Inventor
GILBERT ADAM MATTHEW
US24 patents
⚠️ This page may combine multiple inventors who share the name “GILBERT ADAM MATTHEW”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
PFIZER
13 patentsUS9845301B2Dec 19, 2017
1,1,1-trifluoro-3-hydroxypropan-2-yl carbamate derivatives and 1,1,1-trifluoro-4-hydroxybutan-2-yl carbamate derivatives as MAGL inhibitors
PFIZER8 citations83
US9617258B2Apr 11, 2017
Pyrrolo[2,3-d]pyrimidinyl, pyrrolo[2,3-b]pyrazinyl and pyrrolo[2,3-d]pyridinyl acrylamides
PFIZER13 citations82
US10604519B2Mar 31, 2020
5,7-dihydro-pyrrolo-pyridine derivatives
PFIZER3 citations72
US10428034B2Oct 1, 2019
1,1,1-trifluoro-3-hydroxypropan-2-yl carbamate derivatives and 1,1,1-trifluoro-4-hydroxybutan-2-yl carbamate derivatives as MAGL inhibitors
PFIZER3 citations72
US10328082B2Jun 25, 2019
Methods of use and combinations
PFIZER4 citations69
US9328104B2May 3, 2016
Selective androgen receptor modulators
PFIZER4 citations68
US11905284B2Feb 20, 2024
5,7-dihydro-pyrrolo-pyridine derivatives
PFIZER0 citations62
US12077533B2Sep 3, 2024
Pyrrolo[2,3-d]pyrimidinyl, pyrrolo[2,3-b]pyrazinyl and pyrrolo[2,3-d]pyridinyl acrylamides
PFIZER0 citations61
US11111242B2Sep 7, 2021
Pyrrolo[2,3-d]pyrimidinyl, pyrrolo[2,3-b]pyrazinyl and pyrrolo[2,3-d]pyridinyl acrylamides
PFIZER0 citations61
US10723711B2Jul 28, 2020
1,1,1-trifluoro-3-hydroxypropan-2-yl carbamate derivatives and 1,1,1-trifluoro-4-hydroxybutan-2-yl carbamate derivatives as MAGL inhibitors
PFIZER0 citations51
US10703756B2Jul 7, 2020
Pyrrolo[2,3-D]pyrimidinyl, pyrrolo[2,3-B]pyrazinyl, pyrrolo[2,3-B]pyridinyl acrylamides and epoxides thereof
PFIZER0 citations51
US11198692B2Dec 14, 2021
Dihydro-pyrrolo-pyridine derivatives
PFIZER0 citations49
US11712480B2Aug 1, 2023
Heteroaryl sulfone-based conjugation handles, methods for their preparation, and their use in synthesizing antibody drug conjugates
PFIZER0 citations43
AMERICAN HOME PROD
5 patentsUS6133273AOct 17, 2000
Pyrazolopyrimidine-2,4-dione sulfonamides
AMERICAN HOME PROD63 citations92
US6172222B1Jan 9, 2001
Diaminopyrazoles
AMERICAN HOME PROD14 citations80
US6221874B1Apr 24, 2001
Method of treating bone loss by stimulation of calcitonin
AMERICAN HOME PROD2 citations60
US6319941B1Nov 20, 2001
Diaminopyrazoles
AMERICAN HOME PROD0 citations50
US6313149B1Nov 6, 2001
Diaminopyrazoles
AMERICAN HOME PROD0 citations50
PELLICCIARI ROBERTO
3 patentsUS8299090B2Oct 30, 2012
Thiazolyl-and oxazolyl-isoquinolinones and methods for using them
PELLICCIARI ROBERTO3 citations61
US9079915B2Jul 14, 2015
Thienyl- and furanyl-isoquinolinones and methods for using them
PELLICCIARI ROBERTO0 citations47
US8633215B2Jan 21, 2014
Thienyl-and furanyl-isoquinolinones and methods for using them
PELLICCIARI ROBERTO0 citations47