Inventor
HAUSKE JAMES R
US48 patents
⚠️ This page may combine multiple inventors who share the name “HAUSKE JAMES R”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SEPRACOR INC
31 patentsUS7294637B2Nov 13, 2007
Method of treating addiction or dependence using a ligand for a monamine receptor or transporter
SEPRACOR INC89 citations97
US7132551B2Nov 7, 2006
Ligands for monoamine receptors and transporters, and methods of use thereof
SEPRACOR INC45 citations96
US6992077B2Jan 31, 2006
Spirocyclic ligands for sigma receptors, and libraries and methods of use thereof
SEPRACOR INC43 citations96
US6476019B1Nov 5, 2002
Spirocyclic ligands for sigma receptors, and libraries and methods of use thereof
SEPRACOR INC42 citations96
US6180640B1Jan 30, 2001
Di- and tetra-hydroquinoline-indole antimicrobial agents, uses and compositions related thereto
SEPRACOR INC60 citations95
US6762177B2Jul 13, 2004
Spirocyclic ligands for sigma receptors, and libraries and methods of use thereof
SEPRACOR INC41 citations92
US6699866B2Mar 2, 2004
Thiazole and other heterocyclic ligands for mammalian dopamine, muscarinic and serotonin receptors and transporters, and methods of use thereof
SEPRACOR INC17 citations92
US6677332B1Jan 13, 2004
Heterocyclic analgesic compounds and methods of use thereof
SEPRACOR INC22 citations92
US6645980B1Nov 11, 2003
Heterocyclic analgesic compounds and methods of use thereof
SEPRACOR INC46 citations92
US6207679B1Mar 27, 2001
Antimicrobial agents uses and compositions related thereto
SEPRACOR INC54 citations92
US6172084B1Jan 9, 2001
Quinoline-indole antimicrobial agents, uses and compositions related thereto
SEPRACOR INC50 citations92
US6376670B1Apr 23, 2002
Quinoline-indole antimicrobial agents, uses and compositions related thereto
SEPRACOR INC35 citations91
US7517892B2Apr 14, 2009
Ligands for monoamine receptors and transporters, and methods of use thereof
SEPRACOR INC8 citations84
US6635661B2Oct 21, 2003
Heterocyclic analgesic compounds and methods of use thereof
SEPRACOR INC16 citations84
US6872716B2Mar 29, 2005
Antipsychotic sulfonamide-heterocycles, and methods of use thereof
SEPRACOR INC15 citations83
US6103905AAug 15, 2000
Quinoline-indole antimicrobial agents, uses and compositions related thereto
SEPRACOR INC17 citations83
US6548637B1Apr 15, 2003
Ligands for opioid receptors
SEPRACOR INC17 citations79
US6476050B2Nov 5, 2002
3-substituted piperidines comprising urea functionality, and methods of use thereof
SEPRACOR INC8 citations74
US6177464B1Jan 23, 2001
Ring opening metathesis of alkenes
SEPRACOR INC6 citations74
US7129228B2Oct 31, 2006
Heterocyclic analgesic compounds and methods of use thereof
SEPRACOR INC9 citations73
US6703383B2Mar 9, 2004
Antipsychotic sulfonamide-heterocycles, and methods of use thereof
SEPRACOR INC12 citations73
US6703508B2Mar 9, 2004
Methods for the stereoselective synthesis of substituted piperidines
SEPRACOR INC8 citations72
US7361666B2Apr 22, 2008
Heterocyclic analgesic compounds and methods of use thereof
SEPRACOR INC5 citations63
US7816375B2Oct 19, 2010
Ligands for monoamine receptors and transporters, and methods of use thereof
SEPRACOR INC4 citations62
US7087623B2Aug 8, 2006
Thiazole and other heterocyclic ligands for mammalian dopamine, muscarinic and serotonin receptors and transporters, and methods of use thereof
SEPRACOR INC2 citations62
US7030122B2Apr 18, 2006
1,4-disubstituted piperazine ligands for neurotransmitter receptors
SEPRACOR INC5 citations62
US7446115B2Nov 4, 2008
Peptidomimetic ligands for cellular receptors and ion channels
SEPRACOR INC0 citations52
US6946477B2Sep 20, 2005
3-Substituted piperidines comprising urea functionality, and methods of use thereof
SEPRACOR INC0 citations52
US6486324B2Nov 26, 2002
Ring opening metathesis of alkenes
SEPRACOR INC1 citations52
US7692019B2Apr 6, 2010
Methods for the stereoselective synthesis of substituted piperidines
SEPRACOR INC0 citations51
US7005524B2Feb 28, 2006
Methods for the stereoselective synthesis of substituted piperidines
SEPRACOR INC0 citations51
PFIZER
15 patentsUS5506233AApr 9, 1996
Desosamino derivatives of macrolides as immunosuppressants and antifungal agents
PFIZER26 citations92
US4512982AApr 23, 1985
9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
PFIZER48 citations92
US4465674AAug 14, 1984
Azahomoerythromycin D derivative and intermediates therefor
PFIZER33 citations92
US4518590AMay 21, 1985
9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
PFIZER22 citations82
US4382086AMay 3, 1983
9-Dihydro-11,12-ketal derivatives of erythromycin A and epi-erythromycin A
PFIZER18 citations82
US5359060AOct 25, 1994
Phosponated derivatives of macrolides
PFIZER8 citations74
US4857641AAug 15, 1989
C.12 modified erythromycin A derivatives
PFIZER7 citations74
US6756388B1Jun 29, 2004
Benzothiophenes and related compounds as estrogen agonists
PFIZER11 citations71
US4835141AMay 30, 1989
Neutral macrolide antibiotics from Streptomyces
PFIZER3 citations63
US4363803ADec 14, 1982
3",4"-Oxyallylene erythromycin and oleandomycin, composition and method of use
PFIZER3 citations63
US5563135AOct 8, 1996
Desosamino derivatives of macrolides
PFIZER3 citations62
US5064855ANov 12, 1991
Acid polycyclic ether antibiotic
PFIZER2 citations60
US4956283ASep 11, 1990
Process for preparing macrolide antibiotics by culturing streptomyces hirsutus ATCC 53513
PFIZER1 citations52
US4413119ANov 1, 1983
Semi-synthetic macrolides
PFIZER1 citations52
US4920050AApr 24, 1990
Acidic polycyclic ether antibiotic
PFIZER0 citations49