15, 1997
Substituted 3-phenanthridinone derivatives as 5-alpha-reductase inhibitors
MERCK & CO INC4 citations63
US4752611AJun 21, 1988
Anticoccidial 1,2,3-trazole compounds
MERCK & CO INC3 citations63
US7411073B2Aug 12, 2008
Selective non-steroidal glucocorticoid receptor modulators
MERCK & CO INC5 citations62
US6048869AApr 11, 2000
Tricyclic compounds
MERCK & CO INC3 citations62
US5886005AMar 23, 1999
4-Aza-19-norandrostane derivatives
MERCK & CO INC3 citations62
US4079069AMar 14, 1978
5-Deazariboflavin and its derivatives
MERCK & CO INC3 citations62
US7504402B2Mar 17, 2009
Triazole derivatives as inhibitors of 11-β-hydroxysteroid dehydrogenase-1
MERCK & CO INC4 citations61
US4406902ASep 27, 1983
Dipeptidase inhibitors
MERCK & CO INC5 citations58
US4053602AOct 11, 1977
Compositions for treating coccidiosis containing 5-deazariboflavin and its derivatives
MERCK & CO INC0 citations52
US5132463AJul 21, 1992
1,3-diaryl cyclopentanes and derivatives thereof as PAF antagonists
MERCK & CO INC0 citations51
US4091094AMay 23, 1978
9-Azariboflavin and pharmaceutical composition containing same
MERCK & CO INC1 citations51
US4290966ASep 22, 1981
Process for the preparation of traumatin
MERCK & CO INC0 citations49
US7329683B2Feb 12, 2008
11-β-hydroxysteroid dehydrogenase 1 inhibitors useful for the treatment of diabetes, obesity and dyslipidemia
MERCK & CO INC0 citations37
MERCK SHARP & DOHME
3 patentsUS7732432B2Jun 8, 2010
17-carbamoyloxy cortisol derivatives as selective glucocorticoid receptor modulators
MERCK SHARP & DOHME4 citations62
US7662846B2Feb 16, 2010
Selective spirocyclic glucocorticoid receptor modulators
MERCK SHARP & DOHME0 citations41
US8026264B2Sep 27, 2011
Triazole derivatives as inhibitors of 11-β hydroxysteroid dehydrogenase-1
MERCK SHARP & DOHME0 citations40