Inventor
SMITH II LEON M
US36 patents
⚠️ This page may combine multiple inventors who share the name “SMITH II LEON M”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
BRISTOL MYERS SQUIBB CO
31 patentsUS8367709B2Feb 5, 2013
Dipeptide analogs as coagulation factor inhibitors
BRISTOL MYERS SQUIBB CO42 citations94
US9453018B2Sep 27, 2016
Pyrimidinones as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO13 citations92
US7626039B2Dec 1, 2009
Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO14 citations92
US9902742B2Feb 27, 2018
Macrocycles as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO5 citations84
US9611274B2Apr 4, 2017
Macrocycles as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO5 citations84
US9192607B2Nov 24, 2015
Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO7 citations84
US9108951B2Aug 18, 2015
Substituted 5,6,7,8-tetrahydro-1,6-naphthyridines as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO5 citations84
US9000172B2Apr 7, 2015
Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO7 citations84
US9944625B2Apr 17, 2018
Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO3 citations73
US11053247B2Jul 6, 2021
Pyrimidinones as factor XIA inhibitors
BRISTOL MYERS SQUIBB CO2 citations72
US10336754B2Jul 2, 2019
Pyrimidinones as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO2 citations72
US9777001B2Oct 3, 2017
Macrocycles with aromatic P2′ groups as factor xia inhibitors
BRISTOL MYERS SQUIBB CO3 citations72
US10336730B2Jul 2, 2019
Substituted glycine derived FXIA inhibitors
BRISTOL MYERS SQUIBB CO1 citations63
US12428421B2Sep 30, 2025
Pyrimidinones as factor XIA inhibitors
BRISTOL MYERS SQUIBB CO0 citations62
US10899743B2Jan 26, 2021
Substituted glycine derived FXIA inhibitors
BRISTOL MYERS SQUIBB CO0 citations62
US10000466B2Jun 19, 2018
Substituted 4,5,6,7-tetrahydropyrazolo[3,4-c]pyridines as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO1 citations62
US9447110B2Sep 20, 2016
Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO1 citations62
US10611776B2Apr 7, 2020
Spiroheptane salicylamides and related compounds as inhibitors of rock
BRISTOL MYERS SQUIBB CO1 citations61
US10208021B2Feb 19, 2019
Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations52
US9725435B2Aug 8, 2017
Substituted 4,5,6,7-tetrahydropyrazolo[4,3-c]pyridines as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations52
US9394276B2Jul 19, 2016
Substituted 1,2,3,4-tetrahydro-2,6-naphthyridines as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations52
US9108981B2Aug 18, 2015
Cyclic P1 linkers as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations52
US9951071B2Apr 24, 2018
Dihydropyridone P1 as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations51
US9409908B2Aug 9, 2016
Dihydropyridone p1 as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO1 citations51
US10829501B2Nov 10, 2020
Spiroheptane salicylamides and related compounds as inhibitors of ROCK
BRISTOL MYERS SQUIBB CO0 citations50
US9738655B2Aug 22, 2017
Tetrahydroisoquinolines containing substituted azoles as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO1 citations49
US10160750B2Dec 25, 2018
Diamide macrocycles as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations42
US9403774B2Aug 2, 2016
Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors
BRISTOL MYERS SQUIBB CO0 citations42
US9315519B2Apr 19, 2016
Guanidine substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations42
US10273236B2Apr 30, 2019
Macrocyclic factor XIa inhibitors bearing heterocyclic groups
BRISTOL MYERS SQUIBB CO0 citations41
US9079929B2Jul 14, 2015
Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
BRISTOL MYERS SQUIBB CO0 citations41
PINTO DONALD J P
3 patentsUS9221818B2Dec 29, 2015
Macrocycles as factor XIa inhibitors
PINTO DONALD J P13 citations92
US8604056B2Dec 10, 2013
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors
PINTO DONALD J P0 citations51
US8252830B2Aug 28, 2012
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors
PINTO DONALD J P0 citations51