Inventor
KULAGOWSKI JANUSZ JOZEF
GB51 patents
⚠️ This page may combine multiple inventors who share the name “KULAGOWSKI JANUSZ JOZEF”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK SHARP & DOHME
36 patentsUS6172077B1Jan 9, 2001
Spiro-azacyclic derivatives and their use as therapeutic agents
MERCK SHARP & DOHME149 citations97
US5714498AFeb 3, 1998
Benzimidazole derivatives
MERCK SHARP & DOHME61 citations96
US6114315ASep 5, 2000
Use of NK-1 receptor antagonists for treating major depressive disorders with anxiety
MERCK SHARP & DOHME26 citations92
US5977104ANov 2, 1999
Use of NK-1 receptor antagonists for treating bipolar disorders
MERCK SHARP & DOHME29 citations92
US5952315ASep 14, 1999
Use of NK-1 receptor antagonists for treating bipolar disorders
MERCK SHARP & DOHME34 citations92
US5792768AAug 11, 1998
Antipsychotic benzimidazole derivatives
MERCK SHARP & DOHME40 citations92
US5780475AJul 14, 1998
Antipsychotic indazole derivatives
MERCK SHARP & DOHME30 citations92
US5712285AJan 27, 1998
Pyrrolo-pyridine derivatives
MERCK SHARP & DOHME48 citations92
US5700809ADec 23, 1997
Pyrrolo-pyridine derivatives
MERCK SHARP & DOHME49 citations92
US6225320B1May 1, 2001
Spiro-azacyclic derivatives and their use as therapeutic agents
MERCK SHARP & DOHME24 citations90
US7638629B2Dec 29, 2009
Piperidines and related compounds for treatment of alzheimer's disease
MERCK SHARP & DOHME13 citations83
US6071928AJun 6, 2000
Spiro-piperidine derivatives and their use as therapeutic agents
MERCK SHARP & DOHME21 citations83
US6372754B1Apr 16, 2002
Spirocyclic ketones and their use as tachykinin antagonists
MERCK SHARP & DOHME11 citations74
US6271230B1Aug 7, 2001
Use of NK-1 receptor antagonists for treating cognitive disorders
MERCK SHARP & DOHME6 citations74
US6071927AJun 6, 2000
Spiro-piperidine derivatives and their use as therapeutic agents
MERCK SHARP & DOHME13 citations74
US5925627AJul 20, 1999
Use of NK-1 receptor antagonists for treating movement disorders
MERCK SHARP & DOHME7 citations74
US5700802ADec 23, 1997
Furopyridine derivatives
MERCK SHARP & DOHME12 citations74
US6100256AAug 8, 2000
Use of NK-1 receptors antagonists for treating schizophrenic disorders
MERCK SHARP & DOHME7 citations73
US5849765ADec 15, 1998
Tetrahydropyridine derivatives as dopamine receptor subtype ligands
MERCK SHARP & DOHME14 citations73
US5814644ASep 29, 1998
Indole derivatives as dopamine D4 antagonists
MERCK SHARP & DOHME16 citations73
US5665732ASep 9, 1997
Indazole derivatives
MERCK SHARP & DOHME17 citations73
US5665722ASep 9, 1997
Benzofuran derivatives as D4 receptor antagonists
MERCK SHARP & DOHME11 citations71
US6087348AJul 11, 2000
Use of NK-1 receptor antagonists for treating stress disorders
MERCK SHARP & DOHME3 citations63
US5919781AJul 6, 1999
Use of NK-1 receptor antogonists for treating substance use disorders
MERCK SHARP & DOHME5 citations63
US5700941ADec 23, 1997
Octahydronaphthyridine derivatives
MERCK SHARP & DOHME4 citations63
US6613766B1Sep 2, 2003
Pentaaza-cyclopental[a]naphthalene derivatives as ligands for GABAa α5 receptors
MERCK SHARP & DOHME2 citations62
US6727249B2Apr 27, 2004
Azabicyclic ether derivatives and their use as therapeutic agents
MERCK SHARP & DOHME4 citations61
US7101892B2Sep 5, 2006
Sulfone derivatives as 5-HT7 receptor ligands
MERCK SHARP & DOHME2 citations60
US6555552B2Apr 29, 2003
Azabicyclic amine derivatives and their use as therapeutic agents
MERCK SHARP & DOHME3 citations59
US6096729AAug 1, 2000
Use of NK-1 receptor antagonists for treating amnestic disorders
MERCK SHARP & DOHME0 citations52
US6613765B1Sep 2, 2003
Use of NK-1 receptor antagonists for treating major depressive disorders
MERCK SHARP & DOHME0 citations51
US5861407AJan 19, 1999
Tetrahydropyridine derivatives as dopamine receptor subtype ligands
MERCK SHARP & DOHME1 citations50
US5641787AJun 24, 1997
Indole derivatives as dopamine D4 antagonists
MERCK SHARP & DOHME1 citations50
US5681836AOct 28, 1997
Methanesulfonate salts of antipsychotic benzofuran derivatives
MERCK SHARP & DOHME0 citations42
US7276607B2Oct 2, 2007
5-HT7 receptor antagonists
MERCK SHARP & DOHME0 citations40
US6479486B2Nov 12, 2002
Azabicyclic spiroether derivatives and their use as therapeutic agents
MERCK SHARP & DOHME0 citations39
JANSSEN PHARMACEUTICA NV
9 patentsUS11236084B2Feb 1, 2022
Substituted azaindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11186589B2Nov 30, 2021
Cyanoindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11180487B2Nov 23, 2021
Substituted cyanoindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11136311B2Oct 5, 2021
Heteroaromatic derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11001569B2May 11, 2021
6-membered heteroaromatic substituted cyanoindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US10005773B2Jun 26, 2018
1-(4-pyrimidinyl)-1H-pyrrolo[3,2-c]pyridine derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations40
US10005776B2Jun 26, 2018
Compounds as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations40
US9981963B2May 29, 2018
3-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-c]pyridine derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations39
US9981962B2May 29, 2018
Pyrazole derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations38
MERCK SHARP
1 patentBLENCH TOBY JONATHAN
1 patentMERCH SHARP & DOHME LTD
1 patentCHIESI FARMA SPA
1 patentHOFFMANN LA ROCHE
1 patentShowing the top 50 of 51 patents by PatentIndex Score.