Inventor
STREET LESLIE JOSEPH
GB54 patents
⚠️ This page may combine multiple inventors who share the name “STREET LESLIE JOSEPH”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK SHARP & DOHME
48 patentsUS7176203B2Feb 13, 2007
Imidazo-triazine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME63 citations97
US6476030B1Nov 5, 2002
Pyrazolo-triazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME70 citations94
US6642229B2Nov 4, 2003
3-Phenyl-imidazo-pyrimidine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME21 citations92
US6617326B2Sep 9, 2003
Imidazo-triazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME21 citations92
US6579875B1Jun 17, 2003
Triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME22 citations92
US6500828B1Dec 31, 2002
Triazolo-pyridazine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME18 citations92
US6337331B1Jan 8, 2002
Triazolo-pyrimidine as ligands for GABA receptors
MERCK SHARP & DOHME21 citations92
US6255305B1Jul 3, 2001
Substituted triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME49 citations92
US6200975B1Mar 13, 2001
Substituted 1,2,4-triazolo[3,4-a]phthalazine derivatives as GABA alpha 5 ligands
MERCK SHARP & DOHME42 citations92
US5854268ADec 29, 1998
Azetidine, pyrrolidine and piperidine derivatives
MERCK SHARP & DOHME45 citations91
US6936608B2Aug 30, 2005
Imidazo-triazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME20 citations90
US7030128B2Apr 18, 2006
Imidazo-pyrimidine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME11 citations84
US6914063B2Jul 5, 2005
Imidazo-pyrazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME14 citations84
US6730676B2May 4, 2004
Pyrazino-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME13 citations84
US6444666B1Sep 3, 2002
Triazolopyridazine Derivatives for treating anxiety and enhancing cognition
MERCK SHARP & DOHME15 citations84
US6211219B1Apr 3, 2001
Aminocyclohexane derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME18 citations84
US6914065B2Jul 5, 2005
Imidazo[1,2-C]pyrimidine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME12 citations83
US6900215B2May 31, 2005
Imidazo-pyrimidine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME16 citations83
US6872720B2Mar 29, 2005
Pyrazolo-triazine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME13 citations83
US6828322B2Dec 7, 2004
Triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME14 citations83
US6730681B2May 4, 2004
Triazolo-pyrimidine derivatives as ligands for gaba receptors
MERCK SHARP & DOHME18 citations83
US6699859B1Mar 2, 2004
Triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME13 citations83
US6593325B1Jul 15, 2003
Pyrido-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME15 citations83
US6140347AOct 31, 2000
Azetidine, pyrrolidine and piperidine derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME18 citations83
US6025374AFeb 15, 2000
Azetidine, pyrrolidine and piperidine derivatives as 5HT1 receptor agonists
MERCK SHARP & DOHME20 citations83
US6541484B2Apr 1, 2003
Pyrazolo-pyridine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME19 citations82
US6303597B1Oct 16, 2001
Triazolo-pyridazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME12 citations74
US6608062B1Aug 19, 2003
Imidazo-triazine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME12 citations73
US6479506B1Nov 12, 2002
Triazolo-pyridine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME13 citations73
US6333336B1Dec 25, 2001
Pyrazolo-pyridine derivatives as ligands for GABA receptors
MERCK SHARP & DOHME13 citations73
US5981529ANov 9, 1999
Substituted indolylpropyl-piperazine derivatives as 5-HT1D α agonists
MERCK SHARP & DOHME13 citations73
US6465462B1Oct 15, 2002
Substituted triazolo pyridazine derivatives as inverse agonists of the GABAAα5 receptor subtype
MERCK SHARP & DOHME9 citations72
US6630471B1Oct 7, 2003
Substituted triazolo-pyridazine derivative, pharmaceutical compositions made therefrom
MERCK SHARP & DOHME12 citations70
US6969716B2Nov 29, 2005
5-phenyl[1,2,4]triazines as ligands for GABA-A α2/α3 receptors for treating anxiety or depression
MERCK SHARP & DOHME6 citations62
US6297235B1Oct 2, 2001
Triazolopyridazine derivatives for treating anxiety and enhancing cognition
MERCK SHARP & DOHME6 citations62
US6127388AOct 3, 2000
Azetidine, pyrrolidine and piperidine derivatives as 5-HT1D receptor agonists
MERCK SHARP & DOHME6 citations62
US5998416ADec 7, 1999
Piperazine, piperidine and tetrahydropyridine derivatives as 5-HT receptor agonists
MERCK SHARP & DOHME2 citations62
US5998415ADec 7, 1999
Bicyclic heteroaryl-alkylene-(homo)piperazinones and thione analogues thereof, their preparation, and their use of as selective agonists of 5-HT1 -like receptors
MERCK SHARP & DOHME6 citations62
US5925638AJul 20, 1999
Substituted 1-indolylpropyl-4-benzylpiperazine derivatives
MERCK SHARP & DOHME4 citations62
US5919783AJul 6, 1999
Indoline and azaindoline derivatives as 5-HT1D alpha receptor agonists
MERCK SHARP & DOHME4 citations62
US5807857ASep 15, 1998
Piperazine, piperidine and tetrahydropyridine derivative of indol-3-alkyl as 5-HT1D-α agonists
MERCK SHARP & DOHME6 citations62
US7626056B2Dec 1, 2009
Cyclohexanesulfonyl derivatives as GlyT1 inhibitors to treat schizophrenia
MERCK SHARP & DOHME5 citations61
US6960598B2Nov 1, 2005
(1,8) naphthyridines as gaba ligands, their pharmaceutical compositions and uses
MERCK SHARP & DOHME2 citations61
US5854247ADec 29, 1998
Piperazine, piperidine and tetrahydropyridine derivatives useful as 5-HT1 recepter agonists
MERCK SHARP & DOHME6 citations59
US7485640B2Feb 3, 2009
Imidazopyrazinones as GABA-A receptor anxiolytics
MERCK SHARP & DOHME1 citations52
US6448249B1Sep 10, 2002
Substituted 1,2,4-triazolo[3,4-A]phthalazine derivatives as GABAα5 ligands
MERCK SHARP & DOHME1 citations52
US5902819AMay 11, 1999
Triazole derivatives
MERCK SHARP & DOHME1 citations51
US5889008AMar 30, 1999
Substituted 1-indolylpropyl-4-phenethylpiperazadine derivatives
MERCK SHARP & DOHME1 citations51
MERCK SHARPE & DOHME LTD
1 patentMERCK SHARPE & DOHME
1 patentShowing the top 50 of 54 patents by PatentIndex Score.