Inventor

JONAS ROCHUS

DE46 patents

Patents

46 patents

US5869516AFeb 9, 1999

Aminothiophene carboxylic acid amides and the use thereof as phosphodiesterase inhibitors

MERCK PATENT GMBH33 citations92

US6130223AOct 10, 2000

Thienopyrimidine with phosphodiesterase V inhibiting effect

MERCK PATENT GMBH32 citations92

US5434149AJul 18, 1995

Thiadiazinones

MERCK PATENT GMBH20 citations92

US4916128AApr 10, 1990

Thiadiazinones

MERCK PATENT GMBH29 citations91

US4258062AMar 24, 1981

Phenoxy-amino-propanols

MERCK PATENT GMBH40 citations91

US6787548B1Sep 7, 2004

Thienopyrimidines as phosphodiesterase inhibitors

MERCK PATENT GMBH15 citations84

US7491742B2Feb 17, 2009

Imidazole derivatives as phosphodiesterase VII inhibitors

MERCK PATENT GMBH13 citations83

US4171370AOct 16, 1979

Phenoxy-amino-propanols

MERCK PATENT GMBH24 citations81

US4590180AMay 20, 1986

Use of adenosine derivatives as psychopharmacological agents

MERCK PATENT GMBH19 citations80

US4016281AApr 5, 1977

Tetralone and indanone compounds

MERCK PATENT GMBH19 citations76

US6777419B1Aug 17, 2004

Pyrazolo [4,3-d]pyrimidines

MERCK PATENT GMBH12 citations74

US6495557B1Dec 17, 2002

Condensed thienopyrimidines with phosphodiesterase-v inhibiting action

MERCK PATENT GMBH10 citations73

US6420368B1Jul 16, 2002

Thienopyrimidines

MERCK PATENT GMBH7 citations73

US5747489AMay 5, 1998

Arylalkyl-thiadiazinones

MERCK PATENT GMBH11 citations73

US5276027AJan 4, 1994

Thiadiazinones

MERCK PATENT GMBH11 citations73

US3989833ANov 2, 1976

Pharmaceutical compositions containing adenine derivatives

MERCK PATENT GMBH8 citations73

US5026705AJun 25, 1991

Benzimidazolylpyridazinones

MERCK PATENT GMBH13 citations72

US4923869AMay 8, 1990

Benzimidazolylpyridazinones

MERCK PATENT GMBH12 citations72

US4575505AMar 11, 1986

Pharmaceutical compositions containing 2-aryltetraazaindenes for treating ulcers or cardiac insufficiency or blood pressure abnormalities

MERCK PATENT GMBH5 citations72

US4477454AOct 16, 1984

2-Aryltetraazaindenes for treating cardiac insufficiency

MERCK PATENT GMBH7 citations72

US4260628AApr 7, 1981

2-Guanidinomethyl-indolines

MERCK PATENT GMBH9 citations71

US7259168B2Aug 21, 2007

2-Aminoalkyl-thieno[2,3-d]pyrimidines

MERCK PATENT GMBH2 citations63

US6780867B2Aug 24, 2004

Thienopyrimidines

MERCK PATENT GMBH5 citations63

US6696446B1Feb 24, 2004

Benzoylpyridazines, their preparation and use

MERCK PATENT GMBH3 citations63

US6531473B2Mar 11, 2003

Method of treatment using arylalkylpyridazinones

MERCK PATENT GMBH4 citations63

US5137885AAug 11, 1992

Thiadiazinones

MERCK PATENT GMBH5 citations63

US4616090AOct 7, 1986

2-arylimidazopyridines intermediates

MERCK PATENT GMBH3 citations63

US6495554B2Dec 17, 2002

Thienopyrimidines

MERCK PATENT GMBH2 citations62

US6025354AFeb 15, 2000

Arylalkyl-thiadiazinones

MERCK PATENT GMBH3 citations62

US4070461AJan 24, 1978

Biphenylyl ethers

MERCK PATENT GMBH2 citations62

US4060609ANov 29, 1977

Biphenylyl ethers and method of use

MERCK PATENT GMBH2 citations62

US5104881AApr 14, 1992

2-arylimidazopyridines

MERCK PATENT GMBH3 citations61

US4654344AMar 31, 1987

Pharmaceutical compositions for treating ulcers containing 2-aryltetraazaindenes

MERCK PATENT GMBH1 citations61

US3980797ASep 14, 1976

Hexahydro-diazepino-indole derivatives

MERCK PATENT GMBH6 citations60

US5206363AApr 27, 1993

Process for the resolution of enantiomers of 5-heteroaryl-1,3,4-thiadiazinones

MERCK PATENT GMBH4 citations54

US6376493B1Apr 23, 2002

Benzoylpyridazines

MERCK PATENT GMBH1 citations52

US5378702AJan 3, 1995

Thiadizinones

MERCK PATENT GMBH1 citations52

US4070357AJan 24, 1978

Process for the preparation of indoline derivatives

MERCK PATENT GMBH0 citations51

US7060823B2Jun 13, 2006

5-aminoalkyl-pyrazolo[4,3-d]pyrimidines with a phosphodiesterase v-inhibiting effect

MERCK PATENT GMBH0 citations42

JONAS ROCHUS

Patents

4-(arylaminomethylene)-2,4-dihydro-3-pyrazolones

Arylalkylpyridazinones

Arylalkyl diazinones

Imidazole compounds used as phosphodiesterase VII inhibitors

Pyrrole derivatives as phosphodiesterase VII inhibitors

Isoxazole derivatives to be used as phosphodiesterase VII inhibitors

Arylalkanoylpyridazines

Aminothiophene carboxylic acid amides and the use thereof as phosphodiesterase inhibitors

Thienopyrimidine with phosphodiesterase V inhibiting effect

Thiadiazinones

Thiadiazinones

Phenoxy-amino-propanols

Thienopyrimidines as phosphodiesterase inhibitors

Imidazole derivatives as phosphodiesterase VII inhibitors

Phenoxy-amino-propanols

Use of adenosine derivatives as psychopharmacological agents

Tetralone and indanone compounds

Pyrazolo [4,3-d]pyrimidines

Condensed thienopyrimidines with phosphodiesterase-v inhibiting action

Thienopyrimidines

Arylalkyl-thiadiazinones

Thiadiazinones

Pharmaceutical compositions containing adenine derivatives

Benzimidazolylpyridazinones

Benzimidazolylpyridazinones

Pharmaceutical compositions containing 2-aryltetraazaindenes for treating ulcers or cardiac insufficiency or blood pressure abnormalities

2-Aryltetraazaindenes for treating cardiac insufficiency

2-Guanidinomethyl-indolines

2-Aminoalkyl-thieno[2,3-d]pyrimidines

Thienopyrimidines

Benzoylpyridazines, their preparation and use

Method of treatment using arylalkylpyridazinones

Thiadiazinones

2-arylimidazopyridines intermediates

Thienopyrimidines

Arylalkyl-thiadiazinones

Biphenylyl ethers

Biphenylyl ethers and method of use

2-arylimidazopyridines

Pharmaceutical compositions for treating ulcers containing 2-aryltetraazaindenes

Hexahydro-diazepino-indole derivatives

Process for the resolution of enantiomers of 5-heteroaryl-1,3,4-thiadiazinones

Benzoylpyridazines

Thiadizinones

Process for the preparation of indoline derivatives

5-aminoalkyl-pyrazolo[4,3-d]pyrimidines with a phosphodiesterase v-inhibiting effect