Inventor
GRAHAM SAMUEL L
US52 patents
⚠️ This page may combine multiple inventors who share the name “GRAHAM SAMUEL L”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
MERCK & CO INC
46 patentsUS5872136AFeb 16, 1999
Arylheteroaryl inhibitors of farnesyl-protein transferase
MERCK & CO INC115 citations98
US5852010ADec 22, 1998
Inhibitors of farnesyl-protein transferase
MERCK & CO INC101 citations98
US6297239B1Oct 2, 2001
Inhibitors of prenyl-protein transferase
MERCK & CO INC67 citations96
US6077853AJun 20, 2000
Inhibitors of farnesyl-protein transferase
MERCK & CO INC65 citations96
US5965578AOct 12, 1999
Inhibitors of farnesyl-protein transferase
MERCK & CO INC89 citations96
US5340828AAug 23, 1994
Inhibitors of farnesyl protein transferase
MERCK & CO INC71 citations96
US5238922AAug 24, 1993
Inhibitors of farnesyl protein transferase
MERCK & CO INC105 citations96
US5352705AOct 4, 1994
Inhibitors of farnesyl protein transferase
MERCK & CO INC65 citations95
US5585359ADec 17, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC76 citations94
US7205293B2Apr 17, 2007
Benodiazepine spirohydantoin CGRP receptor antagonists
MERCK & CO INC28 citations93
US5998407ADec 7, 1999
Inhibitors of farnesyl-protein transferase
MERCK & CO INC22 citations93
US5859015AJan 12, 1999
N-heterocyclic piperazinyl and H-heterocyclic piperazinonyl inhibitors of farnesyl-protein transferase
MERCK & CO INC49 citations93
US5736539AApr 7, 1998
Inhibitors of farnesyl-protein transferase
MERCK & CO INC39 citations93
US5491164AFeb 13, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC46 citations93
US5439918AAug 8, 1995
Inhibitors of farnesyl-protein transferase
MERCK & CO INC38 citations93
US4668697AMay 26, 1987
Elevated intraocular pressure lowering benzo-[b]-thiophene-2-sulfonamide derivatives, compositions, and method of use therefor
MERCK & CO INC40 citations93
US7034026B2Apr 25, 2006
Inhibitors of Akt activity
MERCK & CO INC43 citations92
US6562823B1May 13, 2003
Inhibitors of prenyl-protein transferase
MERCK & CO INC23 citations92
US6103723AAug 15, 2000
Inhibitors of farnesyl-protein transferase
MERCK & CO INC50 citations92
US5661161AAug 26, 1997
Inhibitors of farnesyl-protein transferase
MERCK & CO INC30 citations92
US5504212AApr 2, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC53 citations92
US5470832ANov 28, 1995
Inhibitors of geranylgeranyl-protein transferase
MERCK & CO INC23 citations91
US5326773AJul 5, 1994
Inhibitors of farnesyl-protein transferase
MERCK & CO INC54 citations91
US6127366AOct 3, 2000
Inhibitors of farnesyl-protein transferase
MERCK & CO INC54 citations90
US6284755B1Sep 4, 2001
Inhibitors of prenyl-protein transferase
MERCK & CO INC16 citations84
US6500841B1Dec 31, 2002
Inhibitors of farnesyl-protein transferase
MERCK & CO INC7 citations74
US5571835ANov 5, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC16 citations74
US5536750AJul 16, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC14 citations74
US5523456AJun 4, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC11 citations74
US5480893AJan 2, 1996
Inhibitors of farnesyl protein transferase
MERCK & CO INC14 citations74
US4840963AJun 20, 1989
2-Sulfamoyl-1H-indole derivatives for the treatment of elevated intraocular pressure
MERCK & CO INC14 citations74
US4665090AMay 12, 1987
Substituted thiophene-2-sulfonamide antiglaucoma agents
MERCK & CO INC7 citations74
US4544667AOct 1, 1985
2-Sulfamoylbenzo[b]furan derivatives for the treatment of elevated intraocular pressure
MERCK & CO INC8 citations74
US4795811AJan 3, 1989
Intermediates for preparing HMG-CoA reductase inhibitors
MERCK & CO INC9 citations72
US5468733ANov 21, 1995
Inhibitors of farnesyl-protein transferase
MERCK & CO INC18 citations71
US4847289AJul 11, 1989
Thiophene sulfonamide antiglaucoma agents
MERCK & CO INC13 citations71
US5652257AJul 29, 1997
Heterocycle-containing inhibitors of farnesyl-protein transferase
MERCK & CO INC3 citations63
US4788192ANov 29, 1988
2-Sulfamoylbenzo(b)thiophene derivatives pharmaceutical compositions and use
MERCK & CO INC2 citations63
US4721794AJan 26, 1988
Substituted thiophene-2-sulfonamide antiglaucoma agents
MERCK & CO INC2 citations63
US4510155AApr 9, 1985
6(or 5)-Hydroxybenzothiazole-2-sulfonamide-O-sulfate salts for the topical treatment of elevated intraocular pressure
MERCK & CO INC3 citations63
US6333335B1Dec 25, 2001
Phenyl-protein transferase inhibitors
MERCK & CO INC1 citations52
US5703241ADec 30, 1997
Inhibitor of farnesyl-protein transferase
MERCK & CO INC0 citations52
US5753650AMay 19, 1998
Inhibitors of farnesyl-protein transferase
MERCK & CO INC0 citations51
US5504115AApr 2, 1996
Inhibitors of farnesyl protein transferase
MERCK & CO INC1 citations51
US4812463AMar 14, 1989
Alkanesulfonamides as antiglaucoma agents
MERCK & CO INC1 citations51
US5576293ANov 19, 1996
Inhibitors of farnesyl-protein transferase
MERCK & CO INC1 citations50
MERCK SHARP & DOHME
2 patentsSLOAN KETTERING INST CANCER
1 patentCOBURN CRAIG A
1 patentShowing the top 50 of 52 patents by PatentIndex Score.