Inventor
TRYBULSKI EUGENE J
50 patents
⚠️ This page may combine multiple inventors who share the name “TRYBULSKI EUGENE J”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
HOFFMANN LA ROCHE
26 patentsUS4481142ANov 6, 1984
Pyrimido-2-benzazepines
HOFFMANN LA ROCHE25 citations82
US4469633ASep 4, 1984
N-oxides of 5-oxo-1-phenyl-2-benzazepines
HOFFMANN LA ROCHE23 citations82
US4318854AMar 9, 1982
Intermediates in the production of 2-benzazepines
HOFFMANN LA ROCHE10 citations74
US4436662AMar 13, 1984
Pyrrolo[3,4-d][2]benzazepinones
HOFFMANN LA ROCHE2 citations63
US4431823AFeb 14, 1984
1H-Pyrrole-3-carbonitrile-4(2-benzoyl)phenyl derivatives as intermediates for pyrrolo[3,4-D][2]benzazepines
HOFFMANN LA ROCHE2 citations63
US4354973AOct 19, 1982
Pyrrolo[3,4-d][2]benzazepines
HOFFMANN LA ROCHE2 citations63
US4547581AOct 15, 1985
Pyrimido-2-benzazepines and intermediates in their preparation
HOFFMANN LA ROCHE4 citations62
US4549988AOct 29, 1985
3H-2-Benzazepines
HOFFMANN LA ROCHE1 citations52
US4548750AOct 22, 1985
Pyrimido[4,5-d][2]benzazepines useful as sedatives and anxiolytic agents
HOFFMANN LA ROCHE1 citations52
US4546183AOct 8, 1985
Pyrimido-2-benzazepines
HOFFMANN LA ROCHE0 citations52
US4460781AJul 17, 1984
4-(2-Benzoylphenyl-1-pyazole and 4-(2-benzoylphenyl)-1-pyrazoline derivatives
HOFFMANN LA ROCHE0 citations52
US4428878AJan 31, 1984
Pyrrolo[3,4-d][2]benzazepines
HOFFMANN LA ROCHE0 citations52
US4428879AJan 31, 1984
Pyrrolo[3,4,-d][2]benzazepines
HOFFMANN LA ROCHE0 citations52
US4427589AJan 24, 1984
Pyrimido[4,5-d][2]benzazepines
HOFFMANN LA ROCHE1 citations52
US4409390AOct 11, 1983
Pyrrolo[3,4-D][2]Benzazepines
HOFFMANN LA ROCHE1 citations52
US4405518ASep 20, 1983
Pyrrolo[3,4-d] [2] benzazepines
HOFFMANN LA ROCHE0 citations52
US4402876ASep 6, 1983
Production of 2-benzazepines
HOFFMANN LA ROCHE0 citations52
US4394311AJul 19, 1983
Production of 2-benzazepines
HOFFMANN LA ROCHE0 citations52
US4388239AJun 14, 1983
Production of 1-halophenyl and 1-phenyl-3,4-dihydro-5H-2-benzazepine-5-ones
HOFFMANN LA ROCHE0 citations52
US4379765AApr 12, 1983
Pyrazolobenzazepines
HOFFMANN LA ROCHE1 citations52
US4379090AApr 5, 1983
Process for the preparation of 1-(phenyl and halophenyl)-3,4-dihydro-4-[(dimethylamino)methylene]5H-2-benzazepin-5-one-2-oxides
HOFFMANN LA ROCHE0 citations52
US4299971ANov 10, 1981
Triazolobenzazepines
HOFFMANN LA ROCHE0 citations52
US4260772AApr 7, 1981
Intermediates for triazolobenzazepines
HOFFMANN LA ROCHE0 citations52
US4260773AApr 7, 1981
Intermediates for triazolobenzazepines
HOFFMANN LA ROCHE0 citations52
US4259503AMar 31, 1981
Triazole intermediates for triazolobenzazepines
HOFFMANN LA ROCHE0 citations52
US4243589AJan 6, 1981
Triazolobenzazepines and processes for their production
HOFFMANN LA ROCHE0 citations52
AMERICAN CYANAMID CO
12 patentsUS5128483AJul 7, 1992
Dibromovinyl and acetylene-1-pyrrolidinecarboxylic acid intermediates
AMERICAN CYANAMID CO9 citations73
US5001142AMar 19, 1991
1-substituted-2-(3-amino-1-propynyl)pyrrolidine derivatives
AMERICAN CYANAMID CO7 citations73
US4990520AFeb 5, 1991
2-,4- or 5-substituted thiazole derivatives
AMERICAN CYANAMID CO11 citations73
US4937235AJun 26, 1990
3- or 4-substituted oxotremorine derivatives
AMERICAN CYANAMID CO8 citations73
US5089518AFeb 18, 1992
3- or 4-substituted oxotremorine derivatives and a method of treating cholinergic dysfunction therewith
AMERICAN CYANAMID CO3 citations62
US5025099AJun 18, 1991
(3-amino-1-propynyl)methylthiothiophene derivatives
AMERICAN CYANAMID CO2 citations62
US5637731AJun 10, 1997
Substituted oxotremorine derivatives
AMERICAN CYANAMID CO1 citations51
US5550257AAug 27, 1996
Substituted oxotremorine derivatives
AMERICAN CYANAMID CO1 citations51
US5451685ASep 19, 1995
Substituted oxotremorine derivatives
AMERICAN CYANAMID CO0 citations51
US5356885AOct 18, 1994
Substituted oxotremorine derivatives and pharmaceutical use thereof
AMERICAN CYANAMID CO0 citations51
US4952600AAug 28, 1990
3- or 4-substituted oxotremorine derivatives and a method of treating central chloinergic dsyfunction therewith
AMERICAN CYANAMID CO1 citations51
US5346910ASep 13, 1994
Maleimide derivatives of oxotremorine
AMERICAN CYANAMID CO0 citations41
WYETH CORP
8 patentsUS6903091B2Jun 7, 2005
Biphenyl vasopressin agonists
WYETH CORP26 citations92
US6511974B1Jan 28, 2003
Tricyclic vasopressin agonists
WYETH CORP42 citations92
US7138393B2Nov 21, 2006
Biologically active vasopressin agonist metabolites
WYETH CORP18 citations83
US7678787B2Mar 16, 2010
Pyrrolobenzodiazepine pyridine carboxamides and derivatives as follicle-stimulating hormone receptor antagonists
WYETH CORP15 citations79
US7465722B2Dec 16, 2008
Biphenyl vasopressin agonists
WYETH CORP3 citations62
US7223752B2May 29, 2007
Biphenyl vasopressin agonists
WYETH CORP0 citations51
US7585871B2Sep 8, 2009
Phenanthridine carbonyl phenols
WYETH CORP0 citations37
US7601856B2Oct 13, 2009
Benzofurans as potassium ion channel modulators
WYETH CORP0 citations36
AMERICAN HOME PROD
3 patentsUS6235900B1May 22, 2001
Tricyclic pyridine N-oxides vasopressin agonists
AMERICAN HOME PROD32 citations92
US5880122AMar 9, 1999
3-Carboxamide derivatives of 5H-pyrrolo 2,1-c! 1,4!-benzodiazepines
AMERICAN HOME PROD46 citations92
US5932745AAug 3, 1999
Process for converting propargylic amine-N-oxides to enaminones
AMERICAN HOME PROD27 citations86