Inventor
DUSZA JOHN P
US51 patents
⚠️ This page may combine multiple inventors who share the name “DUSZA JOHN P”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.
AMERICAN CYANAMID CO
44 patentsUS5753648AMay 19, 1998
Tricyclic benzazepine vasopressin antagonists
AMERICAN CYANAMID CO70 citations96
US5536718AJul 16, 1996
Tricyclic benzazepine vasopressin antagonists
AMERICAN CYANAMID CO86 citations96
US4654343AMar 31, 1987
N-substituted-N[3-(1,2,4-triazolo[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureas
AMERICAN CYANAMID CO60 citations96
US4626538ADec 2, 1986
[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO106 citations96
US4521422AJun 4, 1985
Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones
AMERICAN CYANAMID CO71 citations96
US4178449ADec 11, 1979
Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines
AMERICAN CYANAMID CO62 citations96
US6399621B1Jun 4, 2002
N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1, 5-α]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto
AMERICAN CYANAMID CO78 citations95
US4876252AOct 24, 1989
4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines
AMERICAN CYANAMID CO89 citations95
US4788195ANov 29, 1988
4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines
AMERICAN CYANAMID CO104 citations95
US5538977AJul 23, 1996
3-Substituted-7-[3-(imidazol-1-yl)phenyl]-pyrazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO19 citations93
US4900836AFeb 13, 1990
(3-amino-1H-pyrazol-4-yl) (aryl)methanones
AMERICAN CYANAMID CO38 citations93
US4654347AMar 31, 1987
Aryl and heteroaryl[[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]methanones
AMERICAN CYANAMID CO43 citations93
US4281000AJul 28, 1981
Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents
AMERICAN CYANAMID CO30 citations93
US5700796ADec 23, 1997
Tricyclic benzazepine vasopressin antagonists
AMERICAN CYANAMID CO20 citations92
US5169850ADec 8, 1992
N-(dialkylamino)methylene)-substituted pyrazolo(1,5-a)-pyrimidine-3-carboxamides and N-(dialkylamino)methylene-substituted-4,5-dihydropyrazolo-(1,5-a)-pyrimidine-3-carboxamides
AMERICAN CYANAMID CO30 citations92
US4847256AJul 11, 1989
4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines
AMERICAN CYANAMID CO34 citations92
US4576943AMar 18, 1986
Pyrazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO30 citations92
US4209621AJun 24, 1980
(Substituted-phenyl)-1,2,4-triazolo[4,3-a]-pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO47 citations90
US4582833AApr 15, 1986
2-(substituted-1-piperazinyl)[1,2,4]triazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO19 citations82
US4421753ADec 20, 1983
1-(5-Amino-4H-1,2,4-triazol-3-yl)-4-substituted-piperazines
AMERICAN CYANAMID CO26 citations82
US4260756AApr 7, 1981
6- And 8-heteroaryl-1,2,4-triazolo[4,3-b]pyridazines
AMERICAN CYANAMID CO26 citations82
US4236005ANov 25, 1980
Imidazo[1,5-a]pyrimidines
AMERICAN CYANAMID CO23 citations82
US5612334AMar 18, 1997
Tricyclic benzazepine vasopressin antagonists
AMERICAN CYANAMID CO12 citations74
US4980472ADec 25, 1990
Method of making (3-amino-1H-pyrazol-4-yl) (aryl)methanones
AMERICAN CYANAMID CO8 citations74
US4451479AMay 29, 1984
Therapeutically active 3-amino-1-halogenated phenyl-2-pyrazolines and their C4 and C5 analogs
AMERICAN CYANAMID CO8 citations74
US4444774AApr 24, 1984
7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidines
AMERICAN CYANAMID CO13 citations74
US4432991AFeb 21, 1984
Therapeutically active 3-amino-1-phenyl(and substituted phenyl)-2-pyrazolines
AMERICAN CYANAMID CO10 citations74
US4347251AAug 31, 1982
Novel 3-substituted amino-1-substituted heteroaryl-2-pyrazolines
AMERICAN CYANAMID CO12 citations74
US4260767AApr 7, 1981
2-Pyridylhydrazides
AMERICAN CYANAMID CO8 citations74
US5059691AOct 22, 1991
N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides
AMERICAN CYANAMID CO8 citations73
US5037980AAug 6, 1991
Phenyl imidazo[1,2-a]pyrimidines
AMERICAN CYANAMID CO2 citations63
US4551530ANov 5, 1985
Pyridyl imidazo[1,2-a]pyrimidines
AMERICAN CYANAMID CO5 citations63
US4448973AMay 15, 1984
Therapeutically active 3-substituted amino-1-phenyl and substituted phenyl-2-pyrazolines
AMERICAN CYANAMID CO3 citations63
US4393217AJul 12, 1983
Substituted phenyl-5-aminopyrazoles
AMERICAN CYANAMID CO3 citations63
US4376122AMar 8, 1983
Novel 3-substituted amino-1-heteroaryl-2-pyrazolines
AMERICAN CYANAMID CO4 citations63
US4374988AFeb 22, 1983
4-Heteroarylimidazo-[1,5-A]pyrimidines
AMERICAN CYANAMID CO6 citations63
US4888345ADec 19, 1989
4,8-disubstituted-1,2-dihydro and 1,2,3,4-tetrahydroimidazo-[1,5-a] pyrimidines
AMERICAN CYANAMID CO2 citations62
US4767765AAug 30, 1988
N-substituted-N-[3-(1,2,4-triazolo-[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureas
AMERICAN CYANAMID CO4 citations62
US5059709AOct 22, 1991
Process for the synthesis of α-[(dialkylamino)substituted-methylene]-β-oxo-(substituted)propanentriles
AMERICAN CYANAMID CO2 citations59
US4447442AMay 8, 1984
3-Trifluoroacetylamino-1-aryl-2-pyrazolines
AMERICAN CYANAMID CO4 citations57
US4892873AJan 9, 1990
N-substituted -N-(3-(1,2,4-triazolo-(4,3-b)pyridazin-6-yl)phenyl)alkanamides, carbamates and ureas
AMERICAN CYANAMID CO1 citations52
US4622401ANov 11, 1986
Heterocyclic substituted-amino-pyrazolines
AMERICAN CYANAMID CO0 citations52
US4360680ANov 23, 1982
Therapeutically active 3-amino-1-phenyl and substituted phenyl-2-pyrazolines
AMERICAN CYANAMID CO1 citations52
US4348527ASep 7, 1982
3-Trifluoroacetyl amino-1-aryl-2-pyrazolines
AMERICAN CYANAMID CO1 citations52
WYETH CORP
6 patentsUS6903091B2Jun 7, 2005
Biphenyl vasopressin agonists
WYETH CORP26 citations92
US6511974B1Jan 28, 2003
Tricyclic vasopressin agonists
WYETH CORP42 citations92
US7053083B2May 30, 2006
Cyclohexylphenyl vasopressin agonists
WYETH CORP23 citations91
US7465722B2Dec 16, 2008
Biphenyl vasopressin agonists
WYETH CORP3 citations62
US7329653B2Feb 12, 2008
Cyclohexylphenyl vasopressin agonists
WYETH CORP0 citations51
US7223752B2May 29, 2007
Biphenyl vasopressin agonists
WYETH CORP0 citations51
Showing the top 50 of 51 patents by PatentIndex Score.