Inventor
JOHNS BRIAN A
US24 patents
⚠️ This page may combine multiple inventors who share the name “JOHNS BRIAN A”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
SMITHKLINE BEECHAM CORP
17 patentsUS6962914B2Nov 8, 2005
Pyrazolopyridinyl pyridine and pyrimidine therapeutic compounds
SMITHKLINE BEECHAM CORP22 citations92
US6919352B2Jul 19, 2005
Pyrazolopyridinyl pyridine and pyrimidine therapeutic compounds
SMITHKLINE BEECHAM CORP25 citations91
US7304068B2Dec 4, 2007
Substituted pyrazolo [1,5-A] pyrimidinyls and pharmaceutical uses therefore
SMITHKLINE BEECHAM CORP14 citations83
US7186714B2Mar 6, 2007
Imidazo[1,2-α]pyridine derivatives for the prophylaxis and treatment of herpes viral infections
SMITHKLINE BEECHAM CORP10 citations83
US7141569B2Nov 28, 2006
Antiviral pyrazolopyridine compounds
SMITHKLINE BEECHAM CORP9 citations73
US7030134B2Apr 18, 2006
Pyrazolopyridinyl pyridine and pyrimidine therapeutic compounds
SMITHKLINE BEECHAM CORP9 citations73
US7109209B2Sep 19, 2006
Pyrazolopyridines, process for their preparation and use as therapeutic compounds
SMITHKLINE BEECHAM CORP8 citations72
US7034030B2Apr 25, 2006
Pyralopyridines, process for their preparation and use as therapeutic compounds
SMITHKLINE BEECHAM CORP6 citations72
US7812016B2Oct 12, 2010
Naphthyridine integrase inhibitors
SMITHKLINE BEECHAM CORP4 citations62
US7244740B2Jul 17, 2007
Imidazo-pyridine derivatives for use in the treatment of herpes viral infection
SMITHKLINE BEECHAM CORP6 citations62
US7199120B2Apr 3, 2007
Pyrazolo-pyridine derivatives as antiherpes agents
SMITHKLINE BEECHAM CORP5 citations62
US7153863B2Dec 26, 2006
Therapeutic compounds based on pyrazolopyridline derivatives
SMITHKLINE BEECHAM CORP4 citations61
US7087618B2Aug 8, 2006
Pyrazolopyridinyl pyrimidine therapeutic compounds
SMITHKLINE BEECHAM CORP3 citations61
US7153855B2Dec 26, 2006
Pyrazolopyridinyl pyrimidine therapeutic compounds
SMITHKLINE BEECHAM CORP4 citations58
US7160897B2Jan 9, 2007
Therapeutic compounds
SMITHKLINE BEECHAM CORP0 citations51
US7163940B2Jan 16, 2007
Pyrazolopyridinyl pyrimidine therapeutic compounds
SMITHKLINE BEECHAM CORP1 citations47
US7247626B2Jul 24, 2007
Pyrazolopyrimidine derivatives and pharmaceutical compositions containing them
SMITHKLINE BEECHAM CORP0 citations41
SHIONOGI & CO
6 patentsUS8778943B2Jul 15, 2014
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-α]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides
SHIONOGI & CO30 citations95
US9051337B2Jun 9, 2015
Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides
SHIONOGI & CO27 citations92
US10927129B2Feb 23, 2021
N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity
SHIONOGI & CO3 citations83
US9273065B2Mar 1, 2016
Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors
SHIONOGI & CO3 citations83
US11267823B2Mar 8, 2022
Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1′,2′:4,5]pyrazino[1,2-a]pyrrolo[1,2-c]pyrimidines having HIV integrase inhibitory activity
SHIONOGI & CO2 citations72
US8691823B2Apr 8, 2014
Prodrugs of (4aS, 13ar)-N-[(2,4-difluorophenyl)methyl]-10-hydroxy-9-11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1H-pyrido[1,2-a]pyrrolo[1′,2′:3:4]imidazo[1,2-d]pyrazine-8-carboxamide and their use in the treatment of HIV infection
SHIONOGI & CO0 citations49