Inventor
SCHAUS JOHN M
US79 patents
Patents
50 patentsUS5741789AApr 21, 1998
Compounds having effects on serotonin-related systems
LILLY CO ELI135 citations98
US5614523AMar 25, 1997
Compounds having effects on serotonin-related systems
LILLY CO ELI115 citations98
US5789402AAug 4, 1998
Compounds having effects on serotonin-related systems
LILLY CO ELI103 citations97
US5627196AMay 6, 1997
Compounds having effects on serotonin-related systems
LILLY CO ELI99 citations97
US6117882ASep 12, 2000
5-HT4 agonists and antagonists
LILLY CO ELI63 citations96
US5576321ANov 19, 1996
Compounds having effects on serotonin-related systems
LILLY CO ELI87 citations96
US5434174AJul 18, 1995
Isoxazole derivatives for the treatment of irritable bowel syndrome
LILLY CO ELI57 citations96
US5389687AFeb 14, 1995
Ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes
LILLY CO ELI49 citations96
US5654320AAug 5, 1997
Indazolecarboxamides
LILLY CO ELI69 citations95
US6069152AMay 30, 2000
5-HT4 agonists and antagonists
LILLY CO ELI31 citations92
US5340838AAug 23, 1994
Method of inhibiting gastric acid secretion with 2-phenylcyclopropylamines
LILLY CO ELI22 citations92
US5244911ASep 14, 1993
6-heterocyclic-4-amino-1,2,2a,3,4,5-hexahydrobenz(cd)indoles and pharmaceutical use thereof
LILLY CO ELI44 citations92
US5229410AJul 20, 1993
6-substituted-hexahydrobenz[cd]indoles
LILLY CO ELI25 citations92
US5026707AJun 25, 1991
Ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes
LILLY CO ELI23 citations92
US5286753AFeb 15, 1994
Ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes and pharmaceutical compositions thereof
LILLY CO ELI20 citations91
US5594034AJan 14, 1997
Method of inhibiting gastric acid secretion with 8-substituted-2-amino-1,2,3,4-tetrahydronapthalene
LILLY CO ELI13 citations82
US5096908AMar 17, 1992
Method of inhibiting gastric acid secretion
LILLY CO ELI18 citations82
US5637624AJun 10, 1997
Ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes and 3-aminochromanes
LILLY CO ELI11 citations74
US5594025AJan 14, 1997
Method of inhibiting gastric acid secretion with 5-substituted-3-aminochromane
LILLY CO ELI5 citations74
US5576352ANov 19, 1996
Method of inhibiting gastric acid secretion with aryloxypropanolamines
LILLY CO ELI6 citations74
US5457120AOct 10, 1995
Method of inhibiting gastric acid secretion with 4- amino-1, 3, 4, 5 tetrahydrobenzo [c,d]indoles
LILLY CO ELI5 citations74
US5258379ANov 2, 1993
Method of inhibiting gastric acid secretion with n-arylpiperazines
LILLY CO ELI16 citations74
US5158956AOct 27, 1992
Method of inhibiting gastric acid secretion with benzodioxanes
LILLY CO ELI15 citations74
US5057515AOct 15, 1991
Method for agonizing a dopamine receptor
LILLY CO ELI10 citations74
US5006525AApr 9, 1991
Dopamine agonists method
LILLY CO ELI12 citations74
US4659832AApr 21, 1987
Process for the preparation of octahydro-oxazolo [4,5-G]quinolines
LILLY CO ELI11 citations74
US6172073B1Jan 9, 2001
Compounds having effects on serotonin-related systems
LILLY CO ELI12 citations73
US5654324AAug 5, 1997
6-heterocyclic-4-amino-1,2,2A,3,4,5-hexahydrobenz[cd]indoles
LILLY CO ELI5 citations73
US5641794AJun 24, 1997
6-heterocyclic-4-amino-1,2,2a,3,4,5-hexahydrobenz[cd]indoles
LILLY CO ELI4 citations73
US5627199AMay 6, 1997
6-heterocyclic-4-amino-1,2,2A,3,4,5-hexahydrobenz [CD] indoles
LILLY CO ELI5 citations73
US5244912ASep 14, 1993
6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz(cd)indoles and pharmaceutical use thereof
LILLY CO ELI10 citations73
US5426229AJun 20, 1995
Ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes
LILLY CO ELI6 citations72
US5364856ANov 15, 1994
6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz[CD]indoles
LILLY CO ELI5 citations72
US4826986AMay 2, 1989
6-Oxo-trans-octa- and decahydroquinolines
LILLY CO ELI12 citations72
US5817676AOct 6, 1998
Indazolecarboxamides
LILLY CO ELI12 citations71
US5457121AOct 10, 1995
Cis-hexahydro-5-(1,2,3,4-tetrahydro-2-naphthalenyl)pyrrolo<3,4-c>pyrroles as inhibitors of serotonin reuptake
LILLY CO ELI5 citations63
US5229409AJul 20, 1993
6-substituted-tetrahydrobenz[cd]indoles
LILLY CO ELI4 citations63
US4977149ADec 11, 1990
Pyridoquinoline dopamine agonists, compositions and use
LILLY CO ELI2 citations63
US4939259AJul 3, 1990
2-oxo-pyrido[2,3-g]quinoline derivatives
LILLY CO ELI3 citations63
US4647667AMar 3, 1987
Octa- and deca-hydroquinoline intermediates
LILLY CO ELI5 citations63
US4567266AJan 28, 1986
Method of preparing octahydro-1H(and 2H)-pyrazolo[3,4-g]quinolines
LILLY CO ELI4 citations63
US4540787ASep 10, 1985
Method of preparing trans-D1-1-alkyl-6-oxodecahydroquinolines
LILLY CO ELI2 citations63
US4471121ASep 11, 1984
Method of resolving trans-d alpha-1-n-propyl-6-oxodecahydroquinoline and di-p-toluoyltartaric acid salts thereof
LILLY CO ELI3 citations63
US5798367AAug 25, 1998
Indazolecarboxamides
LILLY CO ELI4 citations62
US5656653AAug 12, 1997
6-heterocyclic-4-amino-1,2,2A,3,4,5-hexahydrobenz[cd]indoles
LILLY CO ELI2 citations62
US5643910AJul 1, 1997
6-heterocyclic-4-amino-1,2,2A,3,4,5-hexahydrobenz[CD]indoles
LILLY CO ELI1 citations62
US5347013ASep 13, 1994
6-heterocyclic-4-amino-1,2,2a,3,4,5-hexahydrobenz[cd]indoles
LILLY CO ELI2 citations62
US4778894AOct 18, 1988
6 oxo-decahydroquinolines
LILLY CO ELI5 citations62
US4596871AJun 24, 1986
Pyrazole-ring alkylated pyrazoloquinolines
LILLY CO ELI4 citations62
US4507478AMar 26, 1985
2-Mercaptopyrimidohexahydroquinolines and related compounds
LILLY CO ELI4 citations62
Showing the top 50 of 79 patents by PatentIndex Score.