Inventor
SACH GEORGE S
30 patents
Patents
30 patentsUS4532252AJul 30, 1985
3,5-Substituted-2-pyridylalkylamino compounds having histamine H1 -antagonist activity
SMITH KLINE FRENCH LAB19 citations82
US4863936ASep 5, 1989
3,5-Substituted-2-pyridyl-alkylaminocyclobutenediones having histamine h1 -antagonist activity
SMITH KLINE FRENCH LAB15 citations74
US4665078AMay 12, 1987
2-(3-amino-5-halo-2-pyridylalkylamino)-pyrimidones useful as histamine H1-antagonists
SMITH KLINE FRENCH LAB14 citations74
US4640926AFeb 3, 1987
3,5-Substituted-2-pyridylalkylaminothiadiazoles having histamine H1 -antagonist activity
SMITH KLINE FRENCH LAB12 citations74
US4535163AAug 13, 1985
2-Aminoalkyl-pyridine derivatives
SMITH KLINE FRENCH LAB4 citations74
US4486434ADec 4, 1984
Histamine H1 -antagonists
SMITH KLINE FRENCH LAB6 citations74
US4444772AApr 24, 1984
Histamine H1 -antagonists
SMITH KLINE FRENCH LAB5 citations74
US4385058AMay 24, 1983
Pyrimidone derivatives
SMITH KLINE FRENCH LAB11 citations74
US4215126AJul 29, 1980
Alkoxy pyridine compounds
SMITH KLINE FRENCH LAB5 citations74
US4156727AMay 29, 1979
Alkoxy pyridine compounds
SMITH KLINE FRENCH LAB11 citations74
US4154838AMay 15, 1979
Alkoxy pyridine
SMITH KLINE FRENCH LAB12 citations74
US4894372AJan 16, 1990
Pyridine compounds which have useful histamine-H2 antagonist activity
SMITH KLINE FRENCH LAB2 citations63
US4758576AJul 19, 1988
Pyridine derivatives and use as histamine H2 antagonists
SMITH KLINE FRENCH LAB1 citations63
US4584381AApr 22, 1986
5-(Nitro or halogen)-3-(alkyl)-2-(aminoalkyl)pyridines
SMITH KLINE FRENCH LAB1 citations63
US4574126AMar 4, 1986
Pyridine derivatives histamine H2 -antagonists
SMITH KLINE FRENCH LAB3 citations63
US4551466ANov 5, 1985
Pyridyl-2-oxy-propyl-1H-1,2,4-triazole-3,5-diamines
SMITH KLINE FRENCH LAB1 citations63
US4537891AAug 27, 1985
2-(3,5-Substituted-2-pyridylalkylamino)-5-benzyl-4-pyrimidones
SMITH KLINE FRENCH LAB4 citations63
US4537890AAug 27, 1985
2-(3,5-Substituted-2-pyridylalkylamino)-5-oxopyridylmethyl-4-pyrimidones useful as histamine H1 -antagonists
SMITH KLINE FRENCH LAB3 citations63
US4439609AMar 27, 1984
Pyridines
SMITH KLINE FRENCH LAB2 citations63
US4426526AJan 17, 1984
Alkoxypyridyl alkylamines
SMITH KLINE FRENCH LAB1 citations63
US4374839AFeb 22, 1983
Pharmacologically active 1,3-bis[(2-heterocyclyl-methyl-thio)ethyl)ethyl)guanidino]alkane derivatives
SMITH KLINE FRENCH LAB1 citations63
US4282224AAug 4, 1981
Alkoxy-pyridyl substituted alkanes
SMITH KLINE FRENCH LAB1 citations63
US4269844AMay 26, 1981
Alkoxypyridyl N-cyano or N-carbamoylguanidino alkanes, compositions containing same and uses thereof
SMITH KLINE FRENCH LAB1 citations63
US4264608AApr 28, 1981
Pharmacologically active compounds
SMITH KLINE FRENCH LAB1 citations63
US4139624AFeb 13, 1979
Alkoxypyridyl substituted alkanes
SMITH KLINE FRENCH LAB2 citations63
US4771058ASep 13, 1988
3,4-diamino-1,2,5-thiadiazole-1-oxides having histamine H1 -antagonist activity
SMITH KLINE FRENCH LAB0 citations52
US4727076AFeb 23, 1988
Tetrahydroquinolinylalkyl amino pyridones and ring homologues thereof, useful as histamine-H1 -receptor antagonists
SMITH KLINE FRENCH LAB0 citations52
US4607107AAug 19, 1986
(4-aminoalkyl-2-pyridyl alkyl)guanidines
SMITH KLINE FRENCH LAB1 citations52
US4219553AAug 26, 1980
Alkoxy pyridyl substituted alkanes
SMITH KLINE FRENCH LAB1 citations52
US4210652AJul 1, 1980
Pharmacologically active 1,3-bis[1-(2-heteroalkylthio)ethylamino)-2-nitrovinyl-1-amino]propane derivatives
SMITH KLINE FRENCH LAB1 citations52