P

Inventor

DUSZA JOHN P

US51 patents
⚠️ This page may combine multiple inventors who share the name “DUSZA JOHN P”. Patents are grouped by organization below to help distinguish them — per-person disambiguation is on the roadmap.

AMERICAN CYANAMID CO

44 patents
US5753648AMay 19, 1998

Tricyclic benzazepine vasopressin antagonists

AMERICAN CYANAMID CO70 citations96
US5536718AJul 16, 1996

Tricyclic benzazepine vasopressin antagonists

AMERICAN CYANAMID CO86 citations96
US4654343AMar 31, 1987

N-substituted-N[3-(1,2,4-triazolo[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureas

AMERICAN CYANAMID CO60 citations96
US4626538ADec 2, 1986

[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines

AMERICAN CYANAMID CO106 citations96
US4521422AJun 4, 1985

Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones

AMERICAN CYANAMID CO71 citations96
US4178449ADec 11, 1979

Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines

AMERICAN CYANAMID CO62 citations96
US6399621B1Jun 4, 2002

N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1, 5-α]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto

AMERICAN CYANAMID CO78 citations95
US4876252AOct 24, 1989

4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines

AMERICAN CYANAMID CO89 citations95
US4788195ANov 29, 1988

4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines

AMERICAN CYANAMID CO104 citations95
US5538977AJul 23, 1996

3-Substituted-7-[3-(imidazol-1-yl)phenyl]-pyrazolo[1,5-a]pyrimidines

AMERICAN CYANAMID CO19 citations93
US4900836AFeb 13, 1990

(3-amino-1H-pyrazol-4-yl) (aryl)methanones

AMERICAN CYANAMID CO38 citations93
US4654347AMar 31, 1987

Aryl and heteroaryl[[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]methanones

AMERICAN CYANAMID CO43 citations93
US4281000AJul 28, 1981

Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents

AMERICAN CYANAMID CO30 citations93
US5700796ADec 23, 1997

Tricyclic benzazepine vasopressin antagonists

AMERICAN CYANAMID CO20 citations92
US5169850ADec 8, 1992

N-(dialkylamino)methylene)-substituted pyrazolo(1,5-a)-pyrimidine-3-carboxamides and N-(dialkylamino)methylene-substituted-4,5-dihydropyrazolo-(1,5-a)-pyrimidine-3-carboxamides

AMERICAN CYANAMID CO30 citations92
US4847256AJul 11, 1989

4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines

AMERICAN CYANAMID CO34 citations92
US4576943AMar 18, 1986

Pyrazolo[1,5-a]pyrimidines

AMERICAN CYANAMID CO30 citations92
US4209621AJun 24, 1980

(Substituted-phenyl)-1,2,4-triazolo[4,3-a]-pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-a]pyrimidines

AMERICAN CYANAMID CO47 citations90
US4582833AApr 15, 1986

2-(substituted-1-piperazinyl)[1,2,4]triazolo[1,5-a]pyrimidines

AMERICAN CYANAMID CO19 citations82
US4421753ADec 20, 1983

1-(5-Amino-4H-1,2,4-triazol-3-yl)-4-substituted-piperazines

AMERICAN CYANAMID CO26 citations82
US4260756AApr 7, 1981

6- And 8-heteroaryl-1,2,4-triazolo[4,3-b]pyridazines

AMERICAN CYANAMID CO26 citations82
US4236005ANov 25, 1980

Imidazo[1,5-a]pyrimidines

AMERICAN CYANAMID CO23 citations82
US5612334AMar 18, 1997

Tricyclic benzazepine vasopressin antagonists

AMERICAN CYANAMID CO12 citations74
US4980472ADec 25, 1990

Method of making (3-amino-1H-pyrazol-4-yl) (aryl)methanones

AMERICAN CYANAMID CO8 citations74
US4451479AMay 29, 1984

Therapeutically active 3-amino-1-halogenated phenyl-2-pyrazolines and their C4 and C5 analogs

AMERICAN CYANAMID CO8 citations74
US4444774AApr 24, 1984

7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidines

AMERICAN CYANAMID CO13 citations74
US4432991AFeb 21, 1984

Therapeutically active 3-amino-1-phenyl(and substituted phenyl)-2-pyrazolines

AMERICAN CYANAMID CO10 citations74
US4347251AAug 31, 1982

Novel 3-substituted amino-1-substituted heteroaryl-2-pyrazolines

AMERICAN CYANAMID CO12 citations74
US4260767AApr 7, 1981

2-Pyridylhydrazides

AMERICAN CYANAMID CO8 citations74
US5059691AOct 22, 1991

N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides

AMERICAN CYANAMID CO8 citations73
US5037980AAug 6, 1991

Phenyl imidazo[1,2-a]pyrimidines

AMERICAN CYANAMID CO2 citations63
US4551530ANov 5, 1985

Pyridyl imidazo[1,2-a]pyrimidines

AMERICAN CYANAMID CO5 citations63
US4448973AMay 15, 1984

Therapeutically active 3-substituted amino-1-phenyl and substituted phenyl-2-pyrazolines

AMERICAN CYANAMID CO3 citations63
US4393217AJul 12, 1983

Substituted phenyl-5-aminopyrazoles

AMERICAN CYANAMID CO3 citations63
US4376122AMar 8, 1983

Novel 3-substituted amino-1-heteroaryl-2-pyrazolines

AMERICAN CYANAMID CO4 citations63
US4374988AFeb 22, 1983

4-Heteroarylimidazo-[1,5-A]pyrimidines

AMERICAN CYANAMID CO6 citations63
US4888345ADec 19, 1989

4,8-disubstituted-1,2-dihydro and 1,2,3,4-tetrahydroimidazo-[1,5-a] pyrimidines

AMERICAN CYANAMID CO2 citations62
US4767765AAug 30, 1988

N-substituted-N-[3-(1,2,4-triazolo-[4,3-b]pyridazin-6-yl)phenyl]alkanamides, carbamates and ureas

AMERICAN CYANAMID CO4 citations62
US5059709AOct 22, 1991

Process for the synthesis of α-[(dialkylamino)substituted-methylene]-β-oxo-(substituted)propanentriles

AMERICAN CYANAMID CO2 citations59
US4447442AMay 8, 1984

3-Trifluoroacetylamino-1-aryl-2-pyrazolines

AMERICAN CYANAMID CO4 citations57
US4892873AJan 9, 1990

N-substituted -N-(3-(1,2,4-triazolo-(4,3-b)pyridazin-6-yl)phenyl)alkanamides, carbamates and ureas

AMERICAN CYANAMID CO1 citations52
US4622401ANov 11, 1986

Heterocyclic substituted-amino-pyrazolines

AMERICAN CYANAMID CO0 citations52
US4360680ANov 23, 1982

Therapeutically active 3-amino-1-phenyl and substituted phenyl-2-pyrazolines

AMERICAN CYANAMID CO1 citations52
US4348527ASep 7, 1982

3-Trifluoroacetyl amino-1-aryl-2-pyrazolines

AMERICAN CYANAMID CO1 citations52

WYETH CORP

6 patents

Showing the top 50 of 51 patents by PatentIndex Score.