P

Inventor

TAODA YOSHIYUKI

JP32 patents
⚠️ This page may combine multiple inventors who share the name “TAODA YOSHIYUKI”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.

SHIONOGI & CO

19 patents
US8778943B2Jul 15, 2014

Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-α]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides

SHIONOGI & CO30 citations95
US7858788B2Dec 28, 2010

Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity

SHIONOGI & CO47 citations94
US9051337B2Jun 9, 2015

Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides

SHIONOGI & CO27 citations92
US10927129B2Feb 23, 2021

N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity

SHIONOGI & CO3 citations83
US9815835B2Nov 14, 2017

Substituted polycyclic carbamolypyridone derivative

SHIONOGI & CO11 citations83
US9469638B2Oct 18, 2016

Substituted polycyclic carbamoylpyridone derivative

SHIONOGI & CO9 citations83
US9273065B2Mar 1, 2016

Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors

SHIONOGI & CO3 citations83
US9758515B2Sep 12, 2017

Substituted polycyclic carbamoyl pyridone derivative prodrug

SHIONOGI & CO13 citations81
US11453669B2Sep 27, 2022

Polycyclic pyridone derivative

SHIONOGI & CO2 citations73
US11267823B2Mar 8, 2022

Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1′,2′:4,5]pyrazino[1,2-a]pyrrolo[1,2-c]pyrimidines having HIV integrase inhibitory activity

SHIONOGI & CO2 citations72
US10202379B2Feb 12, 2019

Substituted polycyclic carbamoyl pyridone derivative prodrug

SHIONOGI & CO4 citations71
US11814368B2Nov 14, 2023

Triazine derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same

SHIONOGI & CO3 citations68
US12139489B2Nov 12, 2024

Polycyclic carbamoylpyridone derivative

SHIONOGI & CO0 citations59
US11649236B2May 16, 2023

Polycyclic carbamoylpyridone derivative

SHIONOGI & CO0 citations59
US7745453B2Jun 29, 2010

Hydroxypyrimidinone derivatives having inhibitory activity against HIV integrase

SHIONOGI & CO4 citations56
US12559474B2Feb 24, 2026

Triazine derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same

SHIONOGI & CO0 citations55
US9365587B2Jun 14, 2016

Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates

SHIONOGI & CO0 citations51
US8754214B2Jun 17, 2014

Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates

SHIONOGI & CO0 citations51
US8691823B2Apr 8, 2014

Prodrugs of (4aS, 13ar)-N-[(2,4-difluorophenyl)methyl]-10-hydroxy-9-11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1H-pyrido[1,2-a]pyrrolo[1′,2′:3:4]imidazo[1,2-d]pyrazine-8-carboxamide and their use in the treatment of HIV infection

SHIONOGI & CO0 citations49

JOHNS BRIAN ALVIN

3 patents

YOSHIDA HIROSHI

2 patents

UNIV HOKKAIDO NAT UNIV CORP

2 patents

PURDUE PHARMA LP

2 patents

TAKAHASHI CHIKA

1 patent

AKIYAMA TOSHIYUKI

1 patent

FUCHINO KOUKI

1 patent

KAI HIROYUKI

1 patent