Inventor
LU TIANBAO
US65 patents
⚠️ This page may combine multiple inventors who share the name “LU TIANBAO”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
DIMENSIONAL PHARM INC
30 patentsUS6037356AMar 14, 2000
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
DIMENSIONAL PHARM INC67 citations96
US5741819AApr 21, 1998
Arylsulfonylaminobenzene derivatives and the use thereof as factor Xa inhibitors
DIMENSIONAL PHARM INC57 citations96
US6706021B2Mar 16, 2004
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
DIMENSIONAL PHARM INC18 citations92
US6566379B1May 20, 2003
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
DIMENSIONAL PHARM INC13 citations92
US6521663B2Feb 18, 2003
Aminoguanidinyl- and Alkoxyguanidinyl-substituted phenyl acetamides as protease inhibitors
DIMENSIONAL PHARM INC18 citations92
US6350764B2Feb 26, 2002
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
DIMENSIONAL PHARM INC15 citations92
US6235778B1May 22, 2001
Aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC17 citations92
US6204263B1Mar 20, 2001
Pyrazinone protease inhibitors
DIMENSIONAL PHARM INC21 citations92
US5891909AApr 6, 1999
Amidinohydrazones as protease inhibitors
DIMENSIONAL PHARM INC39 citations90
US6326492B1Dec 4, 2001
Heterocyclic protease inhibitors
DIMENSIONAL PHARM INC25 citations89
US6900231B2May 31, 2005
Aminopyridyl-substituted phenyl acetamides as protease inhibitors
DIMENSIONAL PHARM INC15 citations84
US6420397B1Jul 16, 2002
Heteroaryl protease inhibitors and diagnostic imaging agents
DIMENSIONAL PHARM INC15 citations84
US6472399B2Oct 29, 2002
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
DIMENSIONAL PHARM INC13 citations82
US6245763B1Jun 12, 2001
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
DIMENSIONAL PHARM INC13 citations82
US6133315AOct 17, 2000
Amidino protease inhibitors
DIMENSIONAL PHARM INC12 citations82
US6034127AMar 7, 2000
Amidino protease inhibitors
DIMENSIONAL PHARM INC13 citations82
US6706765B2Mar 16, 2004
Aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC12 citations81
US6730783B2May 4, 2004
Process for preparing aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC9 citations74
US6514978B2Feb 4, 2003
Thromboresistant materials incorporating pyrazinone protease inhibitors
DIMENSIONAL PHARM INC11 citations74
US6417161B1Jul 9, 2002
Amino acid amidinohydrazones, alkoxyguanidines and aminoguanidines as protease inhibitors
DIMENSIONAL PHARM INC9 citations74
US6414020B2Jul 2, 2002
Amidino protease inhibitors
DIMENSIONAL PHARM INC4 citations74
US6344466B2Feb 5, 2002
Benzamide and sulfonamide substitued aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC13 citations74
US6344486B1Feb 5, 2002
Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC9 citations74
US6281206B1Aug 28, 2001
Amidino protease inhibitors
DIMENSIONAL PHARM INC8 citations74
US6225302B1May 1, 2001
Amidino protease inhibitors
DIMENSIONAL PHARM INC4 citations74
US6638931B1Oct 28, 2003
Aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC11 citations73
US6518310B2Feb 11, 2003
Aminoguanidines and alkoxyguanidines as protease inhibitors
DIMENSIONAL PHARM INC9 citations73
US6635637B2Oct 21, 2003
Cyclic oxyguanidine protease inhibitors
DIMENSIONAL PHARM INC9 citations71
US6476016B2Nov 5, 2002
Cyclic oxyguanidine pyrazinones as protease inhibitors
DIMENSIONAL PHARM INC12 citations71
US5612369AMar 18, 1997
Thrombin inhibitors
DIMENSIONAL PHARM INC16 citations71
JANSSEN PHARMACEUTICA NV
13 patentsUS8030305B2Oct 4, 2011
Triazolopyridazines as kinase modulators
JANSSEN PHARMACEUTICA NV24 citations91
US7829584B2Nov 9, 2010
Pyridines and pyridine N-oxides as modulators of thrombin
JANSSEN PHARMACEUTICA NV12 citations81
US10214493B2Feb 26, 2019
Indazole derivatives useful as glucagon receptor antagonists
JANSSEN PHARMACEUTICA NV3 citations72
US10000473B2Jun 19, 2018
Indazole derivatives useful as glucagon receptor antagonists
JANSSEN PHARMACEUTICA NV3 citations72
US10888550B2Jan 12, 2021
Pyrazole derivatives as MALT1 inhibitors
JANSSEN PHARMACEUTICA NV3 citations71
US7262210B2Aug 28, 2007
Fluorinated pyridine N-oxide thrombin modulators and process for N-oxidation of nitrogen containing heteroaryls
JANSSEN PHARMACEUTICA NV9 citations71
US10077261B2Sep 18, 2018
Imidazolin-5-one derivative useful as FASN inhibitors for the treatment of cancer
JANSSEN PHARMACEUTICA NV7 citations70
US10954214B2Mar 23, 2021
Pyrazole derivatives as MALT1 inhibitors
JANSSEN PHARMACEUTICA NV5 citations69
US7968725B2Jun 28, 2011
Pyridinyl modulators of γ-secretase
JANSSEN PHARMACEUTICA NV5 citations63
US11098016B2Aug 24, 2021
Indazole derivatives useful as glucagon receptor antagonists
JANSSEN PHARMACEUTICA NV0 citations62
US11040031B2Jun 22, 2021
Pyrazole derivatives as MALT1 inhibitors
JANSSEN PHARMACEUTICA NV2 citations60
US7786116B2Aug 31, 2010
2-amino-quinoline derivatives useful as inhibitors of β-secretase (BACE)
JANSSEN PHARMACEUTICA NV2 citations60
US7662824B2Feb 16, 2010
Acylhydrazones as kinase modulators
JANSSEN PHARMACEUTICA NV2 citations60
ORTHO MCNEIL PHARM INC
3 patentsUS7029654B2Apr 18, 2006
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
ORTHO MCNEIL PHARM INC9 citations74
US7030110B2Apr 18, 2006
Cyclic oxyguanidine pyrazinones as protease inhibitors
ORTHO MCNEIL PHARM INC8 citations71
US7402586B2Jul 22, 2008
Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
ORTHO MCNEIL PHARM INC4 citations70
LU TIANBAO
1 patent3-DIMENSIONAL PHARM INC
1 patentJANSSEN BIOTECH INC
1 patentSHANDONG LUBEI ENTPR GROUP COM
1 patentShowing the top 50 of 65 patents by PatentIndex Score.