Inventor
CHORVAT ROBERT J
US54 patents
⚠️ This page may combine multiple inventors who share the name “CHORVAT ROBERT J”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SEARLE & CO
19 patentsUS4704382ANov 3, 1987
Phenylpiperazine phosphonates
SEARLE & CO44 citations92
US4230626AOct 28, 1980
25-Halocholest-5-ene-3β,22-diols and esters thereof
SEARLE & CO12 citations74
US3991061ANov 9, 1976
Azanaphthaleneacetic acid derivatives
SEARLE & CO9 citations74
US4680295AJul 14, 1987
Octahydropyrido[1,2-c]pyrimidinones and hexahydropyrido[1,2-c]pyrimidinediones
SEARLE & CO4 citations63
US4560754ADec 24, 1985
Substituted 5-phenyl-5-(aminoalkyl)-1,3-diazabicyclo[4.4.0]decan-4-ones and 5-phenyl-5-(aminoalkyl)-1,3-diazabicyclo[4.4.0]dec-2-en-4-ones
SEARLE & CO3 citations63
US4329295AMay 11, 1982
24-Cyclopropylcholene-3β, 22-diols and esters thereof
SEARLE & CO3 citations63
US4299774ANov 10, 1981
25-Alkylcholest-5-ene-3 β,22-diols and esters thereof
SEARLE & CO2 citations63
US4223136ASep 16, 1980
2,3-Dihydro-3-oxo-5H-pyrido[3,4-b][1,4]-benzothiazine-4-carbonitriles
SEARLE & CO6 citations63
US5097035AMar 17, 1992
Monobasic disobutamide derivatives
SEARLE & CO2 citations62
US4639524AJan 27, 1987
Monobasic disobutamide derivatives
SEARLE & CO5 citations62
US4356302AOct 26, 1982
4H-1,4-Benzothiazine derivatives
SEARLE & CO2 citations58
US4567270AJan 28, 1986
Hexahydroindolizinones useful for treating cardiac arrhythmia, thrombotic disorders in mammals
SEARLE & CO2 citations54
US4554353ANov 19, 1985
2,5-Pyrrolidinedione derivatives useful as antiarrhythmic agents
SEARLE & CO1 citations52
US4348328ASep 7, 1982
25-Substituted-5α-cholestane-3β,22S-diol
SEARLE & CO1 citations52
US4053476AOct 11, 1977
7-aza-6-alkoxy-1-tetralones
SEARLE & CO0 citations52
US4012391AMar 15, 1977
11β-Alkyl-2-azaestratrienes and intermediates
SEARLE & CO0 citations52
US4007194AFeb 8, 1977
Process and intermediates for manufacture of 2-azasterioids
SEARLE & CO0 citations52
US4791199ADec 13, 1988
Process for antiarrhythmic 1,3-diazabicyclo[4.4.0]dec-2-en-4-ones
SEARLE & CO1 citations47
US4399279AAug 16, 1983
4H-1,4-Benzothiazine derivatives and intermediates thereto
SEARLE & CO0 citations47
MCELROY JOHN F
10 patentsUS8133904B2Mar 13, 2012
Cannabinoid receptor antagonists/inverse agonists useful for treating obesity
MCELROY JOHN F26 citations92
US8334282B2Dec 18, 2012
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F8 citations83
US8138216B2Mar 20, 2012
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F11 citations83
US8088809B2Jan 3, 2012
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F13 citations83
US8580768B2Nov 12, 2013
Cannabinoid receptor antagonists-inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F5 citations72
US8252791B2Aug 28, 2012
Purine compounds as cannabinoid receptor blockers
MCELROY JOHN F3 citations62
US8236821B2Aug 7, 2012
Substituted N-phenyl-5-phenyl-pyrazolin-3-yl amides as cannabinoid receptor antagonists/inverse agonists useful for treating obesity
MCELROY JOHN F5 citations62
US8853252B2Oct 7, 2014
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F1 citations51
US8648072B2Feb 11, 2014
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F0 citations51
US8217038B2Jul 10, 2012
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
MCELROY JOHN F1 citations51
JENRIN DISCOVERY INC
4 patentsUS7655685B2Feb 2, 2010
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
JENRIN DISCOVERY INC51 citations97
US7666889B2Feb 23, 2010
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
JENRIN DISCOVERY INC15 citations92
US7687481B2Mar 30, 2010
Cannabinoid receptor antagonists/inverse agonists useful for treating obesity
JENRIN DISCOVERY INC13 citations82
US7649115B2Jan 19, 2010
MAO-B inhibitors useful for treating obesity
JENRIN DISCOVERY INC0 citations51
JENRIN DISCOVERY
3 patentsUS9987253B2Jun 5, 2018
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
JENRIN DISCOVERY8 citations83
US9517228B2Dec 13, 2016
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
JENRIN DISCOVERY8 citations83
US9133127B2Sep 15, 2015
Cannabinoid receptor antagonists/inverse agonists useful for treating disease conditions, including metabolic disorders and cancers
JENRIN DISCOVERY0 citations51
SEARLE G D &
3 patentsUS4193930AMar 18, 1980
25-Alkyl-3β-hydroxycholest-5-en-7-ones and esters thereof
SEARLE G D &12 citations74
US4180666ADec 25, 1979
3,9-Dihydro-3,9-dioxo-2H-indeno(2,1-c)-pyridine-4-(carbonitriles/carboxamides)
SEARLE G D &8 citations74
US4205004AMay 27, 1980
25-Alkylcholest-5-ene-3β,22-diols and esters thereof
SEARLE G D &2 citations63
MCELROY JOHN FRANCIS
3 patentsUS8138209B2Mar 20, 2012
Substituted picolinamides as MAO-B inhibitors useful for treating obesity
MCELROY JOHN FRANCIS5 citations55
US8541475B2Sep 24, 2013
MAO-B inhibitors useful for treating obesity
MCELROY JOHN FRANCIS0 citations49
US8088798B2Jan 3, 2012
Cannabinoid receptor antagonists/inverse agonists useful for treating obesity
MCELROY JOHN FRANCIS0 citations49
ACAD PHARMACEUTICALS INCORPORATED
2 patentsACAD PHARMACEUTICALS INC
2 patentsJENRIN DISCOVERY LLC
2 patentsUS11179370B2Nov 23, 2021
Cannabinoid receptor antagonists/inverse agonists useful for treating disease conditions, including metabolic disorders and cancers
JENRIN DISCOVERY LLC0 citations58
US10617673B2Apr 14, 2020
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
JENRIN DISCOVERY LLC0 citations48
G D SERLE & CO
1 patentJENRM DISCOVERY INC
1 patentShowing the top 50 of 54 patents by PatentIndex Score.