Inventor
CASTRO PINEIRO JOSE LUIS
GB49 patents
⚠️ This page may combine multiple inventors who share the name “CASTRO PINEIRO JOSE LUIS”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK SHARP & DOHME
41 patentsUS6756511B2Jun 29, 2004
Gamma-secretase inhibitors
MERCK SHARP & DOHME83 citations96
US6486153B1Nov 26, 2002
Phenylindole derivatives as 5-HT2A receptor ligands
MERCK SHARP & DOHME57 citations94
US7183303B2Feb 27, 2007
Gamma-secretase inhibitors
MERCK SHARP & DOHME33 citations92
US7049296B2May 23, 2006
Gamma-secretase inhibitors
MERCK SHARP & DOHME47 citations92
US6579875B1Jun 17, 2003
Triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME22 citations92
US6500828B1Dec 31, 2002
Triazolo-pyridazine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME18 citations92
US6337331B1Jan 8, 2002
Triazolo-pyrimidine as ligands for GABA receptors
MERCK SHARP & DOHME21 citations92
US6255305B1Jul 3, 2001
Substituted triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME49 citations92
US5681833AOct 28, 1997
Benzodiazepine derivatives
MERCK SHARP & DOHME50 citations92
US5854268ADec 29, 1998
Azetidine, pyrrolidine and piperidine derivatives
MERCK SHARP & DOHME45 citations91
US7030128B2Apr 18, 2006
Imidazo-pyrimidine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME11 citations84
US5977116ANov 2, 1999
Piperazine, piperidine and tetrahydropyridine derivatives
MERCK SHARP & DOHME19 citations84
US6828322B2Dec 7, 2004
Triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME14 citations83
US6593325B1Jul 15, 2003
Pyrido-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME15 citations83
US6140347AOct 31, 2000
Azetidine, pyrrolidine and piperidine derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME18 citations83
US6025374AFeb 15, 2000
Azetidine, pyrrolidine and piperidine derivatives as 5HT1 receptor agonists
MERCK SHARP & DOHME20 citations83
US7105509B2Sep 12, 2006
Benzodiazepine derivatives as APP modulators
MERCK SHARP & DOHME21 citations82
US6489343B2Dec 3, 2002
Tetrahydropyran derivatives and their use as therapeutic agents
MERCK SHARP & DOHME9 citations73
US6479506B1Nov 12, 2002
Triazolo-pyridine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME13 citations73
US6333336B1Dec 25, 2001
Pyrazolo-pyridine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME13 citations73
US6630471B1Oct 7, 2003
Substituted triazolo-pyridazine derivative, pharmaceutical compositions made therefrom
MERCK SHARP & DOHME12 citations70
US7300955B2Nov 27, 2007
Method and materials for treatment of Alzheimer's disease
MERCK SHARP & DOHME5 citations63
US7105507B2Sep 12, 2006
Cyclohexane derivatives and their use as therapeutic agents
MERCK SHARP & DOHME4 citations62
US5837715ANov 17, 1998
3-fluoro-4-aminopiperidine derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME2 citations62
US5807857ASep 15, 1998
Piperazine, piperidine and tetrahydropyridine derivative of indol-3-alkyl as 5-HT1D-α agonists
MERCK SHARP & DOHME6 citations62
US7626056B2Dec 1, 2009
Cyclohexanesulfonyl derivatives as GlyT1 inhibitors to treat schizophrenia
MERCK SHARP & DOHME5 citations61
US7226926B2Jun 5, 2007
8-fluoroimidazo 1,2-a pyridine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME5 citations61
US7595344B2Sep 29, 2009
Sulphones which modulate the action of gamma secretase
MERCK SHARP & DOHME2 citations60
US6110915AAug 29, 2000
Antiemetic use of triazolo-pyridazine derivatives
MERCK SHARP & DOHME4 citations58
US7485640B2Feb 3, 2009
Imidazopyrazinones as GABA-A receptor anxiolytics
MERCK SHARP & DOHME1 citations52
US7435748B2Oct 14, 2008
Gamma-secretase inhibitors
MERCK SHARP & DOHME1 citations52
US7851638B2Dec 14, 2010
Cyclohexanesulfonyl derivatives as GLYT1 inhibitors to treat schizophrenia
MERCK SHARP & DOHME0 citations50
US7598386B2Oct 6, 2009
Sulphones which modulate the action of gamma-secretase
MERCK SHARP & DOHME0 citations50
US7468393B2Dec 23, 2008
Diarylsulfones as 5-HT2A antagonists
MERCK SHARP & DOHME1 citations49
US6051572AApr 18, 2000
Azetidine, pyrrolidine and piperidine derivatives
MERCK SHARP & DOHME0 citations42
US7265110B2Sep 4, 2007
Tetrahydropyran derivatives and their use as therapeutic agents
MERCK SHARP & DOHME0 citations41
US7253205B2Aug 7, 2007
Gem-disubstituted cyclohexane derivatives and their use as therapeutic agents
MERCK SHARP & DOHME0 citations41
US6906085B2Jun 14, 2005
Tetrahydropyran derivatives as neurokinin receptor antagonists
MERCK SHARP & DOHME0 citations41
US6150391ANov 21, 2000
Diazabicyclo-octane derivatives as 5-HT receptor ligands
MERCK SHARP & DOHME0 citations41
US6048878AApr 11, 2000
Substituted piperidine derivatives as selective agonists of 5-HT receptors
MERCK SHARP & DOHME0 citations41
US7371771B2May 13, 2008
Alkenyl-substituted spirocyclic sulfamides as inhibitors of gamma-secretase
MERCK SHARP & DOHME0 citations40