Inventor
LACHAPELLE ERIK ALPHIE
US24 patents
Patents
24 patentsUS9428523B2Aug 30, 2016
2-amino-6-methyl-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8H)-yl-1,3-thiazol-4-yl amides
PFIZER12 citations92
US9315520B2Apr 19, 2016
2-amino-6-methyl-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8H)-yl-1,3-thiazol-4-yl amides
PFIZER15 citations92
US9045499B2Jun 2, 2015
Heteroaryl-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
PFIZER17 citations92
US8865706B2Oct 21, 2014
Heteroaryl-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
PFIZER19 citations92
US9403846B2Aug 2, 2016
Carbocyclic- and heterocyclic-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
PFIZER7 citations84
US9192612B2Nov 24, 2015
Heteroaryl-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
PFIZER13 citations84
US9605007B2Mar 28, 2017
2-amino-6-methyl-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8H)-yl-1,3-thiazol-4-yl amides
PFIZER8 citations83
US9598421B2Mar 21, 2017
Imidazopyridazine compounds
PFIZER6 citations83
US10738063B2Aug 11, 2020
6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-2-carboxamide compounds
PFIZER3 citations72
US10604519B2Mar 31, 2020
5,7-dihydro-pyrrolo-pyridine derivatives
PFIZER3 citations72
US10028962B2Jul 24, 2018
2-amino-6-methy1-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8H)-yl-1,3-thiazol-4-yl amides
PFIZER3 citations72
US9744173B2Aug 29, 2017
2-amino 6-methyl-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8H)-yl-1,3-thiazol-4-yl amides
PFIZER2 citations72
US11472805B2Oct 18, 2022
Tricyclic compounds and their use as phosphodiesterase inhibitors
PFIZER4 citations71
US11339159B2May 24, 2022
Toll-like receptor agonists
PFIZER2 citations71
US11905284B2Feb 20, 2024
5,7-dihydro-pyrrolo-pyridine derivatives
PFIZER0 citations62
US10323042B2Jun 18, 2019
6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-2-carboxamide compounds
PFIZER1 citations62
US12398119B2Aug 26, 2025
Piperazine azaspiro derivatives
PFIZER0 citations60
US12049465B2Jul 30, 2024
Tricyclic compounds and their use as phosphodiesterase inhibitors
PFIZER0 citations60
US11976064B2May 7, 2024
Toll-like receptor agonists
PFIZER0 citations60
US11524954B2Dec 13, 2022
Piperazine azaspiro derivatives
PFIZER0 citations60
US10669279B2Jun 2, 2020
Imidazopyridazine compounds
PFIZER0 citations51
US10077269B2Sep 18, 2018
Imidazopyridazine compounds
PFIZER1 citations51
US11198692B2Dec 14, 2021
Dihydro-pyrrolo-pyridine derivatives
PFIZER0 citations49
US10131669B2Nov 20, 2018
Pyrazolopyrimidine compounds
PFIZER0 citations41