Inventor
TAODA YOSHIYUKI
JP32 patents
⚠️ This page may combine multiple inventors who share the name “TAODA YOSHIYUKI”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SHIONOGI & CO
19 patentsUS8778943B2Jul 15, 2014
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-α]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides
SHIONOGI & CO30 citations95
US7858788B2Dec 28, 2010
Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity
SHIONOGI & CO47 citations94
US9051337B2Jun 9, 2015
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides
SHIONOGI & CO27 citations92
US10927129B2Feb 23, 2021
N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity
SHIONOGI & CO3 citations83
US9815835B2Nov 14, 2017
Substituted polycyclic carbamolypyridone derivative
SHIONOGI & CO11 citations83
US9469638B2Oct 18, 2016
Substituted polycyclic carbamoylpyridone derivative
SHIONOGI & CO9 citations83
US9273065B2Mar 1, 2016
Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors
SHIONOGI & CO3 citations83
US9758515B2Sep 12, 2017
Substituted polycyclic carbamoyl pyridone derivative prodrug
SHIONOGI & CO13 citations81
US11453669B2Sep 27, 2022
Polycyclic pyridone derivative
SHIONOGI & CO2 citations73
US11267823B2Mar 8, 2022
Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1′,2′:4,5]pyrazino[1,2-a]pyrrolo[1,2-c]pyrimidines having HIV integrase inhibitory activity
SHIONOGI & CO2 citations72
US10202379B2Feb 12, 2019
Substituted polycyclic carbamoyl pyridone derivative prodrug
SHIONOGI & CO4 citations71
US11814368B2Nov 14, 2023
Triazine derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same
SHIONOGI & CO3 citations68
US12139489B2Nov 12, 2024
Polycyclic carbamoylpyridone derivative
SHIONOGI & CO0 citations59
US11649236B2May 16, 2023
Polycyclic carbamoylpyridone derivative
SHIONOGI & CO0 citations59
US7745453B2Jun 29, 2010
Hydroxypyrimidinone derivatives having inhibitory activity against HIV integrase
SHIONOGI & CO4 citations56
US12559474B2Feb 24, 2026
Triazine derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same
SHIONOGI & CO0 citations55
US9365587B2Jun 14, 2016
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates
SHIONOGI & CO0 citations51
US8754214B2Jun 17, 2014
Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates
SHIONOGI & CO0 citations51
US8691823B2Apr 8, 2014
Prodrugs of (4aS, 13ar)-N-[(2,4-difluorophenyl)methyl]-10-hydroxy-9-11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1H-pyrido[1,2-a]pyrrolo[1′,2′:3:4]imidazo[1,2-d]pyrazine-8-carboxamide and their use in the treatment of HIV infection
SHIONOGI & CO0 citations49
JOHNS BRIAN ALVIN
3 patentsUS8129385B2Mar 6, 2012
Substituted 5-hydroxy-3,4,6,9,9a, 10-hexanhydro-2h-1-oxa04a,8a-diaza-anthracene-6,10-dioness
JOHNS BRIAN ALVIN66 citations97
US8410103B2Apr 2, 2013
(3S,11aR)-N-[2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydro[1,3]oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide useful as anti-HIV agent
JOHNS BRIAN ALVIN33 citations95
US8183372B2May 22, 2012
Substituted 9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydor-1H-pyrido[1,2-a]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazines
JOHNS BRIAN ALVIN0 citations51