Inventor
QUEROLLE OLIVIER ALEXIS GEORGES
FR33 patents
⚠️ This page may combine multiple inventors who share the name “QUEROLLE OLIVIER ALEXIS GEORGES”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
JANSSEN PHARMACEUTICA NV
21 patentsUS11396517B1Jul 26, 2022
Exo-aza spiro inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV6 citations71
US10611778B2Apr 7, 2020
Fused bicyclic inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV3 citations71
US11530226B2Dec 20, 2022
Azepane inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV1 citations60
US11220517B2Jan 11, 2022
Spiro bicyclic inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV1 citations60
US10975100B2Apr 13, 2021
Fused bicyclic inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV1 citations60
US10745409B2Aug 18, 2020
Azepane inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV1 citations60
US11267804B2Mar 8, 2022
(R)-8-(1-((3-fluorophenyl)amino)ethyl)-N-(2-hydroxyethyl)-2-morpholinoquinoxaline-6-carboxamide for inhibiting phosphoinositide-3-kinase activity
JANSSEN PHARMACEUTICA NV0 citations59
US12473295B2Nov 18, 2025
Substituted straight chain spiro derivatives
JANSSEN PHARMACEUTICA NV0 citations54
US12084462B2Sep 10, 2024
Spiro bicyclic inhibitors of menin-MLL interaction
JANSSEN PHARMACEUTICA NV0 citations50
US11236084B2Feb 1, 2022
Substituted azaindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11186589B2Nov 30, 2021
Cyanoindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11180487B2Nov 23, 2021
Substituted cyanoindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11136311B2Oct 5, 2021
Heteroaromatic derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US11001569B2May 11, 2021
6-membered heteroaromatic substituted cyanoindoline derivatives as NIK inhibitors
JANSSEN PHARMACEUTICA NV0 citations50
US10526316B2Jan 7, 2020
Quinoxaline and pyridopyrazine derivatives as PI3Kβ inhibitors
JANSSEN PHARMACEUTICA NV0 citations49
US10894793B2Jan 19, 2021
Bicyclic pyridine, pyrazine, and pyrimidine derivatives as PI3K beta inhibitors
JANSSEN PHARMACEUTICA NV0 citations48
US11542247B2Jan 3, 2023
Bi-heteroaryl substitute 1,4-benzodiazepines and uses thereof for the treatment of cancer
JANSSEN PHARMACEUTICA NV0 citations47
US11130751B2Sep 28, 2021
Quinoxaline and pyridopyrazine derivatives as PI3K-beta inhibitors
JANSSEN PHARMACEUTICA NV0 citations47
US11155555B2Oct 26, 2021
Compounds
JANSSEN PHARMACEUTICA NV0 citations45
US10202387B2Feb 12, 2019
Heterocyclyl linked imidazopyridazine derivatives as PI3KB inhibitors
JANSSEN PHARMACEUTICA NV0 citations39
US10087187B2Oct 2, 2018
Imidazopyridazine derivatives as PI3KB inhibitors
JANSSEN PHARMACEUTICA NV0 citations39
ASTEX THERAPEUTICS LTD
12 patentsUS9447098B2Sep 20, 2016
Pteridines as FGFR inhibitors
ASTEX THERAPEUTICS LTD35 citations94
US9309242B2Apr 12, 2016
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD26 citations94
US9303029B2Apr 5, 2016
Substituted quinoxalines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD25 citations94
US9464071B2Oct 11, 2016
Pyrazolyl quinoxaline kinase inhibitors
ASTEX THERAPEUTICS LTD24 citations93
US9303030B2Apr 5, 2016
Compounds
ASTEX THERAPEUTICS LTD26 citations93
US9850228B2Dec 26, 2017
Pyrazolyl quinoxaline kinase inhibitors
ASTEX THERAPEUTICS LTD17 citations91
US10052320B2Aug 21, 2018
Substituted quinoxalines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD11 citations84
US10045982B2Aug 14, 2018
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors
ASTEX THERAPEUTICS LTD11 citations84
US9493426B2Nov 15, 2016
Quinazolinone derivatives useful as FGFR kinase modulators
ASTEX THERAPEUTICS LTD20 citations84
US10519137B2Dec 31, 2019
Pyrazolyl quinoxaline kinase inhibitors
ASTEX THERAPEUTICS LTD6 citations83
US9737544B2Aug 22, 2017
Compounds
ASTEX THERAPEUTICS LTD15 citations83
US10272087B2Apr 30, 2019
Pteridines as FGFR inhibitors
ASTEX THERAPEUTICS LTD5 citations73