Inventor
SINCLAIR PETER J
US40 patents
⚠️ This page may combine multiple inventors who share the name “SINCLAIR PETER J”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK & CO INC
25 patentsUS5258389ANov 2, 1993
O-aryl, O-alkyl, O-alkenyl and O-alkynylrapamycin derivatives
MERCK & CO INC432 citations99
US7652049B2Jan 26, 2010
CETP inhibitors
MERCK & CO INC54 citations96
US6852727B2Feb 8, 2005
Benzimisazo[4,5-f]isoquinolinone derivatives
MERCK & CO INC192 citations96
US6498165B1Dec 24, 2002
Src kinase inhibitor compounds
MERCK & CO INC238 citations96
US6329380B1Dec 11, 2001
SRC kinase inhibitor compounds
MERCK & CO INC87 citations96
US6316444B1Nov 13, 2001
SRC kinase inhibitor compounds
MERCK & CO INC120 citations96
US5532248AJul 2, 1996
O-aryl,O-alkyl, and O-alkenyl-macrolides having immunosuppressive activity
MERCK & CO INC66 citations96
US5719296AFeb 17, 1998
Pseudopeptide lactam inhibitors of peptide binding to MHC class II proteins
MERCK & CO INC112 citations95
US5208241AMay 4, 1993
N-heteroaryl, n-alkylheteroaryl, n-alkenylheteroaryl and n-alkynylheteroarylmacrolides having immunosuppressive activity
MERCK & CO INC63 citations94
US5344925ASep 6, 1994
Imidazolidyl macrolides having immunosuppressive activity
MERCK & CO INC20 citations92
US5310901AMay 10, 1994
O-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynlheteroarylrapamycin derivatives
MERCK & CO INC25 citations92
US5262533ANov 16, 1993
Amino O-aryl macrolides having immunosuppressive activity
MERCK & CO INC35 citations92
US5252732AOct 12, 1993
D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity
MERCK & CO INC47 citations92
US5250678AOct 5, 1993
O-aryl, O-alkyl, O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
MERCK & CO INC39 citations92
US5247076ASep 21, 1993
Imidazolidyl macrolides having immunosuppressive activity
MERCK & CO INC45 citations92
US5057499AOct 15, 1991
Avermectin derivatives
MERCK & CO INC23 citations92
US6809199B2Oct 26, 2004
(Halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
MERCK & CO INC47 citations89
US5693648ADec 2, 1997
O-aryl, O-alkyl, O-alkenyl and O-alkynyl-macrolides having immunosuppressive activity
MERCK & CO INC20 citations84
US6022890AFeb 8, 2000
Immunosuppressant tetracyclic triterpenes
MERCK & CO INC11 citations74
US5877184AMar 2, 1999
Macrolides having immunosuppressive activity
MERCK & CO INC9 citations74
US5030622AJul 9, 1991
Avermectin derivatives
MERCK & CO INC11 citations74
US4897383AJan 30, 1990
Avermectin derivatives
MERCK & CO INC7 citations74
US5565560AOct 15, 1996
O-Aryl,O-alkyl,O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
MERCK & CO INC14 citations73
US5349061ASep 20, 1994
O-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity
MERCK & CO INC17 citations73
US4978656ADec 18, 1990
Synthetic derivatives of paraherquamide
MERCK & CO INC8 citations70
MERCK SHARP & DOHME
6 patentsUS7915271B2Mar 29, 2011
1,3-oxazolidin-2-one derivatives useful as CETP inhibitors
MERCK SHARP & DOHME15 citations84
US7910592B2Mar 22, 2011
CETP inhibitors
MERCK SHARP & DOHME13 citations84
US7781426B2Aug 24, 2010
CETP inhibitors
MERCK SHARP & DOHME18 citations82
US7737295B2Jun 15, 2010
CETP inhibitors
MERCK SHARP & DOHME15 citations82
US9403807B2Aug 2, 2016
Mineralocorticoid receptor antagonists
MERCK SHARP & DOHME0 citations50
US7935727B2May 3, 2011
CETP inhibitors
MERCK SHARP & DOHME0 citations41
ALI AMJAD
5 patentsUS8735435B2May 27, 2014
CETP inhibitors
ALI AMJAD5 citations80
US8865707B2Oct 21, 2014
Cholesteryl ester transfer protein inhibitors
ALI AMJAD6 citations72
US8334290B2Dec 18, 2012
CETP inhibitors
ALI AMJAD5 citations60
US8440702B2May 14, 2013
1,3-oxazolidin -2-one derivatives useful as CETP inhibitors
ALI AMJAD1 citations51
US8193365B2Jun 5, 2012
CETP inhibitors
ALI AMJAD1 citations48
HUNT JULIANNE A
3 patentsUS8445480B2May 21, 2013
CETP inhibitors derived from benzoxazole arylamides
HUNT JULIANNE A15 citations81
US8436028B2May 7, 2013
CETP inhibitors derived from benzoxazole arylamides
HUNT JULIANNE A18 citations81
US8293721B2Oct 23, 2012
CETP inhibitors derived from benzoxazole arylamides
HUNT JULIANNE A6 citations71