Inventor
BARTOSZYK GERD
DE48 patents
⚠️ This page may combine multiple inventors who share the name “BARTOSZYK GERD”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK PATENT GMBH
45 patentsUS5532241AJul 2, 1996
Piperidines and piperazines
MERCK PATENT GMBH139 citations98
US6251908B1Jun 26, 2001
Piperazine derivatives
MERCK PATENT GMBH42 citations93
US5418237AMay 23, 1995
Indole derivatives
MERCK PATENT GMBH31 citations93
US5242925ASep 7, 1993
Piperazinylbenzodioxane derivatives
MERCK PATENT GMBH23 citations93
US6395780B1May 28, 2002
Cleavage system inhibitors as potential antipsychotics
MERCK PATENT GMBH19 citations92
US6258813B1Jul 10, 2001
D4 receptor selectivity piperazine derivatives
MERCK PATENT GMBH29 citations92
US5776972AJul 7, 1998
Kappa-opiate agonists for inflammatory bowel disorders
MERCK PATENT GMBH26 citations92
US5767132AJun 16, 1998
Pyridyl chroman
MERCK PATENT GMBH49 citations92
US5472961ADec 5, 1995
Acetamides
MERCK PATENT GMBH30 citations92
US5693655ADec 2, 1997
3-indolylpiperidines
MERCK PATENT GMBH29 citations91
US5670511ASep 23, 1997
Indolepiperidine derivatives
MERCK PATENT GMBH27 citations91
US5532266AJul 2, 1996
Acrylacetamides
MERCK PATENT GMBH37 citations91
US6509340B1Jan 21, 2003
Amide and urea derivatives as 5-HT reuptake inhibitors and as 5-HT1B/1D ligands
MERCK PATENT GMBH30 citations90
US6310068B1Oct 30, 2001
Benzonitriles and benzofluorides
MERCK PATENT GMBH27 citations90
US5232978AAug 3, 1993
1-(2-arylethyl)-pyrrolidines
MERCK PATENT GMBH36 citations90
US7572796B2Aug 11, 2009
Substituted indoles
MERCK PATENT GMBH13 citations84
US7566709B2Jul 28, 2009
1,3,4-Substituted pyrazoles as 5-HT receptor antagonists for the treatment of psychoses and neurological disorders
MERCK PATENT GMBH11 citations84
US6723725B1Apr 20, 2004
Indole derivatives
MERCK PATENT GMBH14 citations83
US7642261B2Jan 5, 2010
Use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
MERCK PATENT GMBH10 citations82
US6462056B1Oct 8, 2002
Oxazolidines as 5-HT2A-antagonists
MERCK PATENT GMBH6 citations74
US5714502AFeb 3, 1998
Piperidinylmethyloxazolidinones
MERCK PATENT GMBH8 citations74
US5561145AOct 1, 1996
4-aryloxy- and 4-arylthiopiperidine derivatives
MERCK PATENT GMBH7 citations74
US6441013B1Aug 27, 2002
Sulphonyloxazolamines as therapeutic active ingredients
MERCK PATENT GMBH12 citations73
US5977161ANov 2, 1999
Kappa-opiate agonists effective in the treatment of postoperative ileus
MERCK PATENT GMBH8 citations73
US6900212B1May 31, 2005
Use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
MERCK PATENT GMBH10 citations71
US7968551B2Jun 28, 2011
Chromenoneindoles
MERCK PATENT GMBH3 citations63
US7960413B2Jun 14, 2011
Pyrazole compounds
MERCK PATENT GMBH6 citations63
US7829565B2Nov 9, 2010
Indole derivatives as serotonin reuptake inhibitors
MERCK PATENT GMBH3 citations63
US7432282B2Oct 7, 2008
Pyridinalkyl-aminoalkyl-IH-indole derivatives having an inhibitory action on 5-HT and serotonin reuptake as antidepressants and anxiolytics
MERCK PATENT GMBH2 citations63
US7329749B2Feb 12, 2008
Piperazinylcarbonylquinolines and -isoquinolines
MERCK PATENT GMBH3 citations62
US7244846B2Jul 17, 2007
Substituted benzofuran-2-carboxamides derivatives
MERCK PATENT GMBH6 citations62
US6960599B2Nov 1, 2005
Heterocyclic aminoalkylpyridine derivatives as psychopharmaceuticals
MERCK PATENT GMBH4 citations62
US6756370B1Jun 29, 2004
Piperidine alcohols
MERCK PATENT GMBH4 citations62
US6548516B1Apr 15, 2003
1-(3-heteroarylpropyl- or -prop-2-enyl)-4-benzylpiperidines used as NMDA receptor antagonists
MERCK PATENT GMBH2 citations62
US7482465B2Jan 27, 2009
Indol derivatives and their use as 5-HT ligands
MERCK PATENT GMBH2 citations61
US7425574B2Sep 16, 2008
Benzofuran oxyethylamines as antidepressants and anxiolytics
MERCK PATENT GMBH2 citations61
US6413989B1Jul 2, 2002
Piperidinylmethyloxazolidinone derivative
MERCK PATENT GMBH2 citations59
US7262216B2Aug 28, 2007
Benzofuran compounds and their use as antidepressants and anxiolytics
MERCK PATENT GMBH1 citations52
US7928128B2Apr 19, 2011
Use of(R)-(−) -2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane and its physiologically acceptable salts
MERCK PATENT GMBH0 citations51
US7371756B2May 13, 2008
Use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
MERCK PATENT GMBH0 citations50
US7479492B2Jan 20, 2009
Use combined 5-HT1A agonists and selective serotonin reuptake inhibitors
MERCK PATENT GMBH0 citations49
US7253202B2Aug 7, 2007
Substituted benzodioxepines
MERCK PATENT GMBH1 citations48
US7872030B2Jan 18, 2011
Use of 2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane and its physiologically acceptable salts
MERCK PATENT GMBH0 citations47
US7842695B2Nov 30, 2010
Substituted pyrazole compounds
MERCK PATENT GMBH0 citations41
US7618988B2Nov 17, 2009
Use of substituted aminomethyl chromans
MERCK PATENT GMBH0 citations38